Literature DB >> 30430872

Intramuscular cobinamide versus saline for treatment of severe hydrogen sulfide toxicity in swine.

Patrick C Ng1, Tara B Hendry-Hofer2, Norma Garrett3, Matthew Brenner4, Sari B Mahon4, Joseph K Maddry5, Philippe Haouzi6, Gerry R Boss7, Thomas F Gibbons8, Allyson A Araña5, Vikhyat S Bebarta2.   

Abstract

INTRODUCTION: Hydrogen sulfide (H2S) is found in petroleum, natural gas, and decaying organic matter. Terrorist groups have attempted to use it in enclosed spaces as a chemical weapon. Mass casualty scenarios have occurred from industrial accidents and release from oil field sites. There is no FDA approved antidote for sulfide poisoning. We have previously reported that intravenous cobinamide is effective for sulfide poisoning. A rapid-acting antidote that is easy to administer intramuscularly (IM) would be ideal for use in a prehospital setting. In this study, we assessed survival in sulfide-poisoned swine treated with IM cobinamide.
METHODS: Eleven swine (45-55 kg) were anesthetized, intubated, and instrumented with continuous femoral and pulmonary artery pressure monitoring. After stabilization, anesthesia was adjusted such that animals ventilated spontaneously with a FiO2 of 0.21. Sodium hydrosulfide (NaHS, 8 mg/mL) was infused intravenously at 0.9 mg/kg.min until apnea or severe hypotension. Animals were randomly assigned to receive cobinamide (4 mg/kg), or no treatment at the apnea/hypotension trigger. The NaHS infusion rate was sustained for 1.5 min post trigger, decreased to 0.2 mg/kg.min for 10 min, and then discontinued.
RESULTS: The amount of NaHS required to produce apnea or hypotension was not statistically different in both groups (cobinamide: 9.0 mg/kg ±6.1; saline: 5.9 mg/kg ±5.5; mean difference: -3.1, 95% CI: -11.3, 5.0). All of the cobinamide treated animals survived (5/5), none of the control (0/6) animals survived (p < .01). Mean time to return to spontaneous ventilation in the cobinamide treated animals was 3.2 (±1.1) min. Time to return to baseline systolic blood pressure (±5%) in cobinamide-treated animals was 5 min.
CONCLUSION: Intramuscular cobinamide was effective in improving survival in this large swine model of severe hydrogen sulfide toxicity.

Entities:  

Keywords:  Cobinamide; hydrogen sulfide toxicity; resuscitation; swine

Mesh:

Substances:

Year:  2018        PMID: 30430872      PMCID: PMC6540978          DOI: 10.1080/15563650.2018.1504955

Source DB:  PubMed          Journal:  Clin Toxicol (Phila)        ISSN: 1556-3650            Impact factor:   4.467


  10 in total

1.  Efficacy of Intravenous Cobinamide Versus Hydroxocobalamin or Saline for Treatment of Severe Hydrogen Sulfide Toxicity in a Swine (Sus scrofa) Model.

Authors:  Vikhyat S Bebarta; Normalynn Garrett; Matthew Brenner; Sari B Mahon; Joseph K Maddry; Susan Boudreau; Maria Castaneda; Gerry R Boss
Journal:  Acad Emerg Med       Date:  2017-08-09       Impact factor: 3.451

2.  Hydraulic fracturing for natural gas: impact on health and environment.

Authors:  David O Carpenter
Journal:  Rev Environ Health       Date:  2016-03       Impact factor: 3.458

Review 3.  Swine as models in biomedical research and toxicology testing.

Authors:  M M Swindle; A Makin; A J Herron; F J Clubb; K S Frazier
Journal:  Vet Pathol       Date:  2011-03-25       Impact factor: 2.221

4.  Cobinamide is effective for treatment of hydrogen sulfide-induced neurological sequelae in a mouse model.

Authors:  Poojya Anantharam; Elizabeth M Whitley; Belinda Mahama; Dong-Suk Kim; Souvarish Sarkar; Cristina Santana; Adriano Chan; Anumantha G Kanthasamy; Arthi Kanthasamy; Gerry R Boss; Wilson K Rumbeiha
Journal:  Ann N Y Acad Sci       Date:  2017-11       Impact factor: 5.691

5.  Nitrocobinamide, a new cyanide antidote that can be administered by intramuscular injection.

Authors:  Adriano Chan; Jingjing Jiang; Alla Fridman; Ling T Guo; G Diane Shelton; Ming-Tao Liu; Carol Green; Kristofer J Haushalter; Hemal H Patel; Jangwoen Lee; David Yoon; Tanya Burney; David Mukai; Sari B Mahon; Matthew Brenner; Renate B Pilz; Gerry R Boss
Journal:  J Med Chem       Date:  2015-02-16       Impact factor: 7.446

Review 6.  Toxicology of hydrogen sulfide.

Authors:  R J Reiffenstein; W C Hulbert; S H Roth
Journal:  Annu Rev Pharmacol Toxicol       Date:  1992       Impact factor: 13.820

Review 7.  Animal models of toxicology testing: the role of pigs.

Authors:  Kristi L Helke; Marvin Michael Swindle
Journal:  Expert Opin Drug Metab Toxicol       Date:  2012-12-10       Impact factor: 4.481

8.  Hydrogen Sulfide--Mechanisms of Toxicity and Development of an Antidote.

Authors:  Jingjing Jiang; Adriano Chan; Sameh Ali; Arindam Saha; Kristofer J Haushalter; Wai-Ling Macrina Lam; Megan Glasheen; James Parker; Matthew Brenner; Sari B Mahon; Hemal H Patel; Rajesh Ambasudhan; Stuart A Lipton; Renate B Pilz; Gerry R Boss
Journal:  Sci Rep       Date:  2016-02-15       Impact factor: 4.379

9.  Midazolam Efficacy Against Acute Hydrogen Sulfide-Induced Mortality and Neurotoxicity.

Authors:  Poojya Anantharam; Dong-Suk Kim; Elizabeth M Whitley; Belinda Mahama; Paula Imerman; Piyush Padhi; Wilson K Rumbeiha
Journal:  J Med Toxicol       Date:  2018-01-09

10.  Hydrogen sulfide exposure in an adult male.

Authors:  Bassam Doujaiji; Jaffar A Al-Tawfiq
Journal:  Ann Saudi Med       Date:  2010 Jan-Feb       Impact factor: 1.526

  10 in total
  2 in total

Review 1.  Hydrogen Sulfide Toxicity: Mechanism of Action, Clinical Presentation, and Countermeasure Development.

Authors:  Patrick C Ng; Tara B Hendry-Hofer; Alyssa E Witeof; Matthew Brenner; Sari B Mahon; Gerry R Boss; Philippe Haouzi; Vikhyat S Bebarta
Journal:  J Med Toxicol       Date:  2019-05-06

2.  Intramuscular cobinamide as an antidote to methyl mercaptan poisoning.

Authors:  Tara B Hendry-Hofer; Patrick C Ng; Alison M McGrath; Kirsten Soules; David S Mukai; Adriano Chan; Joseph K Maddry; Carl W White; Jangwoen Lee; Sari B Mahon; Matthew Brenner; Gerry R Boss; Vikhyat S Bebarta
Journal:  Inhal Toxicol       Date:  2020-12-26       Impact factor: 2.724

  2 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.