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48 in total

1. Crystallographic and kinetic investigations of the covalent complex formed by a specific tetrapeptide aldehyde and the serine protease from Streptomyces griseus.

Authors: G D Brayer; L T Delbaere; M N James; C A Bauer; R C Thompson
Journal: Proc Natl Acad Sci U S A Date: 1979-01 Impact factor: 11.205

2. Caught in the act: visualization of an intermediate in the DNA base-flipping pathway induced by HhaI methyltransferase.

Authors: John R Horton; Gary Ratner; Nilesh K Banavali; Niu Huang; Yongseok Choi; Martin A Maier; Victor E Marquez; Alexander D MacKerell; Xiaodong Cheng
Journal: Nucleic Acids Res Date: 2004-07-23 Impact factor: 16.971

3. Characterization of C-alkyl amidines as bioavailable covalent reversible inhibitors of human DDAH-1.

Authors: Matthew Lluis; Yun Wang; Arthur F Monzingo; Walter Fast; Jon D Robertus
Journal: ChemMedChem Date: 2011-01-03 Impact factor: 3.466

4. Thermodynamic framework for identifying free energy inventories of enzyme catalytic cycles.

Authors: Stephen D Fried; Steven G Boxer
Journal: Proc Natl Acad Sci U S A Date: 2013-07-09 Impact factor: 11.205

5. The far reaches of enzymology.

Authors: Jesse G Zalatan; Daniel Herschlag
Journal: Nat Chem Biol Date: 2009-08 Impact factor: 15.040

6. Testing geometrical discrimination within an enzyme active site: constrained hydrogen bonding in the ketosteroid isomerase oxyanion hole.

Authors: Paul A Sigala; Daniel A Kraut; Jose M M Caaveiro; Brandon Pybus; Eliza A Ruben; Dagmar Ringe; Gregory A Petsko; Daniel Herschlag
Journal: J Am Chem Soc Date: 2008-09-23 Impact factor: 15.419

Review 7. Enzymatic transition states, transition-state analogs, dynamics, thermodynamics, and lifetimes.

Authors: Vern L Schramm
Journal: Annu Rev Biochem Date: 2011 Impact factor: 23.643

8. Ribonuclease a: revealing structure-function relationships with semisynthesis.

Authors: J M Messmore; D N Fuchs; R T Raines
Journal: J Am Chem Soc Date: 1995-08 Impact factor: 15.419

Review 9. Transition States, analogues, and drug development.

Authors: Vern L Schramm
Journal: ACS Chem Biol Date: 2013-01-04 Impact factor: 5.100

10. Preclinical characteristics of the hepatitis C virus NS3/4A protease inhibitor ITMN-191 (R7227).

Authors: Scott D Seiwert; Steven W Andrews; Yutong Jiang; Vladimir Serebryany; Hua Tan; Karl Kossen; P T Ravi Rajagopalan; Shawn Misialek; Sarah K Stevens; Antitsa Stoycheva; Jin Hong; Sharlene R Lim; Xiaoli Qin; Robert Rieger; Kevin R Condroski; Hailong Zhang; Mary Geck Do; Christine Lemieux; Gary P Hingorani; Dylan P Hartley; John A Josey; Lin Pan; Leonid Beigelman; Lawrence M Blatt
Journal: Antimicrob Agents Chemother Date: 2008-09-29 Impact factor: 5.191