Literature DB >> 34410435

The potential utility of [68 Ga]Ga-DOTA-FAPI-04 as a novel broad-spectrum oncological and non-oncological imaging agent-comparison with [18F]FDG.

Lianjun Lan1, Hanxiang Liu2,3,4, Yingwei Wang2,3,4, Jia Deng2,3,4, Dengsai Peng2,3,4, Yue Feng2,3,4, Li Wang2,3,4, Yue Chen5,6,7, Lin Qiu8,9,10.   

Abstract

PURPOSE: This study aimed to compare the detection performance of [68 Ga]Ga-DOTA-FAPI-04 and [18F]FDG PET/CT in the patients with various oncological and non-oncological lesions.
METHODS: A total of 123 patients underwent contemporaneous [68 Ga]Ga-DOTA-FAPI-04 and [18F]FDG PET/CT were included in this prospective study. The maximum standard uptake value (SUVmax) was measured to compare oncological and non-oncological lesion uptake. The sensitivity, specificity, predictive values, and accuracy of [18F]FDG and [68 Ga]Ga-DOTA-FAPI-04 PET/CT for detecting primary, metastatic, and non-oncological lesions were calculated and compared to evaluate the detection efficacy.
RESULTS: The study subjects consisted of 123 patients (69 men and 54 women; mean age 56.11 ± 11.94 years). Among the 102 patients with either newly diagnosed (82 patients) or previously treated solid tumor (20 patients), a total of 88 solid primary malignant tumors in 84/102 patients were detected. Two patients had two primary tumors each and 1 patient had three primary tumors. Among them, 58/102 and 43/102 patients had nodal (376 lesions) and distant metastases (406 lesions), respectively. Eight patients had hematological neoplasm. No malignant oncological diseases were detected in the remaining 13 patients. A total of 145 non-oncological lesions and benign tumors in 52/123 patients were detected incidentally. [68 Ga]Ga-DOTA-FAPI-04 PET/CT demonstrated a significantly higher uptake and detection rate for the primary (SUVmax 10.98 ± 5.83 vs. 8.36 ± 6.43, p < 0.001; sensitivity 97.67 vs. 84.89%; and accuracy 96.59 vs. 82.95%, X2 = 0.538, p = 0.021), nodal (SUVmax 10.50 ± 5.98 vs. 8.20 ± 6.29, p = 0.011; sensitivity 97.59 vs. 84.72%; and accuracy 97.34 vs. 84.31%, X2 = 2.067, p < 0.001), and distant metastatic lesions (SUVmax 9.64 ± 6.45 vs. 6.74 ± 4.83; p < 0.001; sensitivity 98.01 vs. 65.59%; and accuracy 97.04 vs. 65.51%, X2 = 4.897, p < 0.001) of solid tumor than did [18F]FDG PET/CT. [68 Ga]Ga-DOTA-FAPI-04 PET/CT demonstrated a lower activity (SUVmax: 6.84 ± 4.67 vs. 13.09 ± 7.29, p < 0.001) and detection rate (sensitivity 50.65 vs. 96.75%, and accuracy 51.28 vs. 95.51%, X2 = 5.166, p < 0.001) for multiple myeloma and lymphoma compared to [18F]FDG PET/CT. [68 Ga]Ga-DOTA-FAPI-04 and [18F]FDG PET/CT PET/CT demonstrated a comparative activity (SUVmax 6.40 ± 3.95 vs. 5.74 ± 15.78, p = 0.729) and detection efficacy (sensitivity 86.52 vs. 72.34%, and accuracy 84.83 vs. 72.41%, X2 = 9.460, p = 0.007) for non-oncological lesion and benign tumor detection.
CONCLUSIONS: Except for myeloma and lymphoma, [68 Ga]Ga-DOTA-FAPI-04 PET/CT showed a superior detection efficacy for detecting various primary and metastatic lesions than [18F]FDG PET/CT. A comparative detection utility for non-oncological lesion was obtained with both tracers. [68 Ga]Ga-DOTA-FAPI-04 could be used as a broad-spectrum tumor and inflammatory imaging agent in the clinical especially for various solid tumors and non-oncological lesions.
© 2021. The Author(s), under exclusive licence to Springer-Verlag GmbH Germany, part of Springer Nature.

