Literature DB >> 3278180

GABA synaptic mechanisms: stereochemical and conformational requirements.

P Krogsgaard-Larsen1.   

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Year:  1988        PMID： 3278180     DOI： 10.1002/med.2610080103

Source DB:  PubMed          Journal:  Med Res Rev        ISSN： 0198-6325            Impact factor:   12.944


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  10 in total

1.  Activation of single heteromeric GABA(A) receptor ion channels by full and partial agonists.

Authors:  Martin Mortensen; Uffe Kristiansen; Bjarke Ebert; Bente Frølund; Povl Krogsgaard-Larsen; Trevor G Smart
Journal:  J Physiol       Date:  2004-02-27       Impact factor: 5.182

2.  Distinct activities of GABA agonists at synaptic- and extrasynaptic-type GABAA receptors.

Authors:  Martin Mortensen; Bjarke Ebert; Keith Wafford; Trevor G Smart
Journal:  J Physiol       Date:  2010-02-22       Impact factor: 5.182

3.  Stereoselective central nervous system effects of the R- and S-isomers of the GABA uptake blocker N-(4, 4-di-(3-methylthien-2-yl)but-3-enyl) nipecotic acid in the rat.

Authors:  A Cleton; H J de Greef; P M Edelbroek; R A Voskuyl; M Danhof
Journal:  Br J Pharmacol       Date:  1999-12       Impact factor: 8.739

4.  Vigabatrin transport across the human intestinal epithelial (Caco-2) brush-border membrane is via the H+ -coupled amino-acid transporter hPAT1.

Authors:  Emily L Abbot; Danielle S Grenade; David J Kennedy; Kelly M Gatfield; David T Thwaites
Journal:  Br J Pharmacol       Date:  2006-02       Impact factor: 8.739

5.  3-Aminopropylphosphinic acid--a potent, selective GABAB receptor agonist in the guinea-pig ileum and rat anococcygeus muscle.

Authors:  J M Hills; R A Dingsdale; M E Parsons; R E Dolle; W Howson
Journal:  Br J Pharmacol       Date:  1989-08       Impact factor: 8.739

6.  GABA receptors on the somatic muscle cells of the parasitic nematode, Ascaris suum: stereoselectivity indicates similarity to a GABAA-type agonist recognition site.

Authors:  L Holden-Dye; P Krogsgaard-Larsen; L Nielsen; R J Walker
Journal:  Br J Pharmacol       Date:  1989-11       Impact factor: 8.739

7.  Beta-methyl carboline, a benzodiazepine inverse agonist, attenuates the effect of triazolam on the circadian rhythm of locomotor activity.

Authors:  R D Smith; F W Turek
Journal:  Experientia       Date:  1989-04-15

8.  Pharmacology of GABA rho 1 and GABA alpha/beta receptors expressed in Xenopus oocytes and COS cells.

Authors:  T Kusama; C E Spivak; P Whiting; V L Dawson; J C Schaeffer; G R Uhl
Journal:  Br J Pharmacol       Date:  1993-05       Impact factor: 8.739

9.  Central administration of muscimol phase-shifts the mammalian circadian clock.

Authors:  R D Smith; S Inouye; F W Turek
Journal:  J Comp Physiol A       Date:  1989-02       Impact factor: 1.836

10.  N-Substituted Nipecotic Acids as (S)-SNAP-5114 Analogues with Modified Lipophilic Domains.

Authors:  Michael C Böck; Georg Höfner; Klaus T Wanner
Journal:  ChemMedChem       Date:  2020-04-07       Impact factor: 3.466
  10 in total

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