Literature DB >> 28868285

Systemic BRAF/MEK Inhibitors as a Potential Treatment Option in Metastatic Conjunctival Melanoma.

Joel M Mor1, Ludwig M Heindl1.   

Abstract

AIM: In this review, we outline similarities between conjunctival and skin melanoma as well as the effectiveness of combined BRAF/MEK inhibition in melanoma, and discuss the applicability of these agents in conjunctival melanoma.
METHODS: The study provides a PubMed literature review.
RESULTS: Conjunctival melanoma and skin melanoma are genetically and phenotypically related. Both tumors typically harbor BRAF mutations in more than 50% of cases. New targeted therapies in metastatic skin melanoma include selective inhibition of BRAF and MEK. Combined BRAF/MEK inhibition has revolutionized the treatment of metastatic skin melanoma, significantly improving patients' prognoses. While these new substances have been investigated extensively in the treatment of skin melanoma, comparable studies in conjunctival melanoma do not exist owing to the rarity of the malignancy.
CONCLUSIONS: The application of combined BRAF/MEK inhibition in metastatic or unresectable conjunctival melanoma shows great potential for improving patients' prognoses. Future studies are needed to investigate the assumed benefit.

Entities:  

Keywords:  BRAF inhibitor; Conjunctival melanoma; MEK inhibitor; Metastatic disease; Primary acquired melanosis

Year:  2016        PMID: 28868285      PMCID: PMC5566756          DOI: 10.1159/000452473

Source DB:  PubMed          Journal:  Ocul Oncol Pathol        ISSN: 2296-4657


  81 in total

1.  Patterns of regional and distant metastasis in patients with conjunctival melanoma: experience at a cancer center over four decades.

Authors:  B Esmaeli; X Wang; A Youssef; J E Gershenwald
Journal:  Ophthalmology       Date:  2001-11       Impact factor: 12.079

2.  Mitogen-actived protein kinase activation is an early event in melanoma progression.

Authors:  Cynthia Cohen; Angel Zavala-Pompa; Judy H Sequeira; Mamoru Shoji; Deborah G Sexton; George Cotsonis; Francesca Cerimele; Baskaran Govindarajan; Nada Macaron; Jack L Arbiser
Journal:  Clin Cancer Res       Date:  2002-12       Impact factor: 12.531

3.  Immunophenotype of conjunctival melanomas: comparisons with uveal and cutaneous melanomas.

Authors:  Satori Iwamoto; Robert C Burrows; Hans E Grossniklaus; James Orcutt; Robert E Kalina; Michael Boehm; Mark A Bothwell; Rodney Schmidt
Journal:  Arch Ophthalmol       Date:  2002-12

4.  Incidence of sentinel node metastasis in patients with thin primary melanoma (< or = 1 mm) with vertical growth phase.

Authors:  I Bedrosian; M B Faries; D Guerry; R Elenitsas; L Schuchter; R Mick; F R Spitz; L P Bucky; A Alavi; D E Elder; D L Fraker; B J Czerniecki
Journal:  Ann Surg Oncol       Date:  2000-05       Impact factor: 5.344

5.  Conjunctival melanoma: risk factors for recurrence, exenteration, metastasis, and death in 150 consecutive patients.

Authors:  C L Shields; J A Shields; K Gündüz; J Cater; G V Mercado; N Gross; B Lally
Journal:  Arch Ophthalmol       Date:  2000-11

6.  Long-term follow-up of patients with conjunctival melanoma.

Authors:  Cornelia Werschnik; Peter K Lommatzsch
Journal:  Am J Clin Oncol       Date:  2002-06       Impact factor: 2.339

7.  Immunophenotypic differences between uveal and cutaneous melanomas.

Authors:  Satori Iwamoto; Robert C Burrows; Robert E Kalina; David George; Michael Boehm; Mark A Bothwell; Rodney Schmidt
Journal:  Arch Ophthalmol       Date:  2002-04

8.  Conjunctival melanoma: is it increasing in the United States?

Authors:  Guo-Pei Yu; Dan-Nin Hu; Steven McCormick; Paul T Finger
Journal:  Am J Ophthalmol       Date:  2003-06       Impact factor: 5.258

9.  High frequency of BRAF mutations in nevi.

Authors:  Pamela M Pollock; Ursula L Harper; Katherine S Hansen; Laura M Yudt; Mitchell Stark; Christiane M Robbins; Tracy Y Moses; Galen Hostetter; Urs Wagner; John Kakareka; Ghadi Salem; Tom Pohida; Peter Heenan; Paul Duray; Olli Kallioniemi; Nicholas K Hayward; Jeffrey M Trent; Paul S Meltzer
Journal:  Nat Genet       Date:  2002-11-25       Impact factor: 38.330

10.  Absence of BRAF gene mutations in uveal melanomas in contrast to cutaneous melanomas.

Authors:  S C Edmunds; I A Cree; F Dí Nícolantonío; J L Hungerford; J S Hurren; D P Kelsell
Journal:  Br J Cancer       Date:  2003-05-06       Impact factor: 7.640

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  11 in total

1.  [Conjunctival melanoma : Standard operating procedures in diagnosis, treatment and follow-up care].

