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17 in total

1. Selective mGluR5 antagonists MPEP and SIB-1893 decrease NMDA or glutamate-mediated neuronal toxicity through actions that reflect NMDA receptor antagonism.

Authors: D M O'Leary; V Movsesyan; S Vicini; A I Faden
Journal: Br J Pharmacol Date: 2000-12 Impact factor: 8.739

2. Two new non-competitive mGlu1 receptor antagonists are potent tools to unravel functions of this mGlu receptor subtype.

Authors: T Knöpfel
Journal: Br J Pharmacol Date: 2007-05-14 Impact factor: 8.739

3. Enhanced sensitivity to attenuation of conditioned reinstatement by the mGluR 2/3 agonist LY379268 and increased functional activity of mGluR 2/3 in rats with a history of ethanol dependence.

Authors: Peter R Kufahl; Rémi Martin-Fardon; Friedbert Weiss
Journal: Neuropsychopharmacology Date: 2011-08-31 Impact factor: 7.853

4. Direct effects of metabotropic glutamate receptor compounds on native and recombinant N-methyl-D-aspartate receptors.

Authors: A Contractor; R W Gereau; T Green; S F Heinemann
Journal: Proc Natl Acad Sci U S A Date: 1998-07-21 Impact factor: 11.205

5. Interaction between the mGlu receptors 5 antagonist, MPEP, and amphetamine on memory and motor functions in mice.

Authors: Francesca Managò; Sebastien Lopez; Alberto Oliverio; Marianne Amalric; Andrea Mele; Elvira De Leonibus
Journal: Psychopharmacology (Berl) Date: 2012-11-29 Impact factor: 4.530

6. Benzimidazoles as Potent and Orally Active mGlu5 Receptor Antagonists with an Improved PK Profile.

Authors: David Carcache; Ivo Vranesic; Joachim Blanz; Sandrine Desrayaud; Markus Fendt; Ralf Glatthar
Journal: ACS Med Chem Lett Date: 2010-11-02 Impact factor: 4.345

7. Screening cascade and development of potential Positron Emission Tomography radiotracers for mGluR5: in vitro and in vivo characterization.

Authors: Shil Patel; Obinna Ndubizu; Terence Hamill; A Chaudhary; H Donald Burns; R Hargreaves; Raymond E Gibson
Journal: Mol Imaging Biol Date: 2005 Jul-Aug Impact factor: 3.488

8. Recent advances in the design and development of novel negative allosteric modulators of mGlu(5).

Authors: Kyle A Emmitte
Journal: ACS Chem Neurosci Date: 2011-08-17 Impact factor: 4.418

9. Epileptogenesis in vivo enhances the sensitivity of inhibitory presynaptic metabotropic glutamate receptors in basolateral amygdala neurons in vitro.

Authors: V Neugebauer; N B Keele; P Shinnick-Gallagher
Journal: J Neurosci Date: 1997-02-01 Impact factor: 6.167

10. Carnitine inhibits hydrolysis of inositol phospholipids induced by activation of metabotropic receptors.

Authors: M Llansola; V Felipo
Journal: Neurochem Res Date: 1998-12 Impact factor: 3.996