Literature DB >> 32296759

Editorial for Advances in G Protein-Coupled Receptor Signal Transduction Special Issue.

Andrew B Tobin1, Sophie J Bradley1.   

Abstract

Year:  2020        PMID： 32296759      PMCID： PMC7155192          DOI： 10.1021/acsptsci.0c00029

Source DB:  PubMed          Journal:  ACS Pharmacol Transl Sci        ISSN： 2575-9108


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  7 in total

1.  Quantification of ligand bias for clinically relevant β2-adrenergic receptor ligands: implications for drug taxonomy.

Authors:  Emma T van der Westhuizen; Billy Breton; Arthur Christopoulos; Michel Bouvier
Journal:  Mol Pharmacol       Date:  2013-12-23       Impact factor: 4.436

2.  Quantifying ligand bias at seven-transmembrane receptors.

Authors:  Sudarshan Rajagopal; Seungkirl Ahn; David H Rominger; William Gowen-MacDonald; Christopher M Lam; Scott M Dewire; Jonathan D Violin; Robert J Lefkowitz
Journal:  Mol Pharmacol       Date:  2011-05-24       Impact factor: 4.436

Review 3.  Signalling bias in new drug discovery: detection, quantification and therapeutic impact.

Authors:  Terry Kenakin; Arthur Christopoulos
Journal:  Nat Rev Drug Discov       Date:  2012-02-15       Impact factor: 84.694

Review 4.  Biased signalling: from simple switches to allosteric microprocessors.

Authors:  Jeffrey S Smith; Robert J Lefkowitz; Sudarshan Rajagopal
Journal:  Nat Rev Drug Discov       Date:  2018-01-05       Impact factor: 84.694

5.  Biased M1-muscarinic-receptor-mutant mice inform the design of next-generation drugs.

Authors:  Sophie J Bradley; Colin Molloy; Paulina Valuskova; Louis Dwomoh; Miriam Scarpa; Mario Rossi; Lisa Finlayson; Kjell A Svensson; Eyassu Chernet; Vanessa N Barth; Karolina Gherbi; David A Sykes; Caroline A Wilson; Rajendra Mistry; Patrick M Sexton; Arthur Christopoulos; Adrian J Mogg; Elizabeth M Rosethorne; Shuzo Sakata; R A John Challiss; Lisa M Broad; Andrew B Tobin
Journal:  Nat Chem Biol       Date:  2020-02-20       Impact factor: 15.040

Review 6.  Molecular mechanism of β-arrestin-biased agonism at seven-transmembrane receptors.

Authors:  Eric Reiter; Seungkirl Ahn; Arun K Shukla; Robert J Lefkowitz
Journal:  Annu Rev Pharmacol Toxicol       Date:  2011-09-19       Impact factor: 13.820

Review 7.  Location, location, location...site-specific GPCR phosphorylation offers a mechanism for cell-type-specific signalling.

Authors:  Andrew B Tobin; Adrian J Butcher; Kok Choi Kong
Journal:  Trends Pharmacol Sci       Date:  2008-07-06       Impact factor: 14.819
  7 in total

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