Literature DB >> 28109627

A final report of a phase I study of veliparib (ABT-888) in combination with low-dose fractionated whole abdominal radiation therapy (LDFWAR) in patients with advanced solid malignancies and peritoneal carcinomatosis with a dose escalation in ovarian and fallopian tube cancers.

Kim A Reiss1, Joseph M Herman2, Deborah Armstrong1, Marianna Zahurak3, Anthony Fyles4, Anthony Brade4, Michael Milosevic4, Laura A Dawson4, Angela Scardina1, Patricia Fischer1, Amy Hacker-Prietz2, Robert J Kinders5, Lihua Wang5, Alice Chen6, Sarah Temkin7, Naomi Horiba7, Lee-Anne Stayner8, Lillian L Siu8, Nilofer S Azad9.   

Abstract

BACKGROUND: The combination of low-dose radiation therapy with PARP inhibition enhances anti-tumor efficacy through potentiating DNA damage. We combined low-dose fractionated whole abdominal radiation (LDFWAR) with ABT-888 in patients with peritoneal carcinomatosis with a dose escalation in ovarian and fallopian cancer patients (OV).
METHODS: Patients were treated with veliparib, 40-400mg orally BID on days 1-21 of 3 28-day cycles on 6 dose levels. Dose levels 5 and 6 included only OV patients. LDFWAR consisted of 21.6Gy in 36 fractions, 0.6Gy twice daily on days 1 and 5 for weeks 1-3 of each cycle. Circulating tumor material and quality of life were serially assessed.
RESULTS: 32pts were treated. Median follow-up was 45months (10-50). The most common treatment-related grade 3 and 4 toxicities were lymphopenia (59%), anemia (9%), thrombocytopenia (12%), neutropenia (6%), leukopenia (6%), nausea (6%), diarrhea (6%), anorexia (6%), vomiting (6%) and fatigue (6%). The maximum tolerated dose was determined to be 250mg PO BID. Median PFS was 3.6months and median OS was 9.1months. In OV patients, OS was longer for platinum-sensitive patients (10.9mo) compared to platinum-resistant patients (5.8mo). QoL decreased for all groups during treatment. Germline BRCA status was known for 14/18 patients with OV cancers, 5 of whom were BRCA mutation carriers. One objective response (3%) was observed.
CONCLUSION: ABT-888 plus LDFWAR is tolerable with gastrointestinal symptoms, fatigue and myelosuppression as the most common toxicities. The single observed objective response was in a germline BRCA mutated, platinum-sensitive patient. Copyright Â
© 2017 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  BRCA; Ovarian cancer; PARP inhibition; Peritoneal carcinomatosis; Radiation; Veliparib

Mesh:

Substances:

Year:  2017        PMID: 28109627      PMCID: PMC5330287          DOI: 10.1016/j.ygyno.2017.01.016

Source DB:  PubMed          Journal:  Gynecol Oncol        ISSN: 0090-8258            Impact factor:   5.482


  21 in total

1.  Low-dose abdominal radiation as a docetaxel chemosensitizer for recurrent epithelial ovarian cancer: a phase I study of the Gynecologic Oncology Group.

Authors:  Charles A Kunos; Michael W Sill; Thomas E Buekers; Joan L Walker; Jeanne M Schilder; S Diane Yamada; Steven E Waggoner; Mohammed Mohiuddin; Paula M Fracasso
Journal:  Gynecol Oncol       Date:  2011-02       Impact factor: 5.482

2.  Chemopotentiation of temozolomide, irinotecan, and cisplatin activity by CEP-6800, a poly(ADP-ribose) polymerase inhibitor.

Authors:  Sheila J Miknyoczki; Susan Jones-Bolin; Sonya Pritchard; Kathryn Hunter; Hugh Zhao; Weihua Wan; Mark Ator; Ronald Bihovsky; Robert Hudkins; Sankar Chatterjee; Andres Klein-Szanto; Craig Dionne; Bruce Ruggeri
Journal:  Mol Cancer Ther       Date:  2003-04       Impact factor: 6.261

3.  The poly(ADP-Ribose) polymerase inhibitor ABT-888 reduces radiation-induced nuclear EGFR and augments head and neck tumor response to radiotherapy.

