Literature DB >> 27659699

Opioid-receptor antagonism increases pain and decreases pleasure in obese and non-obese individuals.

Rebecca C Price1,2, Nicolas V Christou3, Steven B Backman4, Laura Stone2,5, Petra Schweinhardt6,7,8.   

Abstract

RATIONALE: Endogenous opioids inhibit nociceptive processing and promote the experience of pleasure. It has been proposed that pain and pleasure lie at opposite ends of an affective spectrum, but the relationship between pain and pleasure and the role of opioids in mediating this relationship has not been tested.
OBJECTIVES: Here, we used obese individuals as a model of a dysfunctional opioid system to assess the role of the endogenous opioid peptide, beta-endorphin, on pain and pleasure sensitivity.
METHODS: Obese (10M/10F) and age- and gender-matched non-obese (10M/10F) controls were included in the study. Pain sensitivity using threshold, tolerance, and subjective rating assessments and perceived sweet pleasantness using sucrose solutions were assessed in two testing sessions with placebo or the opioid antagonist, naltrexone (0.7 mg/kg body weight). Beta-endorphin levels were assessed in both sessions. RESULTS AND
CONCLUSIONS: Despite having higher levels of baseline beta-endorphin and altered beta-endorphin-reactivity to naltrexone, obese individuals reported a similar increase in pain and decrease in pleasantness following naltrexone compared to non-obese individuals. Beta-endorphin levels did not correlate with pain or pleasantness in either group, but naltrexone-induced changes in pain and pleasantness were mildly correlated. Moreover, naltrexone-induced changes in pain were related to depression scores, while naltrexone-induced changes in sweet pleasantness were related to anxiety scores, indicating that pain and pleasantness are related, but influenced by different processes.

Entities:  

Keywords:  Anxiety; Beta-endorphin; Depression; Naltrexone; Obesity; Opioid

Mesh:

Substances:

Year:  2016        PMID: 27659699     DOI: 10.1007/s00213-016-4417-4

Source DB:  PubMed          Journal:  Psychopharmacology (Berl)        ISSN: 0033-3158            Impact factor:   4.530


  71 in total

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Review 10.  Effects of alcohol dependence and withdrawal on stress responsiveness and alcohol consumption.

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Journal:  Alcohol Res       Date:  2012
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  5 in total

1.  Effects of opioid receptor stimulation and blockade on touch pleasantness: a double-blind randomised trial.

Authors:  Guro E Løseth; Marie Eikemo; Siri Leknes
Journal:  Soc Cogn Affect Neurosci       Date:  2019-05-17       Impact factor: 3.436

2.  Endogenous opioids contribute to the feeling of pain relief in humans.

Authors:  Laura Sirucek; Rebecca Christine Price; Wiebke Gandhi; Marie-Eve Hoeppli; Emma Fahey; Annie Qu; Susanne Becker; Petra Schweinhardt
Journal:  Pain       Date:  2021-12-01       Impact factor: 6.961

3.  Pain-Related Anxiety among Adults with Obesity and Chronic Pain: Relations with Pain, Opioid Misuse, and Mental Health.

Authors:  Andrew H Rogers; Brooke Y Kauffman; Lorra Garey; Gordon J G Asmundson; Michael J Zvolensky
Journal:  Behav Med       Date:  2020-10-14       Impact factor: 3.879

4.  Pharmacological fMRI provides evidence for opioidergic modulation of discrimination of facial pain expressions.

Authors:  Yili Zhao; Markus Rütgen; Lei Zhang; Claus Lamm
Journal:  Psychophysiology       Date:  2020-11-03       Impact factor: 4.016

Review 5.  Safety and efficacy of naltrexone for weight loss in adult patients - a systematic review.

Authors:  Agnieszka Kulak-Bejda; Grzegorz Bejda; Napoleon Waszkiewicz
Journal:  Arch Med Sci       Date:  2020-09-10       Impact factor: 3.318

  5 in total

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