Literature DB >> 32009149

A phase I/II study of veliparib (ABT-888) with radiation and temozolomide in newly diagnosed diffuse pontine glioma: a Pediatric Brain Tumor Consortium study.

Patricia A Baxter1, Jack M Su1, Arzu Onar-Thomas2, Catherine A Billups2, Xiao-Nan Li1, Tina Young Poussaint3, Edward R Smith3, Patrick Thompson4, Adekunle Adesina1, Pete Ansell5, Vincent Giranda5, Arnold Paulino6, Lindsey Kilburn7, Ibrahim Quaddoumi2, Alberto Broniscer2, Susan M Blaney1, Ira J Dunkel8, Maryam Fouladi9.   

Abstract

BACKGROUND: A Pediatric Brain Tumor Consortium (PBTC) phase I/II trial of veliparib and radiation followed by veliparib and temozolomide (TMZ) was conducted in children with newly diagnosed diffuse intrinsic pontine glioma (DIPG). The objectives were to: (i) estimate the recommended phase II dose (RP2D) of veliparib with concurrent radiation; (ii) evaluate the pharmacokinetic parameters of veliparib during radiation; (iii) evaluate feasibility of intrapatient TMZ dose escalation; (iv) describe toxicities of protocol therapy; and (v) estimate the overall survival distribution compared with historical series.
METHODS: Veliparib was given Monday through Friday b.i.d. during radiation followed by a 4-week rest. Patients then received veliparib at 25 mg/m2 b.i.d. and TMZ 135 mg/m2 daily for 5 days every 28 days. Intrapatient dose escalation of TMZ was investigated for patients experiencing minimal toxicity.
RESULTS: Sixty-six patients (65 eligible) were enrolled. The RP2D of veliparib was 65 mg/m2 b.i.d. with radiation. Dose-limiting toxicities during radiation with veliparib therapy included: grade 2 intratumoral hemorrhage (n = 1), grade 3 maculopapular rash (n = 2), and grade 3 nervous system disorder (generalized neurologic deterioration) (n = 1). Intrapatient TMZ dose escalation during maintenance was not tolerated. Following a planned interim analysis, it was concluded that this treatment did not show a survival benefit compared with PBTC historical controls, and accrual was stopped for futility. The 1- and 2-year overall survival rates were 37.2% (SE 7%) and 5.3% (SE 3%), respectively.
CONCLUSION: Addition of veliparib to radiation followed by TMZ and veliparib was tolerated but did not improve survival for patients with newly diagnosed DIPG. TRIAL REGISTRATION: NCT01514201.
© The Author(s) 2020. Published by Oxford University Press on behalf of the Society for Neuro-Oncology. All rights reserved. For permissions, please e-mail: journals.permissions@oup.com.

Entities:  

Keywords:  ABT-888; CNS tumors; DIPG; PARP inhibition; veliparib

Mesh:

Substances:

Year:  2020        PMID: 32009149      PMCID: PMC7283021          DOI: 10.1093/neuonc/noaa016

Source DB:  PubMed          Journal:  Neuro Oncol        ISSN: 1522-8517            Impact factor:   12.300


  44 in total

1.  Monitoring event times in early phase clinical trials: some practical issues.

Authors:  Peter F Thall; Leiko H Wooten; Nizar M Tannir
Journal:  Clin Trials       Date:  2005       Impact factor: 2.486

2.  Predicting outcome of children with diffuse intrinsic pontine gliomas using multiparametric imaging.

Authors:  Sean J Hipp; Emilie Steffen-Smith; Dima Hammoud; Joanna H Shih; Robyn Bent; Katherine E Warren
Journal:  Neuro Oncol       Date:  2011-07-13       Impact factor: 12.300

3.  Automated Processing of Dynamic Contrast-Enhanced MRI: Correlation of Advanced Pharmacokinetic Metrics with Tumor Grade in Pediatric Brain Tumors.

Authors:  S Vajapeyam; C Stamoulis; K Ricci; M Kieran; T Young Poussaint
Journal:  AJNR Am J Neuroradiol       Date:  2016-09-15       Impact factor: 3.825

4.  Veliparib in combination with whole brain radiation therapy in patients with brain metastases: results of a phase 1 study.

Authors:  Minesh P Mehta; Ding Wang; Fen Wang; Lawrence Kleinberg; Anthony Brade; H Ian Robins; Aruna Turaka; Terri Leahy; Diane Medina; Hao Xiong; Nael M Mostafa; Martin Dunbar; Ming Zhu; Jane Qian; Kyle Holen; Vincent Giranda; Walter J Curran
Journal:  J Neurooncol       Date:  2015-02-15       Impact factor: 4.130

5.  Whole-genome profiling of pediatric diffuse intrinsic pontine gliomas highlights platelet-derived growth factor receptor alpha and poly (ADP-ribose) polymerase as potential therapeutic targets.

Authors:  Maryam Zarghooni; Ute Bartels; Eric Lee; Pawel Buczkowicz; Andrew Morrison; Annie Huang; Eric Bouffet; Cynthia Hawkins
Journal:  J Clin Oncol       Date:  2010-02-08       Impact factor: 44.544

6.  A phase I trial of veliparib (ABT-888) and temozolomide in children with recurrent CNS tumors: a pediatric brain tumor consortium report.

Authors:  Jack M Su; Patrick Thompson; Adekunle Adesina; Xiao-Nan Li; Lindsay Kilburn; Arzu Onar-Thomas; Mehmet Kocak; Brenda Chyla; Evelyn McKeegan; Katherine E Warren; Stewart Goldman; Ian F Pollack; Maryam Fouladi; Alice Chen; Vincent Giranda; James Boyett; Larry Kun; Susan M Blaney
Journal:  Neuro Oncol       Date:  2014-06-07       Impact factor: 12.300

7.  Poly-ADP-Ribose Polymerase as a Therapeutic Target in Pediatric Diffuse Intrinsic Pontine Glioma and Pediatric High-Grade Astrocytoma.

Authors:  Yevgen Chornenkyy; Sameer Agnihotri; Man Yu; Pawel Buczkowicz; Patricia Rakopoulos; Brian Golbourn; Livia Garzia; Robert Siddaway; Stephie Leung; James T Rutka; Michael D Taylor; Peter B Dirks; Cynthia Hawkins
Journal:  Mol Cancer Ther       Date:  2015-09-08       Impact factor: 6.261

8.  MRI as a central component of clinical trials analysis in brainstem glioma: a report from the Pediatric Brain Tumor Consortium (PBTC).

Authors:  Tina Young Poussaint; Mehmet Kocak; Sridhar Vajapeyam; Roger I Packer; Richard L Robertson; Russell Geyer; Daphne Haas-Kogan; Ian F Pollack; Gilbert Vezina; Robert Zimmerman; Soonmee Cha; Zoltan Patay; James M Boyett; Larry E Kun
Journal:  Neuro Oncol       Date:  2011-02-04       Impact factor: 12.300

Review 9.  Poly (ADP-ribose) polymerase inhibitors: recent advances and future development.

Authors:  Clare L Scott; Elizabeth M Swisher; Scott H Kaufmann
Journal:  J Clin Oncol       Date:  2015-03-16       Impact factor: 44.544

Review 10.  The role of poly(ADP-ribosyl)ation in DNA damage response and cancer chemotherapy.

Authors:  M Li; X Yu
Journal:  Oncogene       Date:  2014-09-15       Impact factor: 9.867

View more
  16 in total

Review 1.  PARkinson's: From cellular mechanisms to potential therapeutics.

Authors:  Zsofia Lengyel-Zhand; Laura N Puentes; Robert H Mach
Journal:  Pharmacol Ther       Date:  2021-08-12       Impact factor: 12.310

Review 2.  The Role of PARP Inhibitors in Patients with Primary Malignant Central Nervous System Tumors.

Authors:  Susan E Gueble; Juan C Vasquez; Ranjit S Bindra
Journal:  Curr Treat Options Oncol       Date:  2022-10-15

Review 3.  Medulloblastoma drugs in development: Current leads, trials and drawbacks.

Authors:  Jiachen Wen; M Kyle Hadden
Journal:  Eur J Med Chem       Date:  2021-02-08       Impact factor: 6.514

4.  PARP-mediated PARylation of MGMT is critical to promote repair of temozolomide-induced O6-methylguanine DNA damage in glioblastoma.

Authors:  Shaofang Wu; Xiaolong Li; Feng Gao; John F de Groot; Dimpy Koul; W K Alfred Yung
Journal:  Neuro Oncol       Date:  2021-06-01       Impact factor: 12.300

5.  Blocking PARP activity with the inhibitor veliparib enhances radiotherapy sensitivity in endometrial carcinoma.

Authors:  Jing Wang; Weizhen Xing; Yanling Lin; Nuray Uskenbayeva; Hongchao Yan; Yang Xu; Lisha Fang
Journal:  J Clin Lab Anal       Date:  2022-04-14       Impact factor: 3.124

6.  Non-invasive Urinary Biomarkers in Moyamoya Disease.

Authors:  Julie Sesen; Jessica Driscoll; Alexander Moses-Gardner; Darren B Orbach; David Zurakowski; Edward R Smith
Journal:  Front Neurol       Date:  2021-04-01       Impact factor: 4.003

Review 7.  DNA damage repair: historical perspectives, mechanistic pathways and clinical translation for targeted cancer therapy.

Authors:  Ruixue Huang; Ping-Kun Zhou
Journal:  Signal Transduct Target Ther       Date:  2021-07-09

Review 8.  Radiation in Combination With Targeted Agents and Immunotherapies for Pediatric Central Nervous System Tumors - Progress, Opportunities, and Challenges.

Authors:  Bo Qiu; Cassie Kline; Sabine Mueller
Journal:  Front Oncol       Date:  2021-06-30       Impact factor: 6.244

9.  Glioblastoma multiforme (GBM): An overview of current therapies and mechanisms of resistance.

Authors:  Wei Wu; Jessica L Klockow; Michael Zhang; Famyrah Lafortune; Edwin Chang; Linchun Jin; Yang Wu; Heike E Daldrup-Link
Journal:  Pharmacol Res       Date:  2021-07-21       Impact factor: 10.334

Review 10.  DDRugging glioblastoma: understanding and targeting the DNA damage response to improve future therapies.

Authors:  Ola Rominiyi; Spencer J Collis
Journal:  Mol Oncol       Date:  2021-06-11       Impact factor: 6.603

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.