Authors:  Somaira Nowsheen; James A Bonner; Eddy S Yang
Journal:  Radiother Oncol       Date:  2011-06-28       Impact factor: 6.280

4.  A Phase I study of veliparib (ABT-888) in combination with low-dose fractionated whole abdominal radiation therapy in patients with advanced solid malignancies and peritoneal carcinomatosis.

Authors:  Kim A Reiss; Joseph M Herman; Marianna Zahurak; Anthony Brade; Laura A Dawson; Angela Scardina; Caitlin Joffe; Emily Petito; Amy Hacker-Prietz; Robert J Kinders; Lihua Wang; Alice Chen; Sarah Temkin; Naomi Horiba; Lillian L Siu; Nilofer S Azad
Journal:  Clin Cancer Res       Date:  2014-10-29       Impact factor: 12.531

Review 5.  Poly (ADP-ribose) polymerase inhibitors: recent advances and future development.

Authors:  Clare L Scott; Elizabeth M Swisher; Scott H Kaufmann
Journal:  J Clin Oncol       Date:  2015-03-16       Impact factor: 44.544

6.  Niraparib Maintenance Therapy in Platinum-Sensitive, Recurrent Ovarian Cancer.

Authors:  Mansoor R Mirza; Bradley J Monk; Jørn Herrstedt; Amit M Oza; Sven Mahner; Andrés Redondo; Michel Fabbro; Jonathan A Ledermann; Domenica Lorusso; Ignace Vergote; Noa E Ben-Baruch; Christian Marth; Radosław Mądry; René D Christensen; Jonathan S Berek; Anne Dørum; Anna V Tinker; Andreas du Bois; Antonio González-Martín; Philippe Follana; Benedict Benigno; Per Rosenberg; Lucy Gilbert; Bobbie J Rimel; Joseph Buscema; John P Balser; Shefali Agarwal; Ursula A Matulonis
Journal:  N Engl J Med       Date:  2016-10-07       Impact factor: 91.245

7.  Specific killing of BRCA2-deficient tumours with inhibitors of poly(ADP-ribose) polymerase.

Authors:  Helen E Bryant; Niklas Schultz; Huw D Thomas; Kayan M Parker; Dan Flower; Elena Lopez; Suzanne Kyle; Mark Meuth; Nicola J Curtin; Thomas Helleday
Journal:  Nature       Date:  2005-04-14       Impact factor: 69.504

8.  Targeted antitumour therapy--future perspectives.

Authors:  M Ranson; G Jayson
Journal:  Br J Cancer       Date:  2005-06       Impact factor: 7.640

9.  Olaparib maintenance therapy in patients with platinum-sensitive relapsed serous ovarian cancer: a preplanned retrospective analysis of outcomes by BRCA status in a randomised phase 2 trial.

Authors:  Jonathan Ledermann; Philipp Harter; Charlie Gourley; Michael Friedlander; Ignace Vergote; Gordon Rustin; Clare L Scott; Werner Meier; Ronnie Shapira-Frommer; Tamar Safra; Daniela Matei; Anitra Fielding; Stuart Spencer; Brian Dougherty; Maria Orr; Darren Hodgson; J Carl Barrett; Ursula Matulonis
Journal:  Lancet Oncol       Date:  2014-05-31       Impact factor: 41.316

Review 10.  Dose escalation methods in phase I cancer clinical trials.

Authors:  Christophe Le Tourneau; J Jack Lee; Lillian L Siu
Journal:  J Natl Cancer Inst       Date:  2009-05-12       Impact factor: 13.506

View more
  18 in total

Review 1.  PARP inhibitors: Clinical utility and possibilities of overcoming resistance.