Entities:  

Keywords:  Broad-spectrum imaging agent; Fibroblast activation protein (FAP); [18F]FDG; [68 Ga]Ga-DOTA-FAPI-04

Mesh:

Substances:

Year:  2021        PMID: 34410435     DOI: 10.1007/s00259-021-05522-w

Source DB:  PubMed          Journal:  Eur J Nucl Med Mol Imaging        ISSN: 1619-7070            Impact factor:   9.236


  34 in total

1.  Increased expression of fibroblast activation protein-alpha in keloid fibroblasts: implications for development of a novel treatment option.

Authors:  Kirstin Dienus; Ardeshir Bayat; Brendan F Gilmore; Oliver Seifert
Journal:  Arch Dermatol Res       Date:  2010-09-26       Impact factor: 3.017

Review 2.  Emerging roles of serine proteinases in tissue turnover in arthritis.

Authors:  J M Milner; A Patel; A D Rowan
Journal:  Arthritis Rheum       Date:  2008-12

3.  Development of Quinoline-Based Theranostic Ligands for the Targeting of Fibroblast Activation Protein.

Authors:  Thomas Lindner; Anastasia Loktev; Annette Altmann; Frederik Giesel; Clemens Kratochwil; Jürgen Debus; Dirk Jäger; Walter Mier; Uwe Haberkorn
Journal:  J Nucl Med       Date:  2018-04-06       Impact factor: 10.057

4.  Loss of cells expressing fibroblast activation protein has variable effects in models of TGF-β and chronic bleomycin-induced fibrosis.

Authors:  Toru Kimura; James Monslow; Astero Klampatsa; Michael Leibowitz; Jing Sun; Maria Liousia; Patrick Woodruff; Edmund Moon; Leslie Todd; Ellen Puré; Steven M Albelda
Journal:  Am J Physiol Lung Cell Mol Physiol       Date:  2019-06-12       Impact factor: 5.464

5.  Cell surface glycoprotein of reactive stromal fibroblasts as a potential antibody target in human epithelial cancers.

Authors:  P Garin-Chesa; L J Old; W J Rettig
Journal:  Proc Natl Acad Sci U S A       Date:  1990-09       Impact factor: 11.205

Review 6.  Fibroblast activation protein and chronic liver disease.

Authors:  Xin Maggie Wang; Tsun-Wen Yao; Naveed A Nadvi; Brenna Osborne; Geoffrey W McCaughan; Mark D Gorrell
Journal:  Front Biosci       Date:  2008-01-01

7.  Molecular cloning of fibroblast activation protein alpha, a member of the serine protease family selectively expressed in stromal fibroblasts of epithelial cancers.

Authors:  M J Scanlan; B K Raj; B Calvo; P Garin-Chesa; M P Sanz-Moncasi; J H Healey; L J Old; W J Rettig
Journal:  Proc Natl Acad Sci U S A       Date:  1994-06-07       Impact factor: 11.205

8.  Fibroblast activation protein alpha is expressed by chondrocytes following a pro-inflammatory stimulus and is elevated in osteoarthritis.

Authors:  Jennifer M Milner; Lara Kevorkian; David A Young; Debra Jones; Robin Wait; Simon T Donell; Emma Barksby; Angela M Patterson; Jim Middleton; Benjamin F Cravatt; Ian M Clark; Andrew D Rowan; Timothy E Cawston
Journal:  Arthritis Res Ther       Date:  2006-01-03       Impact factor: 5.156

9.  Fibroblast activation protein is expressed by rheumatoid myofibroblast-like synoviocytes.

Authors:  Stefan Bauer; Michael C Jendro; Andreas Wadle; Sascha Kleber; Frank Stenner; Robert Dinser; Anja Reich; Erica Faccin; Stefan Gödde; Harald Dinges; Ulf Müller-Ladner; Christoph Renner
Journal:  Arthritis Res Ther       Date:  2006       Impact factor: 5.156

10.  A Tumor-Imaging Method Targeting Cancer-Associated Fibroblasts.

Authors:  Anastasia Loktev; Thomas Lindner; Walter Mier; Jürgen Debus; Annette Altmann; Dirk Jäger; Frederik Giesel; Clemens Kratochwil; Philippe Barthe; Christian Roumestand; Uwe Haberkorn
Journal:  J Nucl Med       Date:  2018-04-06       Impact factor: 10.057

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  12 in total

1.  [18F]FAPI-42 PET/CT versus [18F]FDG PET/CT for imaging of recurrent or metastatic gastrointestinal stromal tumors.

