Literature DB >> 27742728

Effect of Sitagliptin on Kidney Function and Respective Cardiovascular Outcomes in Type 2 Diabetes: Outcomes From TECOS.

Jan H Cornel1, George L Bakris2, Susanna R Stevens3, Michael Alvarsson4, Willem A Bax1, Lee-Ming Chuang5, Samuel S Engel6, Renato D Lopes3, Darren K McGuire7, Axel Riefflin8, Helena Wachslicht Rodbard9, Isaac Sinay10, Tsvetalina Tankova11, Julio Wainstein12, Eric D Peterson3, Rury R Holman13.   

Abstract

OBJECTIVE: To evaluate chronic kidney disease (CKD) and cardiovascular outcomes in TECOS (Clinical trial reg. no. NCT00790205, clinicaltrials.gov) participants with type 2 diabetes and cardiovascular disease treated with sitagliptin, a dipeptidyl peptidase 4 inhibitor, according to baseline estimated glomerular filtration rate (eGFR). RESEARCH DESIGN AND METHODS: We used data from 14,671 TECOS participants assigned in a double-blind design to receive sitagliptin or placebo added to existing therapy, while aiming for glycemic equipoise between groups. Cardiovascular and CKD outcomes were evaluated over a median period of 3 years, with participants categorized at baseline into eGFR stages 1, 2, 3a, and 3b (≥90, 60-89, 45-59, or 30-44 mL/min/1.73 m2, respectively).
RESULTS: Participants with eGFR stage 3b were older, were more often female, and had a longer duration of diabetes. Four-point major adverse cardiovascular event rates increased with lower baseline eGFR (3.52, 3.55, 5.74, and 7.34 events/100 patient-years for stages 1-3b, respectively). Corresponding adjusted hazard ratios for stages 2, 3a, and 3b versus stage 1 were 0.93 (95% CI 0.82-1.06), 1.28 (1.10-1.49), and 1.39 (1.13-1.72), respectively. Sitagliptin therapy was not associated with cardiovascular outcomes for any eGFR stage (interaction P values were all >0.44). Kidney function declined at the same rate in both treatment groups, with a marginally lower but constant eGFR difference (-1.3 mL/min/1.73 m2) in those participants who were assigned to sitagliptin. Treatment differences in these eGFR values remained after adjustment for region, baseline eGFR, baseline HbA1c, time of assessment, and within-study HbA1c levels.
CONCLUSIONS: Impaired kidney function is associated with worse cardiovascular outcomes. Sitagliptin has no clinically significant impact on cardiovascular or CKD outcomes, irrespective of baseline eGFR.
© 2016 by the American Diabetes Association.

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Year:  2016        PMID: 27742728     DOI: 10.2337/dc16-1415

Source DB:  PubMed          Journal:  Diabetes Care        ISSN: 0149-5992            Impact factor:   19.112


  54 in total

Review 1.  Sitagliptin: A Review in Type 2 Diabetes.

Authors:  Lesley J Scott
Journal:  Drugs       Date:  2017-02       Impact factor: 9.546

Review 2.  Antihyperglycemic agents as novel natriuretic therapies in diabetic kidney disease.

Authors:  David León Jiménez; David Z I Cherney; Petter Bjornstad; Luis Castilla-Guerra; José Pablo Miramontes González
Journal:  Am J Physiol Renal Physiol       Date:  2018-08-01

3.  The renoprotective effect and safety of a DPP-4 inhibitor, sitagliptin, at a small dose in type 2 diabetic patients with a renal dysfunction when changed from other DPP-4 inhibitors: REAL trial.

Authors:  Koichi Kanozawa; Yuichi Noguchi; Souichi Sugahara; Satoko Nakamura; Hirohisa Yamamoto; Keiko Kaneko; Rika Kono; Saeko Sato; Tomonari Ogawa; Hajime Hasegawa; Shigehiro Katayama
Journal:  Clin Exp Nephrol       Date:  2017-12-23       Impact factor: 2.801

Review 4.  Role of Impaired Nutrient and Oxygen Deprivation Signaling and Deficient Autophagic Flux in Diabetic CKD Development: Implications for Understanding the Effects of Sodium-Glucose Cotransporter 2-Inhibitors.

Authors:  Milton Packer
Journal:  J Am Soc Nephrol       Date:  2020-04-10       Impact factor: 10.121

5.  Effects of Diabetes Medications Targeting the Incretin System on the Kidney.

Authors:  Richard J MacIsaac; Merlin C Thomas
Journal:  Clin J Am Soc Nephrol       Date:  2018-01-10       Impact factor: 8.237

Review 6.  Cardiovascular Safety of Antidiabetic Drugs in the Hospital Setting.

Authors:  Stacey A Seggelke; Mark C Lindsay; Ingrid Hazlett; Rebecca Sanagorski; Robert H Eckel; Cecilia C Low Wang
Journal:  Curr Diab Rep       Date:  2017-08       Impact factor: 4.810

Review 7.  Diagnosis and Management of Type 2 Diabetic Kidney Disease.

Authors:  Simit M Doshi; Allon N Friedman
Journal:  Clin J Am Soc Nephrol       Date:  2017-03-09       Impact factor: 8.237

Review 8.  More than just an enzyme: Dipeptidyl peptidase-4 (DPP-4) and its association with diabetic kidney remodelling.

Authors:  Shreyasi Gupta; Utpal Sen
Journal:  Pharmacol Res       Date:  2019-08-08       Impact factor: 7.658

Review 9.  Cardiovascular outcome trials of glucose-lowering medications: an update.

Authors:  Philip Home
Journal:  Diabetologia       Date:  2019-01-03       Impact factor: 10.122

Review 10.  Incretin drugs in diabetic kidney disease: biological mechanisms and clinical evidence.

Authors:  Radica Z Alicic; Emily J Cox; Joshua J Neumiller; Katherine R Tuttle
Journal:  Nat Rev Nephrol       Date:  2020-11-20       Impact factor: 28.314

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