Literature DB >> 7278998

Super-active enkephalin analogues. Simple tripeptide hydroxyalkylamides exhibit surprisingly high and long-lasting opioid activities.

Y Kiso, M Yamaguchi, T Akita, H Moritoki, M Takei, H Nakamura.   

Abstract

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Year:  1981        PMID： 7278998     DOI： 10.1007/BF01047210

Source DB:  PubMed          Journal:  Naturwissenschaften        ISSN： 0028-1042


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  15 in total

1.  A method for evaluating both non-narcotic and narcotic analgesics.

Authors:  E SIEGMUND; R CADMUS; G LU
Journal:  Proc Soc Exp Biol Med       Date:  1957 Aug-Sep

2.  Analgesia induced in vivo by central administration of enkephalin in rat.

Authors:  J D Belluzzi; N Grant; V Garsky; D Sarantakis; C D Wise; L Stein
Journal:  Nature       Date:  1976-04-15       Impact factor: 49.962

3.  Extremely rapid degradation of [3H] methionine-enkephalin by various rat tissues in vivo and in vitro.

Authors:  A Dupont; L Cusan; M Garon; G Alvarado-Urbina; F Labrie
Journal:  Life Sci       Date:  1977-10-01       Impact factor: 5.037

4.  (D-met2, pro5)-enkephalinamide: a potent morphine-like analgesic.

Authors:  J I Székely; A Z Rónai; Z Dunai-Kovács; E Miglécz; I Berzétri; S Bajusz; L Gráf
Journal:  Eur J Pharmacol       Date:  1977-06-01       Impact factor: 4.432

5.  Evidence for analgesic activity of enkephalin in the mouse.

Authors:  H H Buscher; R C Hill; D Römer; F Cardinaux; A Closse; D Hauser; J Pless
Journal:  Nature       Date:  1976-06-03       Impact factor: 49.962

6.  Morphine-like activities of synthetic enkephalin analogues.

Authors:  H Moritoki; Y Kiso; T Kageyama; K Matsumoto
Journal:  J Pharm Pharmacol       Date:  1981-01       Impact factor: 3.765

7.  Tetrapeptide acyl-hydrazide analogs of enkephalin: a new group of potent analgesics.

Authors:  M Fujino; S Shinagawa; K Kawai; H Ishii
Journal:  Naturwissenschaften       Date:  1979-12

8.  Identification of two related pentapeptides from the brain with potent opiate agonist activity.

Authors:  J Hughes; T W Smith; H W Kosterlitz; L A Fothergill; B A Morgan; H R Morris
Journal:  Nature       Date:  1975-12-18       Impact factor: 49.962

9.  Comparative study of 1-cyclohexyl-4-(1,2-diphenylethyl)-piperazine and its enantiomorphs on analgesic and othe pharmacological activities in experimental animals.

Authors:  H Nakamura; M Shimizu
Journal:  Arch Int Pharmacodyn Ther       Date:  1976-05

10.  Kinetic parameters of narcotic agonists and antagonists, with particular reference to N-allylnoroxymorphone (naloxone).

Authors:  H W Kosterlitz; A J Watt
Journal:  Br J Pharmacol Chemother       Date:  1968-06
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  1 in total

1.  Development of novel lipophilic derivatives of DADLE (leucine enkephalin analogue): intestinal permeability characateristics of DADLE derivatives in rats.

Authors:  T Uchiyama; A Kotani; H Tatsumi; T Kishida; A Okamoto; N Okada; M Murakami; T Fujita; Y Fujiwara; Y Kiso; S Muranishi; A Yamamoto
Journal:  Pharm Res       Date:  2000-12       Impact factor: 4.200
  1 in total

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