Literature DB >> 31209792

Trifluridine/Tipiracil (TAS-102) for refractory metastatic colorectal cancer in clinical practice: a feasible alternative for patients with good performance status.

C Carriles1, P Jimenez-Fonseca2, M Sánchez-Cánovas3, P Pimentel4, A Carmona-Bayonas3, T García4, M Carbajales-Álvarez5, A Lozano-Blázquez5.   

Abstract

INTRODUCTION: Our aim was to assess efficacy and safety and prognostic factors associated with TAS-102 in clinical practice.
METHOD: Retrospective, multicenter, and observational study including patients with advanced refractory colorectal cancer who started TAS-102 between March 2016 and August 2018. The primary end point was overall survival (OS). Secondary end points included progression-free survival, toxicity and analyze prognostic factors present at the beginning of TAS-102. RESULT: 84 patients were evaluable. The median OS was 8.30 (95% CI 6.23-9.87) months and PFS was 2.62 (95% CI 2.36-3.05) months. In multivariate analysis, ECOG 0 and reduced dose combined with more cycles were associated with better prognosis. Patients with an ECOG > 0 had worse prognosis (HR 3.34, 95% CI 1.09-10.27, p = 0.035). 95.2% experienced some type of adverse effect and 45.2% had grade ≥ 3 toxicities.
CONCLUSION: Results suggest reconsidering TAS-102 in patients with ECOG > 0, something that should be investigated in prospective randomized clinical trials.

Entities:  

Keywords:  ECOG; Multivariate; PROGNOSIS; Progression-free survival; Survival; Toxicity

Mesh:

Substances:

Year:  2019        PMID: 31209792     DOI: 10.1007/s12094-019-02154-3

Source DB:  PubMed          Journal:  Clin Transl Oncol        ISSN: 1699-048X            Impact factor:   3.405


  10 in total

1.  Trifluridine/Tipiracil (TAS-102) in Refractory Metastatic Colorectal Cancer: A Multicenter Register in the Frame of the Italian Compassionate Use Program.

Authors:  Chiara Cremolini; Daniele Rossini; Erika Martinelli; Filippo Pietrantonio; Sara Lonardi; Silvia Noventa; Emiliano Tamburini; Giovanni Luca Frassineti; Stefania Mosconi; Federico Nichetti; Sabina Murgioni; Teresa Troiani; Beatrice Borelli; Gemma Zucchelli; Alessandro Dal Maso; Vincenzo Sforza; Gianluca Masi; Carlotta Antoniotti; Maria Di Bartolomeo; Rosalba Miceli; Fortunato Ciardiello; Alfredo Falcone
Journal:  Oncologist       Date:  2018-05-08

2.  Randomized trial of TAS-102 for refractory metastatic colorectal cancer.

Authors:  Robert J Mayer; Eric Van Cutsem; Alfredo Falcone; Takayuki Yoshino; Rocio Garcia-Carbonero; Nobuyuki Mizunuma; Kentaro Yamazaki; Yasuhiro Shimada; Josep Tabernero; Yoshito Komatsu; Alberto Sobrero; Eveline Boucher; Marc Peeters; Ben Tran; Heinz-Josef Lenz; Alberto Zaniboni; Howard Hochster; James M Cleary; Hans Prenen; Fabio Benedetti; Hirokazu Mizuguchi; Lukas Makris; Masanobu Ito; Atsushi Ohtsu
Journal:  N Engl J Med       Date:  2015-05-14       Impact factor: 91.245

3.  Safety and Efficacy of Trifluridine/Tipiracil Monotherapy in Clinical Practice for Patients With Metastatic Colorectal Cancer: Experience at a Single Institution.

Authors:  Daisuke Kotani; Kohei Shitara; Akihito Kawazoe; Shota Fukuoka; Yasutoshi Kuboki; Hideaki Bando; Wataru Okamoto; Takashi Kojima; Toshihiko Doi; Atsushi Ohtsu; Takayuki Yoshino
Journal:  Clin Colorectal Cancer       Date:  2015-11-27       Impact factor: 4.481

4.  Regorafenib monotherapy for previously treated metastatic colorectal cancer (CORRECT): an international, multicentre, randomised, placebo-controlled, phase 3 trial.