Authors:  Jan-Peter Glossmann; Nicole Skoetz; Barbara Starbatty; Martina Bischoff; Serge Leyvraz; Henrike Westekemper; Ludwig M Heindl
Journal:  Ophthalmologe       Date:  2018-06       Impact factor: 1.059

2.  Two Late Recurrences of Conjunctival Melanoma.

Authors:  Niels J Brouwer; Stijn W Genders; Marina Marinkovic; Sjoerd G van Duinen; Martine J Jager; Gré P M Luyten
Journal:  Ocul Oncol Pathol       Date:  2018-12-12

3.  Dabrafenib and Trametinib for BRAF-Mutated Conjunctival Melanoma.

Authors:  Jenna May Kim; Sarah Weiss; John H Sinard; Renelle Pointdujour-Lim
Journal:  Ocul Oncol Pathol       Date:  2019-07-26

4.  Synergistic inhibition of MEK and reciprocal feedback networks for targeted intervention in malignancy.

Authors:  Yanan Li; Qingrong Dong; Yukun Cui
Journal:  Cancer Biol Med       Date:  2019-08       Impact factor: 4.248

Review 5.  Sentinel lymph node biopsy in the management of conjunctival melanoma: current insights.

Authors:  Joel M Mor; Alexander C Rokohl; Konrad R Koch; Ludwig M Heindl
Journal:  Clin Ophthalmol       Date:  2019-07-23

Review 6.  Conjunctival Melanoma: Genetic and Epigenetic Insights of a Distinct Type of Melanoma.

Authors:  Ernesto Rossi; Giovanni Schinzari; Brigida Anna Maiorano; Monica Maria Pagliara; Alessandro Di Stefani; Emilio Bria; Ketty Peris; Maria Antonietta Blasi; Giampaolo Tortora
Journal:  Int J Mol Sci       Date:  2019-10-31       Impact factor: 5.923

7.  Fangchinoline suppresses conjunctival melanoma by directly binding FUBP2 and inhibiting the homologous recombination pathway.

Authors:  Keting Bao; Yongyun Li; Jinlian Wei; Ruoxi Li; Jie Yang; Jiahao Shi; Baoli Li; Jin Zhu; Fei Mao; Renbing Jia; Jian Li
Journal:  Cell Death Dis       Date:  2021-04-07       Impact factor: 8.469

8.  PD-L1 Expression in 65 Conjunctival Melanomas and Its Association with Clinical Outcome.

Authors:  Sandra Lassalle; Sacha Nahon-Esteve; Eric Frouin; Camille Boulagnon-Rombi; Nicolas Josselin; Nathalie Cassoux; Raymond Barnhill; Boris Scheller; Stéphanie Baillif; Paul Hofman
Journal:  Int J Mol Sci       Date:  2020-11-30       Impact factor: 5.923

9.  Molecular Genetics of Conjunctival Melanoma and Prognostic Value of TERT Promoter Mutation Analysis.

Authors:  Natasha M van Poppelen; Jolique A van Ipenburg; Quincy van den Bosch; Jolanda Vaarwater; Tom Brands; Bert Eussen; Frank Magielsen; Hendrikus J Dubbink; Dion Paridaens; Erwin Brosens; Nicole Naus; Annelies de Klein; Emine Kiliç; Robert M Verdijk
Journal:  Int J Mol Sci       Date:  2021-05-28       Impact factor: 5.923

10.  Transcriptional characterization of conjunctival melanoma identifies the cellular tumor microenvironment and prognostic gene signatures.

Authors:  Julian Wolf; Claudia Auw-Haedrich; Anja Schlecht; Stefaniya Boneva; Hans Mittelviefhaus; Thabo Lapp; Hansjürgen Agostini; Thomas Reinhard; Günther Schlunck; Clemens A K Lange
Journal:  Sci Rep       Date:  2020-10-12       Impact factor: 4.379

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