Literature DB >> 30118684

Combined oral contraceptive interference with the ability of ulipristal acetate to delay ovulation: A prospective cohort study.

Alison B Edelman1, Jeffrey T Jensen2, Sara McCrimmon3, Marci Messerle-Forbes3, Andrea O'Donnell3, Jon D Hennebold2.   

Abstract

OBJECTIVE: To determine if a combined oral contraceptive (COC) initiated shortly after ulipristal acetate (UPA) administration interferes with its mechanism of action. STUDY
DESIGN: Healthy, reproductive-age women of normal BMI with proven ovulation (serum progesterone >3 ng/ml) were enrolled for three cycles (Cycle 1, UPA only; Cycle 2 washout; Cycle 3 UPA plus COC). During Cycles 1 and 3, subjects were monitored with transvaginal ultrasound and blood sampling for progesterone and LH every other day until a dominant follicle measuring >15 mm was visualized. In both treatment cycles, subjects received UPA (30mg) and were followed daily with similar monitoring for up to 7 days. In Cycle 3 only, subjects initiated a daily COC (0.15 mg levonorgestrel/30 μg ethinyl estradiol) 2 days after UPA. The study had 80% power to detect a 15% difference in the proportion of cycles with at least a 5-day delay in follicle rupture. We assessed follicle rupture as >50% decrease in mean size and adjudicated unclear outcomes with serum hormones.
RESULTS: A total of 36 women enrolled and 33 completed all study procedures [age 28.4 years (SD 3.9); BMI 23.4 (SD 2.4)]. Compared to Cycle 1, more subjects demonstrated evidence of follicle rupture in <5 days in Cycle 3 [1/33 (3%) vs. 9/33 (27%), p = .008]. We also included data from 2 subjects who experienced rupture prior to COC dosing in the analysis.
CONCLUSION: UPA's effectiveness is significantly reduced by administering COCs 2 days later. IMPLICATIONS: This study demonstrates that UPA's efficacy as an emergency contraceptive is reduced with early exposure to COCs.
Copyright © 2018 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  Contraceptive initiation; Emergency contraception; Oral contraceptives; Ovulation inhibition; Pharmacodynamics; Ulipristal acetate

Mesh:

Substances:

Year:  2018        PMID: 30118684      PMCID: PMC6204102          DOI: 10.1016/j.contraception.2018.08.003

Source DB:  PubMed          Journal:  Contraception        ISSN: 0010-7824            Impact factor:   3.375


  12 in total

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Authors:  Orla M Conneely
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2.  A prospective, randomized, pharmacodynamic study of quick-starting a desogestrel progestin-only pill following ulipristal acetate for emergency contraception.

Authors:  V Brache; L Cochon; I J M Duijkers; D P Levy; N Kapp; C Monteil; J L Abitbol; C Klipping
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3.  Ulipristal acetate prevents ovulation more effectively than levonorgestrel: analysis of pooled data from three randomized trials of emergency contraception regimens.

Authors:  Vivian Brache; Leila Cochon; Maëva Deniaud; Horacio B Croxatto
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4.  The effects on ovarian activity of ulipristal acetate when 'quickstarting' a combined oral contraceptive pill: a prospective, randomized, double-blind parallel-arm, placebo-controlled study.

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Review 6.  The critical roles of progesterone receptor (PGR) in ovulation, oocyte developmental competence and oviductal transport in mammalian reproduction.

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7.  Ulipristal acetate versus levonorgestrel for emergency contraception: a randomised non-inferiority trial and meta-analysis.

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8.  Ulipristal blocks ovulation by inhibiting progesterone receptor-dependent pathways intrinsic to the ovary.

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9.  Immediate pre-ovulatory administration of 30 mg ulipristal acetate significantly delays follicular rupture.

Authors:  V Brache; L Cochon; C Jesam; R Maldonado; A M Salvatierra; D P Levy; E Gainer; H B Croxatto
Journal:  Hum Reprod       Date:  2010-07-15       Impact factor: 6.918

10.  Suppression of follicular rupture with meloxicam, a cyclooxygenase-2 inhibitor: potential for emergency contraception.

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Journal:  Hum Reprod       Date:  2009-11-19       Impact factor: 6.918

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2.  Double Dosing Levonorgestrel-Based Emergency Contraception for Individuals With Obesity: A Randomized Controlled Trial.

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3.  The effects of vilaprisan on the pharmacodynamics and pharmacokinetics of a combined oral contraceptive-A randomized controlled trial.

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