Literature DB >> 30583040

Decreasing the Toxicity of Radiation Therapy: Radioprotectors and Radiomitigators Being Developed by the National Cancer Institute Through Small Business Innovation Research Contracts.

Kaveh Zakeri1, Deepa Narayanan2, Bhadrasain Vikram3, Greg Evans2, C Norman Coleman3, Pataje G S Prasanna4.   

Abstract

PURPOSE: The use of radioprotectors and radiomitigators could improve the therapeutic index of radiation therapy. With the intention of accelerating translation of radiation-effect modulators (radioprotectors and mitigators), the Radiation Research Program and SBIR (Small Business Innovation Research) Development Center within the National Cancer Institute issued 4 Requests for Proposals (RFPs) from 2010 to 2013. Twelve SBIR contract awards in total were made in response to the 4 RFPs from September 2011 through September 2014. Here, we provide an update on the status of SBIR contract projects for the development of radiation-effect modulators. METHODS AND MATERIALS: To assess the status of research and development efforts under the 4 RFPs on radiation-effect modulators, we searched PubMed for research articles, google.com for published abstracts, clinicaltrials.gov for ongoing or completed clinical trials, and company websites for press releases and other news. All information obtained and reported here is publicly available and thus protects the intellectual property of the investigators and companies.
RESULTS: Of the 12 SBIR projects funded, 5 (42%) transitioned successfully from phase 1 to phase 2 SBIR funding, and among the Fast-Track contracts, this rate was 100% (3 of 3). The Internet search identified 3 abstracts and 6 publications related to the aims of the SBIR contracts. One-third of the companies (4 of 12) have successfully launched a total of 8 clinical trials to demonstrate the safety and efficacy of their investigational agents. Two drugs are in clinical trials for their indication as a radioprotector, and 2 drugs are under evaluation for their anticancer properties (an immunomodulator and a small molecule inhibitor).
CONCLUSIONS: The National Cancer Institute's SBIR has provided pivotal funding to small businesses for the development of radioprotectors and radiomitigators, which resulted in multiple early-phase clinical trials. Longer follow-up is needed to determine the full impact of these novel therapeutics that enter clinical practice. Published by Elsevier Inc.

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Mesh:

Year:  2018        PMID: 30583040      PMCID: PMC6458068          DOI: 10.1016/j.ijrobp.2018.12.027

Source DB:  PubMed          Journal:  Int J Radiat Oncol Biol Phys        ISSN: 0360-3016            Impact factor:   7.038


  10 in total

Review 1.  Development of investigational radiation modifiers.

Authors:  A Dimitrios Colevas; J Martin Brown; Stephen Hahn; James Mitchell; Kevin Camphausen; C Norman Coleman
Journal:  J Natl Cancer Inst       Date:  2003-05-07       Impact factor: 13.506

2.  Toll-like receptor 5 agonist protects mice from dermatitis and oral mucositis caused by local radiation: implications for head-and-neck cancer radiotherapy.

Authors:  Lyudmila G Burdelya; Anatoli S Gleiberman; Ilia Toshkov; Semra Aygun-Sunar; Meghana Bapardekar; Patricia Manderscheid-Kern; David Bellnier; Vadim I Krivokrysenko; Elena Feinstein; Andrei V Gudkov
Journal:  Int J Radiat Oncol Biol Phys       Date:  2011-10-14       Impact factor: 7.038

3.  A Phase I Study of ABC294640, a First-in-Class Sphingosine Kinase-2 Inhibitor, in Patients with Advanced Solid Tumors.

Authors:  Carolyn D Britten; Elizabeth Garrett-Mayer; Steven H Chin; Keisuke Shirai; Besim Ogretmen; Tricia A Bentz; Alan Brisendine; Kate Anderton; Susan L Cusack; Lynn W Maines; Yan Zhuang; Charles D Smith; Melanie B Thomas
Journal:  Clin Cancer Res       Date:  2017-04-18       Impact factor: 12.531

4.  Radiation-Induced Fibrosis: Mechanisms and Opportunities to Mitigate. Report of an NCI Workshop, September 19, 2016.

Authors:  Deborah E Citrin; Pataje G S Prasanna; Amanda J Walker; Michael L Freeman; Iris Eke; Mary Helen Barcellos-Hoff; Molykutty J Arankalayil; Eric P Cohen; Ruth C Wilkins; Mansoor M Ahmed; Mitchell S Anscher; Benjamin Movsas; Jeffrey C Buchsbaum; Marc S Mendonca; Thomas A Wynn; C Norman Coleman
Journal:  Radiat Res       Date:  2017-05-10       Impact factor: 2.841

5.  Mitigation of Radiation-Induced Epithelial Damage by the TLR5 Agonist Entolimod in a Mouse Model of Fractionated Head and Neck Irradiation.

