Literature DB >> 4588275

Optical isomers of aryl-2-piperidylmethanol antimalarial agents. Preparation, optical purity, and absolute stereochemistry.

F I Carroll, J T Blackwell.   

Abstract

Entities:  

Mesh:

Substances:

Year:  1974        PMID: 4588275     DOI: 10.1021/jm00248a015

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


× No keyword cloud information.
  13 in total

1.  In vitro activity of the enantiomers of mefloquine, halofantrine and enpiroline against Plasmodium falciparum.

Authors:  L K Basco; C Gillotin; F Gimenez; R Farinotti; J Le Bras
Journal:  Br J Clin Pharmacol       Date:  1992-05       Impact factor: 4.335

2.  Antimalarial activities of various 4-quinolonemethanols with special attention to WR-142,490 (mefloquine).

Authors:  L H Schmidt; R Crosby; J Rasco; D Vaughan
Journal:  Antimicrob Agents Chemother       Date:  1978-06       Impact factor: 5.191

3.  Identification of (+)-erythro-mefloquine as an active enantiomer with greater efficacy than mefloquine against Mycobacterium avium infection in mice.

Authors:  Luiz E Bermudez; Clark B Inderlied; Peter Kolonoski; Christopher B Chee; Priscilla Aralar; Mary Petrofsky; Toufan Parman; Carol E Green; Anita H Lewin; William Y Ellis; Lowell S Young
Journal:  Antimicrob Agents Chemother       Date:  2012-05-21       Impact factor: 5.191

4.  Mefloquine and psychotomimetics share neurotransmitter receptor and transporter interactions in vitro.

Authors:  Aaron Janowsky; Amy J Eshleman; Robert A Johnson; Katherine M Wolfrum; David J Hinrichs; Jongtae Yang; T Mark Zabriskie; Martin J Smilkstein; Michael K Riscoe
Journal:  Psychopharmacology (Berl)       Date:  2014-02-02       Impact factor: 4.530

5.  Crystal structure of (-)-mefloquine hydrochloride reveals consistency of configuration with biological activity.

Authors:  Jean M Karle; Isabella L Karle
Journal:  Antimicrob Agents Chemother       Date:  2002-05       Impact factor: 5.191

Review 6.  Mefloquine. A review of its antimalarial activity, pharmacokinetic properties and therapeutic efficacy.

Authors:  K J Palmer; S M Holliday; R N Brogden
Journal:  Drugs       Date:  1993-03       Impact factor: 9.546

7.  Crystal structure and molecular structure of mefloquine methylsulfonate monohydrate: implications for a malaria receptor.

Authors:  J M Karle; I L Karle
Journal:  Antimicrob Agents Chemother       Date:  1991-11       Impact factor: 5.191

8.  A high-performance liquid chromatographic method for the quantitative enantioselective analysis of mefloquine stereoisomers.

Authors:  Y Qiu; S Kitamura; J K Guillory
Journal:  Pharm Res       Date:  1992-12       Impact factor: 4.200

9.  Falciparum malaria in eastern Thailand: a randomized trial of the efficacy of a single dose of mefloquine.

Authors:  A L Fontanet; B D Johnston; A M Walker; Y Bergqvist; U Hellgren; W Rooney
Journal:  Bull World Health Organ       Date:  1994       Impact factor: 9.408

10.  Mefloquine and Its Enantiomers Are Active against Mycobacterium tuberculosis In Vitro and in Macrophages.

Authors:  Luiz E Bermudez; Laura Meek
Journal:  Tuberc Res Treat       Date:  2014-12-11
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.