Authors:  Benjamin G Bitler; Zachary L Watson; Lindsay J Wheeler; Kian Behbakht
Journal:  Gynecol Oncol       Date:  2017-10-14       Impact factor: 5.482

Review 2.  Development of new medical treatment for epithelial ovarian cancer recurrence.

Authors:  Rosanna Mancari; Giuseppe Cutillo; Valentina Bruno; Cristina Vincenzoni; Emanuela Mancini; Ermelinda Baiocco; Simone Bruni; Giuseppe Vocaturo; Benito Chiofalo; Enrico Vizza
Journal:  Gland Surg       Date:  2020-08

Review 3.  Soft tissue sarcomas: new opportunity of treatment with PARP inhibitors?

Authors:  Monica Mangoni; Mariangela Sottili; Giulia Salvatore; Domenico Campanacci; Guido Scoccianti; Giovanni Beltrami; Camilla Delli Paoli; Luca Dominici; Virginia Maragna; Emanuela Olmetto; Icro Meattini; Isacco Desideri; Pierluigi Bonomo; Daniela Greto; Lorenzo Livi
Journal:  Radiol Med       Date:  2018-03-26       Impact factor: 3.469

Review 4.  Veliparib in ovarian cancer: a new synthetically lethal therapeutic approach.

Authors:  Stergios Boussios; Peeter Karihtala; Michele Moschetta; Charlotte Abson; Afroditi Karathanasi; Nikolaos Zakynthinakis-Kyriakou; Jake Edward Ryan; Matin Sheriff; Elie Rassy; Nicholas Pavlidis
Journal:  Invest New Drugs       Date:  2019-10-24       Impact factor: 3.850

5.  Patient-derived Models Reveal Impact of the Tumor Microenvironment on Therapeutic Response.

Authors:  Ayesha A Shafi; Matthew J Schiewer; Renée de Leeuw; Emanuela Dylgjeri; Peter A McCue; Neelima Shah; Leonard G Gomella; Costas D Lallas; Edouard J Trabulsi; Margaret M Centenera; Theresa E Hickey; Lisa M Butler; Ganesh Raj; Wayne D Tilley; Edna Cukierman; Karen E Knudsen
Journal:  Eur Urol Oncol       Date:  2018-06-06

6.  Blocking PARP activity with the inhibitor veliparib enhances radiotherapy sensitivity in endometrial carcinoma.

Authors:  Jing Wang; Weizhen Xing; Yanling Lin; Nuray Uskenbayeva; Hongchao Yan; Yang Xu; Lisha Fang
Journal:  J Clin Lab Anal       Date:  2022-04-14       Impact factor: 3.124

Review 7.  Radiation Treatment in Women with Ovarian Cancer: Past, Present, and Future.

Authors:  Emma C Fields; William P McGuire; Lilie Lin; Sarah M Temkin
Journal:  Front Oncol       Date:  2017-08-21       Impact factor: 6.244

8.  Current status and future prospects of PARP inhibitor clinical trials in ovarian cancer.

Authors:  Xuan Jiang; Weihua Li; Xiaoying Li; Huimin Bai; Zhenyu Zhang
Journal:  Cancer Manag Res       Date:  2019-05-10       Impact factor: 3.989

Review 9.  Poly-(ADP-ribose)-polymerase inhibitors as radiosensitizers: a systematic review of pre-clinical and clinical human studies.

Authors:  Paul Lesueur; François Chevalier; Jean-Baptiste Austry; Waisse Waissi; Hélène Burckel; Georges Noël; Jean-Louis Habrand; Yannick Saintigny; Florence Joly
Journal:  Oncotarget       Date:  2017-07-07

10.  Study protocols of three parallel phase 1 trials combining radical radiotherapy with the PARP inhibitor olaparib.

Authors:  R de Haan; E van Werkhoven; M M van den Heuvel; H M U Peulen; G S Sonke; P Elkhuizen; M W M van den Brekel; M E T Tesselaar; C Vens; J H M Schellens; B van Triest; M Verheij
Journal:  BMC Cancer       Date:  2019-09-10       Impact factor: 4.430

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.