Literature DB >> 7972340

Neuropharmacology of 5-hydroxytryptamine1B/D receptor ligands.

P Chopin1, C Moret, M Briley.   

Abstract

In spite of a lack of compounds acting selectively at the 5-hydroxytryptamine (5-HT)1B and 5-HT1D receptor subtypes, by cross-relating the available data, this review attempts to tentatively assign behavioural and other in vivo correlates of these receptor subtypes. In addition, a summary of data from microdialysis studies is included to develop an integrated view. Finally, a suggestion is made as to the possible pathophysiological consequences of 5-HT1D receptor dysfunction in man.

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Year:  1994        PMID： 7972340     DOI： 10.1016/0163-7258(94)90051-5

Source DB:  PubMed          Journal:  Pharmacol Ther        ISSN： 0163-7258            Impact factor:   12.310


  11 in total

1.  5-HT(1B) receptors inhibit glutamate release from primary afferent terminals in rat medullary dorsal horn neurons.

Authors:  I-S Choi; J-H Cho; C-H An; J-K Jung; Y-K Hur; J-K Choi; I-S Jang
Journal:  Br J Pharmacol       Date:  2012-09       Impact factor: 8.739

2.  Ex vivo inhibitory effect of the 5-HT uptake blocker citalopram on 5-HT synthesis.

Authors:  C Moret; M Briley
Journal:  J Neural Transm (Vienna)       Date:  1997       Impact factor: 3.575

3.  Presynaptic inhibitory serotonin autoreceptors in the human hippocampus.

Authors:  E Schlicker; K Fink; J Zentner; M Göthert
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1996 Aug-Sep       Impact factor: 3.000

4.  Pharmacological characterizations of recombinant human 5-HT1D alpha and 5-HT1D beta receptor subtypes coupled to adenylate cyclase inhibition in clonal cell lines: apparent differences in drug intrinsic efficacies between human 5-HT1D subtypes.

Authors:  J M Zgombick; L E Schechter; N Adham; S A Kucharewicz; R L Weinshank; T A Branchek
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1996 Aug-Sep       Impact factor: 3.000

5.  5HT1B receptor agonists inhibit light-induced phase shifts of behavioral circadian rhythms and expression of the immediate-early gene c-fos in the suprachiasmatic nucleus.

Authors:  G E Pickard; E T Weber; P A Scott; A F Riberdy; M A Rea
Journal:  J Neurosci       Date:  1996-12-15       Impact factor: 6.167

6.  RU 24969-induced locomotion in rats is mediated by 5-HT1A receptors.

Authors:  H O Kalkman
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1995-11       Impact factor: 3.000

7.  Postsynaptic 5-HT1B receptors modulate electroshock-induced generalised seizures in rats.

Authors:  Tania O Stean; Alan R Atkins; Christian A Heidbreder; Leann P Quinn; Brenda K Trail; Neil Upton
Journal:  Br J Pharmacol       Date:  2005-03       Impact factor: 8.739

8.  Functional behavioral homology between rat 5-HT1B and guinea pig 5-HT1D receptors in the modulation of prepulse inhibition of startle.

Authors:  T E Sipes; M A Geyer
Journal:  Psychopharmacology (Berl)       Date:  1996-06       Impact factor: 4.530

9.  Endophenotypes and serotonergic polymorphisms associated with treatment response in obsessive-compulsive disorder.

Authors:  Fábio M Corregiari; Márcio Bernik; Quirino Cordeiro; Homero Vallada
Journal:  Clinics (Sao Paulo)       Date:  2012       Impact factor: 2.365

10.  5-HT(1B) receptors, ventral orbitofrontal cortex, and aggressive behavior in mice.

Authors:  R M M De Almeida; M M Rosa; D M Santos; D M Saft; Q Benini; K A Miczek
Journal:  Psychopharmacology (Berl)       Date:  2006-03-21       Impact factor: 4.415
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