Authors:  Chunhui Wu; Xinhua Zhang; Yu Zeng; Renbo Wu; Li Ding; Yanzhe Xia; Zhifeng Chen; Xiangsong Zhang; Xiaoyan Wang
Journal:  Eur J Nucl Med Mol Imaging       Date:  2022-08-30       Impact factor: 10.057

2.  Comparison of Diagnostic Efficacy of [68Ga]Ga-FAPI-04 and [18F]FDG PET/CT for Staging and Restaging of Gastric Cancer.

Authors:  Shumao Zhang; Wei Wang; Tingting Xu; Haoyuan Ding; Yi Li; Huipan Liu; Yinxue Huang; Lin Liu; Tao Du; Yan Zhao; Yue Chen; Lin Qiu
Journal:  Front Oncol       Date:  2022-07-01       Impact factor: 5.738

3.  Comparison of [68Ga]Ga-DOTA-FAPI-04 and [18F]FDG Uptake in Esophageal Cancer.

Authors:  Huipan Liu; Zhi Hu; Xiao Yang; Tianyang Dai; Yue Chen
Journal:  Front Oncol       Date:  2022-06-16       Impact factor: 5.738

4.  Comparison of 68Ga-FAPI and 18F-FDG PET/CT in the Evaluation of Patients With Newly Diagnosed Non-Small Cell Lung Cancer.

Authors:  Junhao Wu; Hao Deng; Haoshu Zhong; Tao Wang; Zijuan Rao; Yingwei Wang; Yue Chen; Chunyin Zhang
Journal:  Front Oncol       Date:  2022-07-04       Impact factor: 5.738

5.  18F-FDG and 68 Ga-FAPI PET/CT for the evaluation of periprosthetic joint infection and aseptic loosening in rabbit models.

Authors:  Yiqun Wang; Yu Li; Liang Han; Xiaojun Zhang; Yong Huan; Jiahe Tian; Jun Wang; Cong Zhang; Erpeng Qi; Dongyun Zhang
Journal:  BMC Musculoskelet Disord       Date:  2022-06-20       Impact factor: 2.562

Review 6.  Clinical summary of fibroblast activation protein inhibitor-based radiopharmaceuticals: cancer and beyond.

Authors:  Mengting Li; Muhsin H Younis; Yongxue Zhang; Weibo Cai; Xiaoli Lan
Journal:  Eur J Nucl Med Mol Imaging       Date:  2022-01-31       Impact factor: 10.057

7.  [99mTc]Tc-iFAP Radioligand for SPECT/CT Imaging of the Tumor Microenvironment: Kinetics, Radiation Dosimetry, and Imaging in Patients.

Authors:  Luis Coria-Domínguez; Paola Vallejo-Armenta; Myrna Luna-Gutiérrez; Blanca Ocampo-García; Brenda Gibbens-Bandala; Francisco García-Pérez; Gerardo Ramírez-Nava; Clara Santos-Cuevas; Guillermina Ferro-Flores
Journal:  Pharmaceuticals (Basel)       Date:  2022-05-11

8.  Head-to-Head Comparison of Fibroblast Activation Protein Inhibitors (FAPI) Radiotracers versus [18F]F-FDG in Oncology: A Systematic Review.

Authors:  Giorgio Treglia; Barbara Muoio; Hessamoddin Roustaei; Zahra Kiamanesh; Kamran Aryana; Ramin Sadeghi
Journal:  Int J Mol Sci       Date:  2021-10-17       Impact factor: 5.923

Review 9.  Fibroblast activation protein-based theranostics in cancer research: A state-of-the-art review.

Authors:  Liang Zhao; Jianhao Chen; Yizhen Pang; Kaili Fu; Qihang Shang; Hua Wu; Long Sun; Qin Lin; Haojun Chen
Journal:  Theranostics       Date:  2022-01-09       Impact factor: 11.556

10.  Comparison of [68Ga]-FAPI PET/CT and [18F]-FDG PET/CT in Multiple Myeloma: Clinical Experience.

Authors:  Umut Elboga; Ertan Sahin; Yusuf Burak Cayirli; Merve Okuyan; Gokmen Aktas; Handan Haydaroglu Sahin; Ilkay Dogan; Tulay Kus; Dervis Murat Akkurd; Ufuk Cimen; Vuslat Mumcu; Benan Kilbas; Yusuf Zeki Celen
Journal:  Tomography       Date:  2022-02-01
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