Literature DB >> 28033474

Hypothesizing That Neuropharmacological and Neuroimaging Studies of Glutaminergic-Dopaminergic Optimization Complex (KB220Z) Are Associated With "Dopamine Homeostasis" in Reward Deficiency Syndrome (RDS).

Kenneth Blum1,2,3,4,5,6,7,8,9, Marcelo Febo1, Lyle Fried7, Mona Li2, Kristina Dushaj2, Eric R Braverman2, Thomas McLaughlin10, Bruce Steinberg11, Rajendra D Badgaiyan9.   

Abstract

BACKGROUND: There is need for better treatments of addictive behaviors, both substance and non-substance related, termed Reward Deficiency Syndrome (RDS). While the FDA has approved pharmaceuticals under the umbrella term Medication Assisted Treatment (MAT), these drugs are not optimal.
OBJECTIVES: It is our contention that these drugs work well in the short-term by blocking dopamine function leading to psychological extinction. However, use of buprenorphine/Naloxone over a long period of time results in unwanted addiction liability, reduced emotional affect, and mood changes including suicidal ideation.
METHODS: We are thus proposing a paradigm shift in addiction treatment, with the long-term goal of achieving "Dopamine Homeostasis." While this may be a laudable goal, it is very difficult to achieve. Nevertheless, this commentary briefly reviews past history of developing and subsequently, utilizing a glutaminergic-dopaminergic optimization complex [Kb220Z] shown to be beneficial in at least 20 human clinical trials and in a number of published and unpublished studies.
RESULTS: It is our opinion that, while additional required studies could confirm these findings to date, the cited studies are indicative of achieving enhanced resting state functional connectivity, connectivity volume, and possibly, neuroplasticity. Conclusions/Importance: We are proposing a Reward Deficiency Solution System (RDSS) that includes: Genetic Addiction Risk Score (GARS); Comprehensive Analysis of Reported Drugs (CARD); and a glutaminergic-dopaminergic optimization complex (Kb220Z). Continued investigation of this novel strategy may lead to a better-targeted approach in the long-term, causing dopamine regulation by balancing the glutaminergic-dopaminergic pathways. This may potentially change the landscape of treating all addictions leading us to the promised land.

Entities:  

Keywords:  Dopamine homeostasis; KB220Z; Reward Deficiency Syndrome (RDS); neuroimaging; neuropharmaco-logical

Mesh:

Substances:

Year:  2016        PMID: 28033474      PMCID: PMC5589271          DOI: 10.1080/10826084.2016.1244551

Source DB:  PubMed          Journal:  Subst Use Misuse        ISSN: 1082-6084            Impact factor:   2.164


  57 in total

1.  Reward deficiency syndrome in obesity: a preliminary cross-sectional trial with a Genotrim variant.

Authors:  Kenneth Blum; Thomas J H Chen; Brian Meshkin; B William Downs; Cory A Gordon; Seth Blum; Julie F Mengucci; Eric R Braverman; Vanessa Arcuri; Michael Varshavskiy; Roger Deutsch; Manuel Martinez-Pons
Journal:  Adv Ther       Date:  2006 Nov-Dec       Impact factor: 3.845

2.  Substance use disorder exacerbates brain electrophysiological abnormalities in a psychiatrically-ill population.

Authors:  E R Braverman; K Blum
Journal:  Clin Electroencephalogr       Date:  1996

3.  Improvement of inpatient treatment of the alcoholic as a function of neurotransmitter restoration: a pilot study.

Authors:  K Blum; M C Trachtenberg; J C Ramsay
Journal:  Int J Addict       Date:  1988-09

Review 4.  Neurogenetics and gene therapy for reward deficiency syndrome: are we going to the Promised Land?

Authors:  Kenneth Blum; Peter K Thanos; Rajendra D Badgaiyan; Marcelo Febo; Marlene Oscar-Berman; James Fratantonio; Zsolt Demotrovics; Mark S Gold
Journal:  Expert Opin Biol Ther       Date:  2015-05-14       Impact factor: 4.388

5.  Opioid antagonist challenges in buprenorphine maintained patients.

Authors:  T R Kosten; J H Krystal; D S Charney; L H Price; C H Morgan; H D Kleber
Journal:  Drug Alcohol Depend       Date:  1990-02       Impact factor: 4.492

6.  Community-wide measures of wellness in a remote First Nations community experiencing opioid dependence: evaluating outpatient buprenorphine-naloxone substitution therapy in the context of a First Nations healing program.

Authors:  Dinah Kanate; David Folk; Sharon Cirone; Janet Gordon; Mike Kirlew; Terri Veale; Natalie Bocking; Sara Rea; Len Kelly
Journal:  Can Fam Physician       Date:  2015-02       Impact factor: 3.275

7.  Neurogenetics and clinical evidence for the putative activation of the brain reward circuitry by a neuroadaptagen: proposing an addiction candidate gene panel map.

