Literature DB >> 4993720

1,4-benzodiazepines. Chemistry and some aspects of the structure-activity relationship.

L H Sternbach.   

Abstract

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Year:  1971        PMID： 4993720     DOI： 10.1002/anie.197100341

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  10 in total

Review 1.  Positive allosteric modulators to peptide GPCRs: a promising class of drugs.

Authors:  Tamas Bartfai; Ming-wei Wang
Journal:  Acta Pharmacol Sin       Date:  2013-04-29       Impact factor: 6.150

2.  Peptido-aminobenzophenones--novel latentiated benzo-1,4-diazepines.

Authors:  C H Hassall; S W Holmes; W H Johnson; A Kröhn; C E Smithen; W A Thomas
Journal:  Experientia       Date:  1977-11-15

3.  Photopotentiation of the GABAA receptor with caged diazepam.

Authors:  Lorenzo Sansalone; Joshua Bratsch-Prince; Sicheng Tang; Burjor Captain; David D Mott; Françisco M Raymo
Journal:  Proc Natl Acad Sci U S A       Date:  2019-10-01       Impact factor: 11.205

4.  Clobazam: chemical aspects of the 1,4 and 1,5-benzodiazepines.

Authors:  H Kuch
Journal:  Br J Clin Pharmacol       Date:  1979       Impact factor: 4.335

5.  Regioselective One-Pot Synthesis, Biological Activity and Molecular Docking Studies of Novel Conjugates N-(p-Aryltriazolyl)-1,5-benzodiazepin-2-ones as Potent Antibacterial and Antifungal Agents.

Authors:  Asma Nsira; Hasan Mtiraoui; Sami Chniti; Hanan Al-Ghulikah; Rafik Gharbi; Moncef Msaddek
Journal:  Molecules       Date:  2022-06-22       Impact factor: 4.927

Review 6.  Classics in chemical neuroscience: diazepam (valium).

Authors:  Nicholas E Calcaterra; James C Barrow
Journal:  ACS Chem Neurosci       Date:  2014-02-27       Impact factor: 4.418

Review 7.  The DARK Side of Total Synthesis: Strategies and Tactics in Psychoactive Drug Production.

Authors:  Schuyler A Chambers; Jenna M DeSousa; Eric D Huseman; Steven D Townsend
Journal:  ACS Chem Neurosci       Date:  2018-02-01       Impact factor: 4.418

8.  Diazepam is not a direct allosteric modulator of α1-adrenoceptors, but modulates receptor signaling by inhibiting phosphodiesterase-4.

Authors:  Lisa M Williams; Xiaoji He; Tasneem M Vaid; Alaa Abdul-Ridha; Alice R Whitehead; Paul R Gooley; Ross A D Bathgate; Spencer J Williams; Daniel J Scott
Journal:  Pharmacol Res Perspect       Date:  2018-12-26

9.  Can Mesoporous Silica Speed Up Degradation of Benzodiazepines? Hints from Quantum Mechanical Investigations.

Authors:  Massimo Delle Piane; Marta Corno
Journal:  Materials (Basel)       Date:  2022-02-12       Impact factor: 3.623

10.  A unified model of the GABA(A) receptor comprising agonist and benzodiazepine binding sites.

Authors:  Rikke Bergmann; Kristine Kongsbak; Pernille Louise Sørensen; Tommy Sander; Thomas Balle
Journal:  PLoS One       Date:  2013-01-07       Impact factor: 3.240
  10 in total

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