Literature DB >> 33356664

Intramuscular cobinamide as an antidote to methyl mercaptan poisoning.

Tara B Hendry-Hofer1, Patrick C Ng1,2, Alison M McGrath3, Kirsten Soules1, David S Mukai4, Adriano Chan5, Joseph K Maddry6, Carl W White7, Jangwoen Lee4, Sari B Mahon4, Matthew Brenner4, Gerry R Boss5, Vikhyat S Bebarta1,6.   

Abstract

BACKGROUND: Methyl mercaptan occurs naturally in the environment and is found in a variety of occupational settings, including the oil, paper, plastics, and pesticides industries. It is a toxic gas and deaths from methyl mercaptan exposure have occurred. The Department of Homeland Security considers it a high threat chemical agent that could be used by terrorists. Unfortunately, no specific treatment exists for methyl mercaptan poisoning.
METHODS: We conducted a randomized trial in 12 swine comparing no treatment to intramuscular injection of the vitamin B12 analog cobinamide (2.0 mL, 12.5 mg/kg) following acute inhalation of methyl mercaptan gas. Physiological and laboratory parameters were similar in the control and cobinamide-treated groups at baseline and at the time of treatment.
RESULTS: All six cobinamide-treated animals survived, whereas only one of six control animals lived (17% survival) (p = 0.0043). The cobinamide-treated animals returned to a normal breathing pattern by 3.8 ± 1.1 min after treatment (mean ± SD), while all but one animal in the control group had intermittent gasping, never regaining a normal breathing pattern. Blood pressure and arterial oxygen saturation returned to baseline values within 15 minutes of cobinamide-treatment. Plasma lactate concentration increased progressively until death (10.93 ± 6.02 mmol [mean ± SD]) in control animals, and decreased toward baseline (3.79 ± 2.93 mmol [mean ± SD]) by the end of the experiment in cobinamide-treated animals.
CONCLUSION: We conclude that intramuscular administration of cobinamide improves survival and clinical outcomes in a large animal model of acute, high dose methyl mercaptan poisoning.

Entities:  

Keywords:  Methyl mercaptan; cobinamide; inhalation; methanethiol; swine

Mesh:

Substances:

Year:  2020        PMID: 33356664      PMCID: PMC8063453          DOI: 10.1080/08958378.2020.1866123

Source DB:  PubMed          Journal:  Inhal Toxicol        ISSN: 0895-8378            Impact factor:   2.724


  18 in total

1.  Occupational exposure to chemical agents in the paper industry.

Authors:  K Korhonen; T Liukkonen; W Ahrens; G Astrakianakis; P Boffetta; A Burdorf; D Heederik; T Kauppinen; M Kogevinas; P Osvoll; B A Rix; A Saalo; J Sunyer; I Szadkowska-Stanczyk; K Teschke; H Westberg; K Widerkiewicz
Journal:  Int Arch Occup Environ Health       Date:  2004-09-10       Impact factor: 3.015

2.  The Vitamin B12 Analog Cobinamide Is an Effective Antidote for Oral Cyanide Poisoning.

Authors:  Jangwoen Lee; Sari B Mahon; David Mukai; Tanya Burney; Behdod S Katebian; Adriano Chan; Vikhyat S Bebarta; David Yoon; Gerry R Boss; Matthew Brenner
Journal:  J Med Toxicol       Date:  2016-09-15

3.  Efficacy of Intravenous Cobinamide Versus Hydroxocobalamin or Saline for Treatment of Severe Hydrogen Sulfide Toxicity in a Swine (Sus scrofa) Model.

Authors:  Vikhyat S Bebarta; Normalynn Garrett; Matthew Brenner; Sari B Mahon; Joseph K Maddry; Susan Boudreau; Maria Castaneda; Gerry R Boss
Journal:  Acad Emerg Med       Date:  2017-08-09       Impact factor: 3.451

4.  International data base of exposure measurements in the pulp, paper and paper product industries.

Authors:  T Kauppinen; K Teschke; A Savela; M Kogevinas; P Boffetta
Journal:  Int Arch Occup Environ Health       Date:  1997       Impact factor: 3.015

5.  Intramuscular cobinamide versus saline for treatment of severe hydrogen sulfide toxicity in swine.

Authors:  Patrick C Ng; Tara B Hendry-Hofer; Norma Garrett; Matthew Brenner; Sari B Mahon; Joseph K Maddry; Philippe Haouzi; Gerry R Boss; Thomas F Gibbons; Allyson A Araña; Vikhyat S Bebarta
Journal:  Clin Toxicol (Phila)       Date:  2018-11-15       Impact factor: 4.467

6.  Kinetics and mechanism of the reaction of hydrogen sulfide with diaquacobinamide in aqueous solution.

Authors:  Denis S Salnikov; Sergei V Makarov; Rudi van Eldik; Polina N Kucherenko; Gerry R Boss
Journal:  Eur J Inorg Chem       Date:  2014-09       Impact factor: 2.524

7.  Reactions of mercaptans with cytochrome c oxidase and cytochrome c.

Authors:  J Wilms; J Lub; R Wever
Journal:  Biochim Biophys Acta       Date:  1980-02-08

Review 8.  Hydrogen Sulfide Toxicity: Mechanism of Action, Clinical Presentation, and Countermeasure Development.

Authors:  Patrick C Ng; Tara B Hendry-Hofer; Alyssa E Witeof; Matthew Brenner; Sari B Mahon; Gerry R Boss; Philippe Haouzi; Vikhyat S Bebarta
Journal:  J Med Toxicol       Date:  2019-05-06

9.  Intravenous cobinamide versus hydroxocobalamin for acute treatment of severe cyanide poisoning in a swine (Sus scrofa) model.

Authors:  Vikhyat S Bebarta; David A Tanen; Susan Boudreau; Maria Castaneda; Lee A Zarzabal; Toni Vargas; Gerry R Boss
Journal:  Ann Emerg Med       Date:  2014-04-18       Impact factor: 5.721

10.  Intramuscular aminotetrazole cobinamide as a treatment for inhaled hydrogen sulfide poisoning in a large swine model.

Authors:  Tara B Hendry-Hofer; Patrick C Ng; Alison M McGrath; David Mukai; Matthew Brenner; Sari Mahon; Joseph K Maddry; Gerry R Boss; Vikhyat S Bebarta
Journal:  Ann N Y Acad Sci       Date:  2020-03-31       Impact factor: 5.691

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  2 in total

Review 1.  Versatile enzymology and heterogeneous phenotypes in cobalamin complementation type C disease.

Authors:  Anna J Esser; Srijan Mukherjee; Ilia A Dereven'kov; Sergei V Makarov; Donald W Jacobsen; Ute Spiekerkoetter; Luciana Hannibal
Journal:  iScience       Date:  2022-08-18

2.  Development of sodium tetrathionate as a cyanide and methanethiol antidote.

Authors:  Adriano Chan; Jangwoen Lee; Subrata Bhadra; Nesta Bortey-Sam; Tara B Hendry-Hofer; Vikhyat S Bebarta; Sari B Mahon; Matthew Brenner; Brian Logue; Renate B Pilz; Gerry R Boss
Journal:  Clin Toxicol (Phila)       Date:  2021-07-30       Impact factor: 4.467

  2 in total

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