Authors:  Thomas J H Chen; Kenneth Blum; Amanda L C Chen; Abdalla Bowirrat; William B Downs; Margret A Madigan; Roger L Waite; John A Bailey; Mallory Kerner; Swetha Yeldandi; Neil Majmundar; John Giordano; Siohban Morse; David Miller; Frank Fornari; Eric R Braverman
Journal:  J Psychoactive Drugs       Date:  2011 Apr-Jun

8.  Ethanol acceptance as a function of genotype amounts of brain [Met]enkephalin.

Authors:  K Blum; S F Elston; L DeLallo; A H Briggs; J E Wallace
Journal:  Proc Natl Acad Sci U S A       Date:  1983-11       Impact factor: 11.205

9.  Brain disease model of addiction: why is it so controversial?

Authors:  Nora D Volkow; George Koob
Journal:  Lancet Psychiatry       Date:  2015-08       Impact factor: 27.083

10.  Dopamine neurons modulate neural encoding and expression of depression-related behaviour.

Authors:  Kay M Tye; Julie J Mirzabekov; Melissa R Warden; Emily A Ferenczi; Hsing-Chen Tsai; Joel Finkelstein; Sung-Yon Kim; Avishek Adhikari; Kimberly R Thompson; Aaron S Andalman; Lisa A Gunaydin; Ilana B Witten; Karl Deisseroth
Journal:  Nature       Date:  2012-12-12       Impact factor: 49.962

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  7 in total

1.  Nicotinamide Adenine Dinucleotide (NAD+) and Enkephalinase Inhibition (IV1114589NAD) Infusions Significantly Attenuate Psychiatric Burden Sequalae in Substance Use Disorder (SUD) in Fifty Cases.

Authors:  Kenneth Blum; David Han; David Baron; Shan Kazmi; Igor Elman; Luis Llanos Gomez; Marjorie C Gondre-Lewis; Panyotis K Thanos; Eric R Braverman; Rajendra D Badgaiyan
Journal:  Curr Psychiatry Res Rev       Date:  2022-06-21

Review 2.  Precision Behavioral Management (PBM) and Cognitive Control as a Potential Therapeutic and Prophylactic Modality for Reward Deficiency Syndrome (RDS): Is There Enough Evidence?

Authors:  Margaret A Madigan; Ashim Gupta; Abdalla Bowirrat; David Baron; Rajendra D Badgaiyan; Igor Elman; Catherine A Dennen; Eric R Braverman; Mark S Gold; Kenneth Blum
Journal:  Int J Environ Res Public Health       Date:  2022-05-24       Impact factor: 4.614

3.  Pro-dopamine regulator, KB220Z, attenuates hoarding and shopping behavior in a female, diagnosed with SUD and ADHD.

Authors:  Thomas McLaughlin; Kenneth Blum; Bruce Steinberg; Edward J Modestino; Lyle Fried; David Baron; David Siwicki; Eric R Braverman; Rajendra D Badgaiyan
Journal:  J Behav Addict       Date:  2018-01-10       Impact factor: 6.756

4.  Physical Exercise Interventions for Drug Addictive Disorders.

Authors:  Trevor Archer; Rajendra D Badgaiyan; Kenneth Blum
Journal:  J Reward Defic Syndr Addict Sci       Date:  2017-05-29

5.  Cannabis-Induced Hypodopaminergic Anhedonia and Cognitive Decline in Humans: Embracing Putative Induction of Dopamine Homeostasis.

Authors:  Kenneth Blum; Jag Khalsa; Jean Lud Cadet; David Baron; Abdalla Bowirrat; Brent Boyett; Lisa Lott; Raymond Brewer; Marjorie Gondré-Lewis; Gregory Bunt; Shan Kazmi; Mark S Gold
Journal:  Front Psychiatry       Date:  2021-03-30       Impact factor: 4.157

6.  Would induction of dopamine homeostasis via coupling genetic addiction risk score (GARS®) and pro-dopamine regulation benefit benzodiazepine use disorder (BUD)?

Authors:  K Blum; M Gold; E J Modestino; D Baron; B Boyett; D Siwicki; L Lott; A Podesta; A K Roy; M Hauser; B W Downs; R D Badgaiyan
Journal:  J Syst Integr Neurosci       Date:  2018-05-03

Review 7.  A Review of DNA Risk Alleles to Determine Epigenetic Repair of mRNA Expression to Prove Therapeutic Effectiveness in Reward Deficiency Syndrome (RDS): Embracing "Precision Behavioral Management".

Authors:  Kenneth Blum; Bruce Steinberg; Marjorie C Gondre-Lewis; David Baron; Edward J Modestino; Rajendra D Badgaiyan; B William Downs; Debasis Bagchi; Raymond Brewer; Thomas McLaughlin; Abdalla Bowirrat; Mark Gold
Journal:  Psychol Res Behav Manag       Date:  2021-12-17
  7 in total

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