Literature DB >> 34120336

Pilot randomized placebo-controlled clinical trial of high-dose gabapentin for alcohol use disorder.

John J Mariani1,2, Martina Pavlicova3, Cale Basaraba4, Agnieszka Mamczur-Fuller5, Daniel J Brooks1, Adam Bisaga1,2, Kenneth M Carpenter1,2, Edward V Nunes1,2, Frances R Levin1,2.   

Abstract

BACKGROUND: Despite advances in the development of pharmacotherapy for alcohol use disorder (AUD), there remains a need for medications that can be administered to actively drinking outpatients to promote a reduction in harmful alcohol consumption. The primary aim of this pilot study was to determine whether high-dose gabapentin (3600 mg/daily) is more effective than placebo in reducing harmful alcohol consumption in outpatients with AUD.
METHODS: Forty patients (27 men) who met DSM-IV-TR criteria for alcohol dependence and reporting at least 4 heavy drinking days (HDD) per week were recruited at a single site. Participants were actively drinking at study entry and received double-blind gabapentin (3600 mg/day; n = 19) or placebo (n = 20) for 8 weeks. Study medication was titrated over 5 days and administered in three divided doses (1200 mg three times per day). The proportion of HDD (primary outcome) and percent days abstinent (PDA; secondary outcome) were analyzed using generalized longitudinal mixed models with the predictors being study arm, week, study arm by week interaction, and corresponding baseline drinking measure.
RESULTS: There was a significant interaction between study arm and week for the proportion of HDD per week, F (7, 215) = 3.33, p = 0.002 . There was also a significant interaction between study arm and week for PDA per week, F (7, 215) = 3.11, p = 0.004. The overall retention rate was 67.5% with no significant difference in time-to-dropout between treatment groups. There were no serious adverse events. No participants were removed from the trial due to the development of moderate-to-severe alcohol withdrawal (CIWA-Ar ≥ 13).
CONCLUSIONS: Gabapentin treatment rapidly titrated to a dosage of 3600 mg/day is associated with a reduction in the proportion of HDD per week and an increase in PDA per week in actively drinking outpatients with AUD. High-dose gabapentin is potentially a feasible approach to treating AUD and deserving of further study.
© 2021 by the Research Society on Alcoholism.

Entities:  

Keywords:  alcohol use disorder; gabapentin; pharmacotherapy

Mesh:

Substances:

Year:  2021        PMID: 34120336      PMCID: PMC8462978          DOI: 10.1111/acer.14648

Source DB:  PubMed          Journal:  Alcohol Clin Exp Res        ISSN: 0145-6008            Impact factor:   3.928


  54 in total

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8.  The effect of gabapentin on brain gamma-aminobutyric acid in patients with epilepsy.

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