Literature DB >> 27284492

Effects of modafinil and R-modafinil on brain stimulation reward thresholds: implications for their use in the treatment of psychostimulant dependence.

Brian T Burrows1, Lucas R Watterson1, Meagan A Johnson1, M Foster Olive2.   

Abstract

BACKGROUND: Modafinil and its enantiomer R-modafinil are approved for the treatment of various sleep disorders, and may also be efficacious in the treatment of psychostimulant abuse. However, the ability of modafinil and R-modafinil to alter brain reward function has not yet been assessed.
PURPOSE: This study assessed the effects of modafinil and R-modafinil on brain reward function using the intracranial self-stimulation (ICSS) paradigm. STUDY
DESIGN: Male Sprague-Dawley rats were trained to respond for ICSS using current-intensity threshold determination procedures. Changes in ICSS thresholds were then assessed following administration of modafinil and R-modafinil (50, 100, and 150 mg/kg), or cocaine (2.5 - 20 mg/kg) as a positive control.
RESULTS: ICSS thresholds were reduced by modafinil at the 150 mg/kg dose, as well as by cocaine at the 10 and 20 mg/kg doses. R-modafinil only produced non-significant trends towards reducing ICSS thresholds.
CONCLUSION: Modafinil and R-modafinil have limited effects on brain reward function in otherwise drug-naïve subjects. Additional assessments of these effects in the context of psychostimulant dependence are needed.

Entities:  

Keywords:  R-modafinil; abuse liability; cocaine; intracranial self-stimulation; modafinil; psychostimulant

Year:  2015        PMID: 27284492      PMCID: PMC4896318          DOI: 10.4303/jdar/235958

Source DB:  PubMed          Journal:  J Drug Alcohol Res        ISSN: 2090-8342


  37 in total

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Journal:  Biol Psychiatry       Date:  2012-04-25       Impact factor: 13.382

2.  Modafinil binds to the dopamine uptake carrier site with low affinity.

Authors:  E Mignot; S Nishino; C Guilleminault; W C Dement
Journal:  Sleep       Date:  1994-08       Impact factor: 5.849

3.  Potent rewarding and reinforcing effects of the synthetic cathinone 3,4-methylenedioxypyrovalerone (MDPV).

Authors:  Lucas R Watterson; Peter R Kufahl; Natali E Nemirovsky; Kaveish Sewalia; Megan Grabenauer; Brian F Thomas; Julie A Marusich; Scott Wegner; M Foster Olive
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4.  An evaluation of the abuse potential of modafinil using methylphenidate as a reference.

Authors:  D R Jasinski
Journal:  J Psychopharmacol       Date:  2000-03       Impact factor: 4.153

Review 5.  Modafinil: preclinical, clinical, and post-marketing surveillance--a review of abuse liability issues.

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Journal:  Ann Clin Psychiatry       Date:  2004 Apr-Jun       Impact factor: 1.567

6.  Interactions between modafinil and cocaine during the induction of conditioned place preference and locomotor sensitization in mice: implications for addiction.

Authors:  Tristan Shuman; Denise J Cai; Jennifer R Sage; Stephan G Anagnostaras
Journal:  Behav Brain Res       Date:  2012-08-03       Impact factor: 3.332

Review 7.  New treatments for cocaine dependence: a focused review.

Authors:  Laurent Karila; David Gorelick; Aviv Weinstein; Florence Noble; Amine Benyamina; Sarah Coscas; Lisa Blecha; William Lowenstein; Jean Luc Martinot; Michel Reynaud; Jean Pierre Lépine
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8.  Study of the addictive potential of modafinil in naive and cocaine-experienced rats.

Authors:  V Deroche-Gamonet; M Darnaudéry; L Bruins-Slot; F Piat; M Le Moal; P V Piazza
Journal:  Psychopharmacology (Berl)       Date:  2002-04-20       Impact factor: 4.530

9.  Smoked cocaine self-administration is decreased by modafinil.

Authors:  Carl L Hart; Margaret Haney; Suzanne K Vosburg; Eric Rubin; Richard W Foltin
Journal:  Neuropsychopharmacology       Date:  2007-06-13       Impact factor: 7.853

10.  The Reinforcing and Rewarding Effects of Methylone, a Synthetic Cathinone Commonly Found in "Bath Salts"

Authors:  Lucas R Watterson; Lauren Hood; Kaveish Sewalia; Seven E Tomek; Stephanie Yahn; Craig Trevor Johnson; Scott Wegner; Bruce E Blough; Julie A Marusich; M Foster Olive
Journal:  J Addict Res Ther       Date:  2012-12-01
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  3 in total

1.  Oral modafinil facilitates intracranial self-stimulation in rats: comparison with methylphenidate.

Authors:  Matthew F Lazenka; S Stevens Negus
Journal:  Behav Pharmacol       Date:  2017-06       Impact factor: 2.293

2.  R-Modafinil exerts weak effects on spatial memory acquisition and dentate gyrus synaptic plasticity.

Authors:  Bharanidharan Shanmugasundaram; Yogesh D Aher; Jana Aradska; Marija Ilic; Daniel Daba Feyissa; Predrag Kalaba; Nilima Y Aher; Vladimir Dragacevic; Babak Saber Marouf; Thierry Langer; Harald H Sitte; Harald Hoeger; Gert Lubec; Volker Korz
Journal:  PLoS One       Date:  2017-06-23       Impact factor: 3.240

Review 3.  Modafinil and its structural analogs as atypical dopamine uptake inhibitors and potential medications for psychostimulant use disorder.

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Journal:  Curr Opin Pharmacol       Date:  2020-09-11       Impact factor: 5.547

  3 in total

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