Literature DB >> 33936371

EphA2 as a new target for breast cancer and its potential clinical application.

Lingzhi Zhou1, Xuejing Lu1, Bensi Zhang2, Yaqi Shi2, Zhuang Li1.   

Abstract

PURPOSE: The aim of this research was to study the expression of EphA2 to assess its suitability as a new breast cancer target.
METHODS: Immunohistochemistry (IHC) was used to detect EphA2 protein expression in pathology tissue samples from 250 cases of breast cancer, and the expression of EphA2 mRNA was detected by in situ hybridization (ISH). Breast cancer cells were isolated and cultured. The expression of EphA2 in the cells was detected by the indirect immunofluorescence assay (IFA), and the expression of EphA2 in breast cancer was analysed.
RESULTS: EphA2 protein and mRNA were mainly expressed in tumor cells and vascular endothelial cells. EphA2 protein was expressed in 187 cases, with a positive rate of 74.80%, whereas EphA2 mRNA was expressed in 209 cases, with a positive rate of 83.60%. EphA2 protein and mRNA expression were correlated with lymph node metastasis, clinical stage, and breast cancer histologic grade (P<0.05). In addition, the positive expression rates of EphA2 protein and EphA2 mRNA were correlated (P<0.05). EphA2 was barely expressed in normal breast cells but highly expressed in breast cancer cells.
CONCLUSION: EphA2 is highly expressed in breast cancer tissues and has the potential to be a new breast cancer target, providing a preliminary basis for the development of new targeted drugs for breast cancer and the construction of fluorescent-targeted tracers for fluorescence-guided mastoscopic breast-conserving surgery. IJCEP
Copyright © 2021.

Entities:  

Keywords:  Breast cancer; EphA2; target

Year:  2021        PMID: 33936371      PMCID: PMC8085825     

Source DB:  PubMed          Journal:  Int J Clin Exp Pathol        ISSN: 1936-2625


  22 in total

1.  EphA2 inhibition suppresses proliferation of small-cell lung cancer cells through inducing cell cycle arrest.

Authors:  Hirotoshi Ishigaki; Toshiyuki Minami; Osamu Morimura; Hidemi Kitai; Daisuke Horio; Yuichi Koda; Eriko Fujimoto; Yoshiki Negi; Yasuhiro Nakajima; Maiko Niki; Shingo Kanemura; Eisuke Shibata; Koji Mikami; Ryo Takahashi; Takashi Yokoi; Kozo Kuribayashi; Takashi Kijima
Journal:  Biochem Biophys Res Commun       Date:  2019-09-24       Impact factor: 3.575

2.  Dual targeting for metastatic breast cancer and tumor neovasculature by EphA2-mediated nanocarriers.

Authors:  Zhaoming Guo; Bing He; Lan Yuan; Wenbing Dai; Hua Zhang; Xueqing Wang; Jiancheng Wang; Xuan Zhang; Qiang Zhang
Journal:  Int J Pharm       Date:  2015-05-21       Impact factor: 5.875

3.  Dysregulation of EGFR Pathway in EphA2 Cell Subpopulation Significantly Associates with Poor Prognosis in Colorectal Cancer.

Authors:  Mariangela De Robertis; Luisa Loiacono; Caterina Fusilli; Maria Luana Poeta; Tommaso Mazza; Massimo Sanchez; Luigi Marchionni; Emanuela Signori; Giuseppe Lamorte; Angelo Luigi Vescovi; Jesus Garcia-Foncillas; Vito Michele Fazio
Journal:  Clin Cancer Res       Date:  2016-07-11       Impact factor: 12.531

Review 4.  The EphA2 receptor and ephrinA1 ligand in solid tumors: function and therapeutic targeting.

Authors:  Jill Wykosky; Waldemar Debinski
Journal:  Mol Cancer Res       Date:  2008-12       Impact factor: 5.852

5.  EphA2 Expression Is a Key Driver of Migration and Invasion and a Poor Prognostic Marker in Colorectal Cancer.

Authors:  Philip D Dunne; Sonali Dasgupta; Patrick G Johnston; Sandra Van Schaeybroeck; Jaine K Blayney; Darragh G McArt; Keara L Redmond; Jessica-Anne Weir; Conor A Bradley; Takehiko Sasazuki; Senji Shirasawa; Tingting Wang; Supriya Srivastava; Chee Wee Ong; Ken Arthur; Manuel Salto-Tellez; Richard H Wilson
Journal:  Clin Cancer Res       Date:  2015-08-17       Impact factor: 12.531

6.  EphA2 in the early pathogenesis and progression of non-small cell lung cancer.

Authors:  Jennifer M Brannan; Banibrata Sen; Babita Saigal; Ludmila Prudkin; Carmen Behrens; Luisa Solis; Wenli Dong; B Nebiyou Bekele; Ignacio Wistuba; Faye M Johnson
Journal:  Cancer Prev Res (Phila)       Date:  2009-11-24

7.  Expression of EphA2 and E-cadherin in gastric cancer: correlated with tumor progression and lymphogenous metastasis.

Authors:  Weijie Yuan; Zhikang Chen; Shaobin Wu; Jie Ge; Shi Chang; Xianwei Wang; Jingxiang Chen; Zihua Chen
Journal:  Pathol Oncol Res       Date:  2009-09       Impact factor: 3.201

Review 8.  Emerging and Diverse Functions of the EphA2 Noncanonical Pathway in Cancer Progression.

Authors:  Yue Zhou; Hiroaki Sakurai
Journal:  Biol Pharm Bull       Date:  2017       Impact factor: 2.233

9.  Back-Table Fluorescence-Guided Imaging for Circumferential Resection Margin Evaluation Using Bevacizumab-800CW in Patients with Locally Advanced Rectal Cancer.

Authors:  Steven J de Jongh; Jolien J J Tjalma; Marjory Koller; Matthijs D Linssen; Jasper Vonk; Michael Dobosz; Annelies Jorritsma-Smit; Jan H Kleibeuker; Geke A P Hospers; Klaas Havenga; Patrick H J Hemmer; Arend Karrenbeld; Gooitzen M van Dam; Boudewijn van Etten; Wouter B Nagengast
Journal:  J Nucl Med       Date:  2019-10-18       Impact factor: 10.057

10.  Eph/ephrin profiling in human breast cancer reveals significant associations between expression level and clinical outcome.

Authors:  Dana M Brantley-Sieders; Aixiang Jiang; Krishna Sarma; Akosua Badu-Nkansah; Debra L Walter; Yu Shyr; Jin Chen
Journal:  PLoS One       Date:  2011-09-15       Impact factor: 3.240

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