Literature DB >> 32034430

Expression of fibroblast growth factor receptor 4 and clinical response to lenvatinib in patients with anaplastic thyroid carcinoma: a pilot study.

Haruhiko Yamazaki1, Tomoyuki Yokose2, Hiroyuki Hayashi2, Hiroyuki Iwasaki3, Sachie Osanai2, Nobuyasu Suganuma3, Hirotaka Nakayama4, Katsuhiko Masudo5, Yasushi Rino4, Munetaka Masuda4.   

Abstract

PURPOSE: Fibroblast growth factor receptor 4 (FGFR4) expression has association with tumor malignancy. In thyroid cancers, FGFR4 has been reported to be characteristically expressed in aggressive thyroid tumors, such as anaplastic thyroid carcinoma (ATC).
METHODS: We investigated FGFR4 expression in patients with ATC and analyzed their clinical responses to lenvatinib. Primary tumor samples were obtained from 12 patients with ATC who underwent surgery or core needle biopsy. FGFR4 protein expression in all ATC samples was analyzed via immunohistochemistry, and the treatment efficacy of lenvatinib was evaluated.
RESULTS: The proportion of FGFR4-positive cells in the samples ranged from 0 to 50%. Four patients had partial responses, and three patients had stable diseases as a best clinical response to lenvatinib. The median PFS durations of patients with none, weak, and moderate intensity were 0.5, 3.2 (95% CI 1.1-not estimable [NE]), and 4.6 (95% CI 1.1-NE) months, respectively (p = 0.003).
CONCLUSIONS: Because FGFR4 was expressed in ATC tissues, the FGFR4 expression might be associated with the treatment efficacy of lenvatinib in a part of ATC patients. To clarify whether FGFR4 can serve as a prognostic or predictive factor for lenvatinib therapy, more cases must be accumulated.

Entities:  

Keywords:  Clinical research; Fibroblast growth factor receptor; Lenvatinib; Molecular biology; Thyroid cancer

Mesh:

Substances:

Year:  2020        PMID: 32034430     DOI: 10.1007/s00228-020-02842-y

Source DB:  PubMed          Journal:  Eur J Clin Pharmacol        ISSN: 0031-6970            Impact factor:   2.953


  40 in total

Review 1.  Roles of fibroblast growth factor receptors in carcinogenesis.

Authors:  Ellen Margrethe Haugsten; Antoni Wiedlocha; Sjur Olsnes; Jørgen Wesche
Journal:  Mol Cancer Res       Date:  2010-10-13       Impact factor: 5.852

2.  Thyroid cancer incidence patterns in the United States by histologic type, 1992-2006.

Authors:  Briseis Aschebrook-Kilfoy; Mary H Ward; Mona M Sabra; Susan S Devesa
Journal:  Thyroid       Date:  2010-12-27       Impact factor: 6.568

3.  Fibroblast growth factor receptor 4 as a potential prognostic and therapeutic marker in colorectal cancer.

Authors:  Chen-Sheng Li; Shu-Xiang Zhang; Hong-Jun Liu; Yu-Long Shi; Le-Ping Li; Xiao-Bo Guo; Zhen-Hai Zhang
Journal:  Biomarkers       Date:  2014-01-13       Impact factor: 2.658

4.  Dual inhibition of RET and FGFR4 restrains medullary thyroid cancer cell growth.

Authors:  Shereen Ezzat; Ping Huang; Alan Dackiw; Sylvia L Asa
Journal:  Clin Cancer Res       Date:  2005-02-01       Impact factor: 12.531

5.  Exploratory analysis of biomarkers associated with clinical outcomes from the study of lenvatinib in differentiated cancer of the thyroid.

Authors:  Makoto Tahara; Martin Schlumberger; Rossella Elisei; Mouhammed Amir Habra; Naomi Kiyota; Ralf Paschke; Corina E Dutcus; Taro Hihara; Shannon McGrath; Mark Matijevic; Tadashi Kadowaki; Yasuhiro Funahashi; Steven I Sherman
Journal:  Eur J Cancer       Date:  2017-02-24       Impact factor: 9.162

6.  Expression of fibroblast growth factor-2 and fibroblast growth factor receptor-1 in thyroid diseases: difference between neoplasms and hyperplastic lesions.

