Warning: Undefined array key "mm" in /www/wwwroot/www.ai-bt.com/si.php on line 10 Deprecated: trim(): Passing null to parameter #1 ($string) of type string is deprecated in /www/wwwroot/www.ai-bt.com/si.php on line 10 Competitive inhibition of human skin collagenase by N-benzyloxycarbonyl-L-prolyl-L-alanyl-3-amino-2-oxopropyl-L-leucyl-L- alanylglycine ethyl ester.

Literature DB >> 3030274

Competitive inhibition of human skin collagenase by N-benzyloxycarbonyl-L-prolyl-L-alanyl-3-amino-2-oxopropyl-L-leucyl-L- alanylglycine ethyl ester.

D A Wallace, S R Bates, B Walker, G Kay, J White, D J Guthrie, N L Blumson, D T Elmore.

Abstract

A 'ketomethylene' peptide, N-benzyloxycarbonyl-L-prolyl-L-alanyl-3-amino- 2-oxopropyl-L-leucyl-L-alanylglycine ethyl ester, was synthesized and shown to be a fairly potent competitive inhibitor of human skin collagenase.

Entities: Chemical Species

Mesh：

Substances：

Year: 1986 PMID： 3030274 PMCID： PMC1147360 DOI： 10.1042/bj2390797

Source DB: PubMed Journal: Biochem J ISSN： 0264-6021 Impact factor: 3.857

15 in total

1. Mercaptoimidazolylpropionic acid hydrobromide. Inhibition of tadpole collagenase and related properties.

Authors: J A Yankeelov; H A Parish; A F Spatola
Journal: J Med Chem Date: 1978-07 Impact factor: 7.446

2. Identification and partial characterization of an inhibitor of collagenase from rabbit bone.

Authors: A Sellers; J J Reynolds
Journal: Biochem J Date: 1977-11-01 Impact factor: 3.857

3. The release of collagenase as an inactive proenzyme by bone explants in culture.

Authors: G Vaes
Journal: Biochem J Date: 1972-01 Impact factor: 3.857

Review 4. The determination of collagen and elastin.

Authors: D S Jackson; E G Cleary
Journal: Methods Biochem Anal Date: 1967

5. Metal binding peptide inhibitors of vertebrate collagenase.

Authors: R D Gray; H H Saneii; A F Spatola
Journal: Biochem Biophys Res Commun Date: 1981-08-31 Impact factor: 3.575

6. The collagen substrate specificity of human skin fibroblast collagenase.

Authors: H G Welgus; J J Jeffrey; A Z Eisen
Journal: J Biol Chem Date: 1981-09-25 Impact factor: 5.157

7. A new class of angiotensin-converting enzyme inhibitors.

Authors: A A Patchett; E Harris; E W Tristram; M J Wyvratt; M T Wu; D Taub; E R Peterson; T J Ikeler; J ten Broeke; L G Payne; D L Ondeyka; E D Thorsett; W J Greenlee; N S Lohr; R D Hoffsommer; H Joshua; W V Ruyle; J W Rothrock; S D Aster; A L Maycock; F M Robinson; R Hirschmann; C S Sweet; E H Ulm; D M Gross; T C Vassil; C A Stone
Journal: Nature Date: 1980-11-20 Impact factor: 49.962

Competitive inhibition of human skin collagenase by N-benzyloxycarbonyl-L-prolyl-L-alanyl-3-amino-2-oxopropyl-L-leucyl-L- alanylglycine ethyl ester.

1. Mercaptoimidazolylpropionic acid hydrobromide. Inhibition of tadpole collagenase and related properties.

2. Identification and partial characterization of an inhibitor of collagenase from rabbit bone.

3. The release of collagenase as an inactive proenzyme by bone explants in culture.

Review 4. The determination of collagen and elastin.

5. Metal binding peptide inhibitors of vertebrate collagenase.

6. The collagen substrate specificity of human skin fibroblast collagenase.

7. A new class of angiotensin-converting enzyme inhibitors.

8. A recording viscometer for assaying mammalian collagenase.

9. Synthesis of peptides of arginine chloromethyl ketone. Selective inactivation of human plasma kallikrein.

10. Inhibition of angiotensin converting enzyme by phosphoramidates and polyphosphates.

Review 1. Matrix metalloproteinases. Novel targets for directed cancer therapy.