Authors:  Ilia A Toshkov; Anatoli S Gleiberman; Vadim L Mett; Alan D Hutson; Anurag K Singh; Andrei V Gudkov; Lyudmila G Burdelya
Journal:  Radiat Res       Date:  2017-03-21       Impact factor: 2.841

6.  Nuclear Countermeasure Activity of TP508 Linked to Restoration of Endothelial Function and Acceleration of DNA Repair.

Authors:  Barbara Olszewska-Pazdrak; Scott D McVicar; Kempaiah Rayavara; Stephanie M Moya; Carla Kantara; Chris Gammarano; Paulina Olszewska; Gerald M Fuller; Laurie E Sower; Darrell H Carney
Journal:  Radiat Res       Date:  2016-07-07       Impact factor: 2.841

7.  New paradigms and future challenges in radiation oncology: an update of biological targets and technology.

Authors:  Stanley L Liauw; Philip P Connell; Ralph R Weichselbaum
Journal:  Sci Transl Med       Date:  2013-02-20       Impact factor: 17.956

8.  Radioprotectors and Radiomitigators for Improving Radiation Therapy: The Small Business Innovation Research (SBIR) Gateway for Accelerating Clinical Translation.

Authors:  Pataje G S Prasanna; Deepa Narayanan; Kory Hallett; Eric J Bernhard; Mansoor M Ahmed; Gregory Evans; Bhadrasain Vikram; Michael Weingarten; C Norman Coleman
Journal:  Radiat Res       Date:  2015-08-18       Impact factor: 2.841

9.  Nonclinical Safety and Toxicokinetics of MnTnBuOE-2-PyP5+ (BMX-001).

Authors:  Shayne Cox Gad; Dexter W Sullivan; Ivan Spasojevic; Cesar V Mujer; Charles B Spainhour; James D Crapo
Journal:  Int J Toxicol       Date:  2016-04-20       Impact factor: 2.032

10.  BIO 300, a nanosuspension of genistein, mitigates pneumonitis/fibrosis following high-dose radiation exposure in the C57L/J murine model.

Authors:  Isabel L Jackson; Andrew Zodda; Ganga Gurung; Radmila Pavlovic; Michael D Kaytor; Michael A Kuskowski; Zeljko Vujaskovic
Journal:  Br J Pharmacol       Date:  2017-11-03       Impact factor: 8.739

  10 in total
  3 in total

1.  Tumor Heterogeneity Research and Innovation in Biologically Based Radiation Therapy From the National Cancer Institute Radiation Research Program Portfolio.

Authors:  Jeffrey C Buchsbaum; Michael G Espey; Ceferino Obcemea; Jacek Capala; Mansoor Ahmed; Pataje G Prasanna; Bhadrasain Vikram; Julie A Hong; Beverly Teicher; Molykutty J Aryankalayil; Michelle A Bylicky; C Norman Coleman
Journal:  J Clin Oncol       Date:  2022-03-04       Impact factor: 50.717

2.  Thermal Stability Kinetics and Shelf Life Estimation of the Redox-Active Therapeutic and Mimic of Superoxide Dismutase Enzyme, Mn(III) meso-Tetrakis(N-ethylpyridinium-2-yl)porphyrin Chloride (MnTE-2-PyPCl5, BMX-010).

Authors:  Clarissa G C Maia; Bárbara C R de Araujo; Maria B de Freitas-Marques; Israel F da Costa; Maria Irene Yoshida; Wagner da Nova Mussel; Rita de Cássia O Sebastião; Júlio S Rebouças
Journal:  Oxid Med Cell Longev       Date:  2021-12-06       Impact factor: 6.543

3.  Therapy-Induced Senescence: Opportunities to Improve Anticancer Therapy.

Authors:  Pataje G Prasanna; Deborah E Citrin; Jeffrey Hildesheim; Mansoor M Ahmed; Sundar Venkatachalam; Gabriela Riscuta; Dan Xi; Guangrong Zheng; Jan van Deursen; Jorg Goronzy; Stephen J Kron; Mitchell S Anscher; Norman E Sharpless; Judith Campisi; Stephen L Brown; Laura J Niedernhofer; Ana O'Loghlen; Alexandros G Georgakilas; Francois Paris; David Gius; David A Gewirtz; Clemens A Schmitt; Mohamed E Abazeed; James L Kirkland; Ann Richmond; Paul B Romesser; Scott W Lowe; Jesus Gil; Marc S Mendonca; Sandeep Burma; Daohong Zhou; C Norman Coleman
Journal:  J Natl Cancer Inst       Date:  2021-10-01       Impact factor: 11.816

  3 in total

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