Authors:  Axel Grothey; Eric Van Cutsem; Alberto Sobrero; Salvatore Siena; Alfredo Falcone; Marc Ychou; Yves Humblet; Olivier Bouché; Laurent Mineur; Carlo Barone; Antoine Adenis; Josep Tabernero; Takayuki Yoshino; Heinz-Josef Lenz; Richard M Goldberg; Daniel J Sargent; Frank Cihon; Lisa Cupit; Andrea Wagner; Dirk Laurent
Journal:  Lancet       Date:  2012-11-22       Impact factor: 79.321

5.  Optimizing Treatment Sequence for Late-line Metastatic Colorectal Cancer Patients Using Trifluridine/Tipiracil and Regorafenib.

Authors:  Matthias Unseld; Magdalena Drimmel; Alexander Siebenhüner; Andreas Gleiss; Daniela Bianconi; Markus Kieler; Werner Scheithauer; Thomas Winder; Gerald W Prager
Journal:  Clin Colorectal Cancer       Date:  2018-06-08       Impact factor: 4.481

6.  ESMO consensus guidelines for the management of patients with metastatic colorectal cancer.

Authors:  E Van Cutsem; A Cervantes; R Adam; A Sobrero; J H Van Krieken; D Aderka; E Aranda Aguilar; A Bardelli; A Benson; G Bodoky; F Ciardiello; A D'Hoore; E Diaz-Rubio; J-Y Douillard; M Ducreux; A Falcone; A Grothey; T Gruenberger; K Haustermans; V Heinemann; P Hoff; C-H Köhne; R Labianca; P Laurent-Puig; B Ma; T Maughan; K Muro; N Normanno; P Österlund; W J G Oyen; D Papamichael; G Pentheroudakis; P Pfeiffer; T J Price; C Punt; J Ricke; A Roth; R Salazar; W Scheithauer; H J Schmoll; J Tabernero; J Taïeb; S Tejpar; H Wasan; T Yoshino; A Zaanan; D Arnold
Journal:  Ann Oncol       Date:  2016-07-05       Impact factor: 32.976

7.  Phase I study of TAS-102 treatment in Japanese patients with advanced solid tumours.

Authors:  T Doi; A Ohtsu; T Yoshino; N Boku; Y Onozawa; A Fukutomi; S Hironaka; W Koizumi; T Sasaki
Journal:  Br J Cancer       Date:  2012-06-26       Impact factor: 7.640

8.  Feasibility and effectiveness of trifluridine/tipiracil in metastatic colorectal cancer: real-life data from The Netherlands.

Authors:  Johannes J M Kwakman; G Vink; J H Vestjens; L V Beerepoot; J W de Groot; R L Jansen; F L Opdam; H Boot; G J Creemers; J M van Rooijen; M Los; A J E Vulink; H Schut; E van Meerten; A Baars; P Hamberg; E Kapiteijn; D W Sommeijer; C J A Punt; M Koopman
Journal:  Int J Clin Oncol       Date:  2017-12-04       Impact factor: 3.402

9.  Clinical outcome of patients with chemorefractory metastatic colorectal cancer treated with trifluridine/tipiracil (TAS-102): a single Italian institution compassionate use programme.

Authors:  Vincenzo Sforza; Erika Martinelli; Claudia Cardone; Giulia Martini; Stefania Napolitano; Pietro Paolo Vitiello; Pasquale Vitale; Nicoletta Zanaletti; Alfonso Reginelli; Maurizio Di Bisceglie; Tiziana Pia Latiano; Anna Maria Bochicchio; Fabiana Cecere; Francesco Selvaggi; Fortunato Ciardiello; Teresa Troiani
Journal:  ESMO Open       Date:  2017-09-21

10.  Efficacy of trifluridine and tipiracil (TAS-102) versus placebo, with supportive care, in a randomized, controlled trial of patients with metastatic colorectal cancer from Spain: results of a subgroup analysis of the phase 3 RECOURSE trial.

Authors:  F Longo-Muñoz; G Argiles; J Tabernero; A Cervantes; C Gravalos; C Pericay; S Gil-Calle; H Mizuguchi; A Carrato-Mena; M L Limón; R Garcia-Carbonero
Journal:  Clin Transl Oncol       Date:  2016-07-21       Impact factor: 3.405

  10 in total
  1 in total

Review 1.  TAS-102 Monotherapy and Combination Therapy with Bevacizumab for Metastatic Colorectal Cancer.

Authors:  Cheng-Jiang Liu; Ting Hu; Ping Shao; Wu-Yang Chu; Yu Cao; Feng Zhang
Journal:  Gastroenterol Res Pract       Date:  2021-12-20       Impact factor: 2.260

  1 in total

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