Literature DB >> 32374500

Pregabalin poisoning and rising recreational use: a retrospective observational series.

Katherine Z Isoardi1,2,3, Gregory Polkinghorne1,2, Keith Harris1,2, Geoffrey K Isbister3,4.   

Abstract

AIMS: With rising use worldwide, pregabalin is increasingly implicated in poisoning deaths. We aimed to investigate the clinical effects and complications of pregabalin poisoning.
METHODS: This is a retrospective review of patients presenting with pregabalin poisoning to two tertiary toxicology units from 1 July 2014 to 30 June 2019. Patients were identified from prospective databases maintained by both units and data were extracted from these in addition to medical records.
RESULTS: There were 488 presentations in 413 patients (237 [57%] male) over the five-year period. The median age was 41 years (IQR 31-50 years). Deliberate self-poisonings accounted for 342 (70%) presentations, with 121 (25%) recreational exposures. Recreational exposures increased over the period from 2 (4%) in the first year to 54 (39%) presentations in the final year. The median dose of pregabalin was 1200 mg (IQR 600-3000 mg, range 75-16 800 mg). Co-ingestions occurred in 427 (88%) presentations, with sedating agents being co-ingested in 387 (79%)-most commonly opioids and benzodiazepines in 201 (41%) and 174 (36%) presentations respectively. Coma (GCS < 9) occurred in 89 (18%) cases, with 52 (11%) patients being intubated. Only one (0.2%) of these patients had not co-ingested a sedating agent. Hypotension occurred in 26 (5%) cases, all with co-ingestants. Seizures occurred in 11 (2%) cases, 3/59 (5%) in pregabalin-only overdoses. The median length of stay was 16.5 hours (IQR 10-25 hours).
CONCLUSIONS: Pregabalin overdose does not cause severe toxicity, but rather mild sedation and, uncommonly, seizures. Coma is common in the presence of sedating co-ingestants. Recreational use is increasing.
© 2020 The British Pharmacological Society.

Entities:  

Keywords:  drug abuse; overdose and poisoning; toxicology

Mesh:

Substances:

Year:  2020        PMID: 32374500      PMCID: PMC7688538          DOI: 10.1111/bcp.14348

Source DB:  PubMed          Journal:  Br J Clin Pharmacol        ISSN: 0306-5251            Impact factor:   4.335


  18 in total

1.  Significant pregabalin toxicity managed with supportive care alone.

Authors:  David M Wood; David J Berry; Guy Glover; Jane Eastwood; Paul I Dargan
Journal:  J Med Toxicol       Date:  2010-12

Review 2.  Abuse and Misuse of Pregabalin and Gabapentin.

Authors:  Kirk E Evoy; Megan D Morrison; Stephen R Saklad
Journal:  Drugs       Date:  2017-03       Impact factor: 9.546

3.  Pharmacokinetic-pharmacodynamic modelling of QT interval prolongation following citalopram overdoses.

Authors:  Lena E Friberg; Geoffrey K Isbister; Stephen B Duffull
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Journal:  Drug Alcohol Depend       Date:  2017-02-28       Impact factor: 4.492

5.  Pregabalin misuse-related ambulance attendances in Victoria, 2012-2017: characteristics of patients and attendances.

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9.  Activated charcoal decreases the risk of QT prolongation after citalopram overdose.

Authors:  Geoffrey K Isbister; Lena E Friberg; Barrie Stokes; Nicholas A Buckley; Christopher Lee; Naren Gunja; Simon G Brown; Ellen MacDonald; Andis Graudins; Anna Holdgate; Stephen B Duffull
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10.  Intentional Drug Overdose Involving Pregabalin and Gabapentin: Findings from the National Self-Harm Registry Ireland, 2007-2015.

Authors:  Caroline Daly; Eve Griffin; Darren M Ashcroft; Roger T Webb; Ivan J Perry; Ella Arensman
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2.  Pregabalin poisoning and rising recreational use: a retrospective observational series.

Authors:  Katherine Z Isoardi; Gregory Polkinghorne; Keith Harris; Geoffrey K Isbister
Journal:  Br J Clin Pharmacol       Date:  2020-06-05       Impact factor: 4.335

3.  Pregabalin poisoning: Evaluation of dose-toxicity relationship.

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