Authors:  K Shingu; M Fujimori; K Ito; Y Hama; Y Kasuga; S Kobayashi; N Itoh; J Amano
Journal:  Endocr J       Date:  1998-02       Impact factor: 2.349

7.  Long-term results of radiotherapy in anaplastic thyroid cancer.

Authors:  Anne-Katrin Dumke; Tanja Pelz; Dirk Vordermark
Journal:  Radiat Oncol       Date:  2014-03-31       Impact factor: 3.481

8.  Fibroblast growth factor receptor 4: a putative key driver for the aggressive phenotype of hepatocellular carcinoma.

Authors:  Christine Gauglhofer; Jakob Paur; Waltraud C Schrottmaier; Bettina Wingelhofer; Daniela Huber; Isabelle Naegelen; Christine Pirker; Thomas Mohr; Christine Heinzle; Klaus Holzmann; Brigitte Marian; Rolf Schulte-Hermann; Walter Berger; Georg Krupitza; Michael Grusch; Bettina Grasl-Kraupp
Journal:  Carcinogenesis       Date:  2014-07-16       Impact factor: 4.944

9.  FGFR4 role in epithelial-mesenchymal transition and its therapeutic value in colorectal cancer.

Authors:  Alberto Peláez-García; Rodrigo Barderas; Sofía Torres; Pablo Hernández-Varas; Joaquín Teixidó; Félix Bonilla; Antonio Garcia de Herreros; J Ignacio Casal
Journal:  PLoS One       Date:  2013-05-16       Impact factor: 3.240

10.  Fibroblast growth factor receptor-2 expression in thyroid tumor progression: potential diagnostic application.

Authors:  Adriano Redler; Giorgio Di Rocco; Domenico Giannotti; Francesca Frezzotti; Maria Giulia Bernieri; Simona Ceccarelli; Sirio D'Amici; Enrica Vescarelli; Anna Paola Mitterhofer; Antonio Angeloni; Cinzia Marchese
Journal:  PLoS One       Date:  2013-08-19       Impact factor: 3.240

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  4 in total

1.  Inflammatory biomarkers and dynamics of neutrophil-to-lymphocyte ratio in lenvatinib treatment for anaplastic thyroid carcinoma.

Authors:  Haruhiko Yamazaki; Hiroyuki Iwasaki; Nobuyasu Suganuma; Soji Toda; Katsuhiko Masudo; Hirotaka Nakayama; Yasushi Rino; Munetaka Masuda
Journal:  Gland Surg       Date:  2021-03

2.  Efficacy and Safety of Lenvatinib in Anaplastic Thyroid Carcinoma: A Meta-Analysis.

Authors:  Dongmei Huang; Jinming Zhang; Xiangqian Zheng; Ming Gao
Journal:  Front Endocrinol (Lausanne)       Date:  2022-06-30       Impact factor: 6.055

3.  Thyroid Hormone Receptor Beta Inhibits PI3K-Akt-mTOR Signaling Axis in Anaplastic Thyroid Cancer via Genomic Mechanisms.

Authors:  Cole D Davidson; Eric L Bolf; Noelle E Gillis; Lauren M Cozzens; Jennifer A Tomczak; Frances E Carr
Journal:  J Endocr Soc       Date:  2021-06-01

4.  FGF-Receptors and PD-L1 in Anaplastic and Poorly Differentiated Thyroid Cancer: Evaluation of the Preclinical Rationale.

Authors:  Pia Adam; Stefan Kircher; Iuliu Sbiera; Viktoria Florentine Koehler; Elke Berg; Thomas Knösel; Benjamin Sandner; Wiebke Kristin Fenske; Hendrik Bläker; Constantin Smaxwil; Andreas Zielke; Bence Sipos; Stephanie Allelein; Matthias Schott; Christine Dierks; Christine Spitzweg; Martin Fassnacht; Matthias Kroiss
Journal:  Front Endocrinol (Lausanne)       Date:  2021-08-12       Impact factor: 5.555

  4 in total

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