Literature DB >> 7932546

Structure-based design of HIV protease inhibitors: 4-hydroxycoumarins and 4-hydroxy-2-pyrones as non-peptidic inhibitors.

S Thaisrivongs1, P K Tomich, K D Watenpaugh, K T Chong, W J Howe, C P Yang, J W Strohbach, S R Turner, J P McGrath, M J Bohanon.   

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Year:  1994        PMID: 7932546     DOI: 10.1021/jm00046a002

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  8 in total

Review 1.  Impact of high-throughput screening in biomedical research.

Authors:  Ricardo Macarron; Martyn N Banks; Dejan Bojanic; David J Burns; Dragan A Cirovic; Tina Garyantes; Darren V S Green; Robert P Hertzberg; William P Janzen; Jeff W Paslay; Ulrich Schopfer; G Sitta Sittampalam
Journal:  Nat Rev Drug Discov       Date:  2011-03       Impact factor: 84.694

2.  Oxidative degradation of a sulfonamide-containing 5,6-dihydro-4-hydroxy-2-pyrone in aqueous/organic cosolvent mixtures.

Authors:  Susan W Hovorka; Michael J Hageman; Christian Schöneich
Journal:  Pharm Res       Date:  2002-04       Impact factor: 4.200

3.  Protein structure-based design of potent orally bioavailable, nonpeptide inhibitors of human immunodeficiency virus protease.

Authors:  S H Reich; M Melnick; J F Davies; K Appelt; K K Lewis; M A Fuhry; M Pino; A J Trippe; D Nguyen; H Dawson
Journal:  Proc Natl Acad Sci U S A       Date:  1995-04-11       Impact factor: 11.205

4.  2-Bromo-2-methyl-N-(4-methyl-2-oxo-2H-chromen-7-yl)propanamide.

Authors:  N Haridharan; V Ramkumar; R Dhamodharan
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2010-07-14

5.  Synthesis and Inhibiting Activity of Some 4-Hydroxycoumarin Derivatives on HIV-1 Protease.

Authors:  Stancho Stanchev; Frank Jensen; Anton Hinkov; Vasil Atanasov; Petia Genova-Kalou; Radka Argirova; Ilia Manolov
Journal:  ISRN Pharm       Date:  2011-07-26

Review 6.  Therapeutic potential of coumarins as antiviral agents.

Authors:  Mohd Zaheen Hassan; Hasnah Osman; Mohamed Ashraf Ali; Mohamed Jawed Ahsan
Journal:  Eur J Med Chem       Date:  2016-07-25       Impact factor: 6.514

Review 7.  Nitrogen-Based Heterocyclic Compounds: A Promising Class of Antiviral Agents against Chikungunya Virus.

Authors:  Andreza C Santana; Ronaldo C Silva Filho; José C J M D S Menezes; Diego Allonso; Vinícius R Campos
Journal:  Life (Basel)       Date:  2020-12-30

Review 8.  Biosynthesis of α-pyrones.

Authors:  Till F Schäberle
Journal:  Beilstein J Org Chem       Date:  2016-03-24       Impact factor: 2.883

  8 in total

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