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Literature DB >> 28244728

The Ecstasy and Agony of Assay Interference Compounds.

Courtney Aldrich¹, Carolyn Bertozzi², Gunda I Georg³, Laura Kiessling⁴, Craig Lindsley⁵, Dennis Liotta⁶, Kenneth M Merz⁷, Alanna Schepartz⁸, Shaomeng Wang³.

Abstract

Mesh：

Substances：
Colloids

Year: 2017 PMID： 28244728 DOI： 10.1021/acschembio.7b00119

Source DB: PubMed Journal: ACS Chem Biol ISSN： 1554-8929 Impact factor: 5.100

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3 in total

1. The relevance of K_i calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor.

Authors: Hannah Wapenaar; Thea van den Bosch; Niek G J Leus; Petra E van der Wouden; Nikolaos Eleftheriadis; Jos Hermans; Gebremedhin Solomon Hailu; Dante Rotili; Antonello Mai; Alexander Dömling; Rainer Bischoff; Hidde J Haisma; Frank J Dekker
Journal: Eur J Med Chem Date: 2017-05-05 Impact factor: 6.514

2. Bitopic fluorescent antagonists of the A_2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners.

Authors: Romain Duroux; Antonella Ciancetta; Philip Mannes; Jinha Yu; Shireesha Boyapati; Elizabeth Gizewski; Said Yous; Francisco Ciruela; John A Auchampach; Zhan-Guo Gao; Kenneth A Jacobson
Journal: Medchemcomm Date: 2017-06-22 Impact factor: 3.597

3. Cytotoxic unsaturated electrophilic compounds commonly target the ubiquitin proteasome system.

Authors: Karthik Selvaraju; Arjan Mofers; Paola Pellegrini; Johannes Salomonsson; Alexandra Ahlner; Vivian Morad; Ellin-Kristina Hillert; Belen Espinosa; Elias S J Arnér; Lasse Jensen; Jonas Malmström; Maria V Turkina; Padraig D'Arcy; Michael A Walters; Maria Sunnerhagen; Stig Linder
Journal: Sci Rep Date: 2019-07-08 Impact factor: 4.379

3 in total

The Ecstasy and Agony of Assay Interference Compounds.

1. The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor.

2. Bitopic fluorescent antagonists of the A2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners.

3. Cytotoxic unsaturated electrophilic compounds commonly target the ubiquitin proteasome system.

1. The relevance of K_i calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor.

2. Bitopic fluorescent antagonists of the A_2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners.