Literature DB >> 27177864

PIK3CA mutations are associated with reduced pathological complete response rates in primary HER2-positive breast cancer: pooled analysis of 967 patients from five prospective trials investigating lapatinib and trastuzumab.

S Loibl1, I Majewski2, V Guarneri3, V Nekljudova4, E Holmes5, E Bria6, C Denkert7, C Schem8, C Sotiriou9, S Loi10, M Untch11, P Conte3, R Bernards2, M Piccart9, G von Minckwitz4, J Baselga12.   

Abstract

BACKGROUND: The predictive value of PIK3CA mutations in HER2 positive (HER2+) breast cancer treated with neoadjuvant anti-HER2 and chemotherapy has been reported, but the power for subgroup analyses was lacking. PATIENTS AND METHODS: We combined individual patient data from five clinical trials evaluating PIK3CA mutations and associations with pathological complete response (pCR), disease-free survival (DFS) and overall survival (OS). Patients received either trastuzumab (T), lapatinib (L) or the combination T/L in addition to a taxane-based chemotherapy. PIK3CA was genotyped in tumour biopsies taken before therapy.
RESULTS: A total of 967 patients were included in this analysis; the median follow-up is 47 months. Overall, the pCR rate was significantly lower in the PIK3CA mutant compared with the wild-type group (16.2% versus 29.6%; P < 0.001). Within the hormone-receptor positive (HR+) subgroup, the PIK3CA mutant group had a pCR rate of only 7.6% compared with 24.2% in the wild-type group (P < 0.001). In contrast, in the HER2+/HR- group, there was no difference in pCR (27.2% versus 36.4%; P = 0.125) according to PIK3CA mutation status (interaction test P = 0.036). According to treatment arm, the pCR rate for mutant versus wild-type was 20.3% versus 27.1% for T (P = 0.343), 11.3% versus 16.9% for L (P = 0.369) and 16.7% versus 39.1% for T/L (P < 0.001). In the HR+ T/L group, the pCR rate was 5.5% versus 33.9% (interaction between HR and PIK3CA genotype P = 0.008). DFS and OS were not significantly different by mutation status, though the incidence rate of events was low. However, HR+/PIK3CA mutant patients seemed to have significantly worse DFS {hazard ratio (HR) 1.56 [95% confidence interval (CI) 1.00-2.45], P = 0.050; Pinteraction = 0.021}. T/L tended to improve DFS compared with T in the wild-type cohort, especially in the HR- group [HR 0.72, 95% CI (0.41-1.25), P = 0.242].
CONCLUSION: Overall PIK3CA mutant/HER2+ tumours had significantly lower pCR rates compared with wild-type tumours, however mainly confined to the HR+/PIK3CA mutant population. No definite conclusions can be drawn regarding survival.
© The Author 2016. Published by Oxford University Press on behalf of the European Society for Medical Oncology. All rights reserved. For permissions, please email: journals.permissions@oup.com.

Entities:  

Keywords:  HER2+ breast cancer; PIK3CA; double anti-HER2 treatment; neoadjuvant; pathological complete response; survival

Mesh:

Substances:

Year:  2016        PMID: 27177864      PMCID: PMC6279074          DOI: 10.1093/annonc/mdw197

Source DB:  PubMed          Journal:  Ann Oncol        ISSN: 0923-7534            Impact factor:   32.976


  22 in total

1.  Pertuzumab plus trastuzumab plus docetaxel for metastatic breast cancer.

Authors:  José Baselga; Javier Cortés; Sung-Bae Kim; Seock-Ah Im; Roberto Hegg; Young-Hyuck Im; Laslo Roman; José Luiz Pedrini; Tadeusz Pienkowski; Adam Knott; Emma Clark; Mark C Benyunes; Graham Ross; Sandra M Swain
Journal:  N Engl J Med       Date:  2011-12-07       Impact factor: 91.245

2.  Dual Blockade with AFatinib and Trastuzumab as NEoadjuvant Treatment for Patients with Locally Advanced or Operable Breast Cancer Receiving Taxane-Anthracycline Containing Chemotherapy-DAFNE (GBG-70).

Authors:  Claus Hanusch; Andreas Schneeweiss; Sibylle Loibl; Michael Untch; Stefan Paepke; Sherko Kümmel; Christian Jackisch; Jens Huober; Jörn Hilfrich; Bernd Gerber; Holger Eidtmann; Carsten Denkert; Serban Costa; Jens Uwe Blohmer; Knut Engels; Nicole Burchardi; Gunter von Minckwitz
Journal:  Clin Cancer Res       Date:  2015-03-30       Impact factor: 12.531

3.  Neoadjuvant carboplatin in patients with triple-negative and HER2-positive early breast cancer (GeparSixto; GBG 66): a randomised phase 2 trial.

Authors:  Gunter von Minckwitz; Andreas Schneeweiss; Sibylle Loibl; Christoph Salat; Carsten Denkert; Mahdi Rezai; Jens U Blohmer; Christian Jackisch; Stefan Paepke; Bernd Gerber; Dirk M Zahm; Sherko Kümmel; Holger Eidtmann; Peter Klare; Jens Huober; Serban Costa; Hans Tesch; Claus Hanusch; Jörn Hilfrich; Fariba Khandan; Peter A Fasching; Bruno V Sinn; Knut Engels; Keyur Mehta; Valentina Nekljudova; Michael Untch
Journal:  Lancet Oncol       Date:  2014-04-30       Impact factor: 41.316

4.  PIK3CA mutations are associated with decreased benefit to neoadjuvant human epidermal growth factor receptor 2-targeted therapies in breast cancer.

Authors:  Ian J Majewski; Paolo Nuciforo; Lorenza Mittempergher; Astrid J Bosma; Holger Eidtmann; Eileen Holmes; Christos Sotiriou; Debora Fumagalli; Jose Jimenez; Claudia Aura; Ludmila Prudkin; Maria Carmen Díaz-Delgado; Lorena de la Peña; Sherene Loi; Catherine Ellis; Nikolaus Schultz; Evandro de Azambuja; Nadia Harbeck; Martine Piccart-Gebhart; René Bernards; José Baselga
Journal:  J Clin Oncol       Date:  2015-01-05       Impact factor: 44.544

5.  Intrinsic subtypes, PIK3CA mutation, and the degree of benefit from adjuvant trastuzumab in the NSABP B-31 trial.

Authors:  Katherine L Pogue-Geile; Nan Song; Jong-Hyeon Jeong; Patrick G Gavin; Seong-Rim Kim; Nicole L Blackmon; Melanie Finnigan; Priya Rastogi; Louis Fehrenbacher; Eleftherios P Mamounas; Sandra M Swain; D Lawrence Wickerham; Charles E Geyer; Joseph P Costantino; Norman Wolmark; Soonmyung Paik
Journal:  J Clin Oncol       Date:  2015-01-05       Impact factor: 44.544

6.  Lapatinib versus trastuzumab in combination with neoadjuvant anthracycline-taxane-based chemotherapy (GeparQuinto, GBG 44): a randomised phase 3 trial.

Authors:  Michael Untch; Sibylle Loibl; Joachim Bischoff; Holger Eidtmann; Manfred Kaufmann; Jens-Uwe Blohmer; Jörn Hilfrich; Dirk Strumberg; Peter A Fasching; Rolf Kreienberg; Hans Tesch; Claus Hanusch; Bernd Gerber; Mahdi Rezai; Christian Jackisch; Jens Huober; Thorsten Kühn; Valentina Nekljudova; Gunter von Minckwitz
Journal:  Lancet Oncol       Date:  2012-01-17       Impact factor: 41.316

7.  Pertuzumab plus trastuzumab in combination with standard neoadjuvant anthracycline-containing and anthracycline-free chemotherapy regimens in patients with HER2-positive early breast cancer: a randomized phase II cardiac safety study (TRYPHAENA).

Authors:  A Schneeweiss; S Chia; T Hickish; V Harvey; A Eniu; R Hegg; C Tausch; J H Seo; Y-F Tsai; J Ratnayake; V McNally; G Ross; J Cortés
Journal:  Ann Oncol       Date:  2013-05-22       Impact factor: 32.976

8.  Double-blind, placebo-controlled, multicenter, randomized, phase IIb neoadjuvant study of letrozole-lapatinib in postmenopausal hormone receptor-positive, human epidermal growth factor receptor 2-negative, operable breast cancer.

Authors:  Valentina Guarneri; Daniele Giulio Generali; Antonio Frassoldati; Fabrizio Artioli; Corrado Boni; Luigi Cavanna; Enrico Tagliafico; Antonino Maiorana; Alberto Bottini; Katia Cagossi; Giancarlo Bisagni; Federico Piacentini; Guido Ficarra; Stefania Bettelli; Enrica Roncaglia; Simona Nuzzo; Ramona Swaby; Catherine Ellis; Clare Holford; Pierfranco Conte
Journal:  J Clin Oncol       Date:  2014-03-03       Impact factor: 44.544

9.  Determination of somatic oncogenic mutations linked to target-based therapies using MassARRAY technology.

Authors:  Maider Ibarrola-Villava; Tania Fleitas; Marta J Llorca-Cardeñosa; Cristina Mongort; Elisa Alonso; Samuel Navarro; Octavio Burgues; Ana Vivancos; Juan Miguel Cejalvo; José Alejandro Perez-Fidalgo; Susana Roselló; Gloria Ribas; Andrés Cervantes
Journal:  Oncotarget       Date:  2016-04-19

10.  Evaluating the predictive value of biomarkers for efficacy outcomes in response to pertuzumab- and trastuzumab-based therapy: an exploratory analysis of the TRYPHAENA study.

Authors:  Andreas Schneeweiss; Stephen Chia; Roberto Hegg; Christoph Tausch; Rahul Deb; Jayantha Ratnayake; Virginia McNally; Graham Ross; Astrid Kiermaier; Javier Cortés
Journal:  Breast Cancer Res       Date:  2014-07-08       Impact factor: 6.466

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  64 in total

1.  HER2-enriched subtype and pathological complete response in HER2-positive breast cancer: A systematic review and meta-analysis.

Authors:  Francesco Schettini; Tomás Pascual; Benedetta Conte; Nuria Chic; Fara Brasó-Maristany; Patricia Galván; Olga Martínez; Barbara Adamo; Maria Vidal; Montserrat Muñoz; Aranzazu Fernández-Martinez; Carla Rognoni; Gaia Griguolo; Valentina Guarneri; Pier Franco Conte; Mariavittoria Locci; Jan C Brase; Blanca Gonzalez-Farre; Patricia Villagrasa; Sabino De Placido; Rachel Schiff; Jamunarani Veeraraghavan; Mothaffar F Rimawi; C Kent Osborne; Sonia Pernas; Charles M Perou; Lisa A Carey; Aleix Prat
Journal:  Cancer Treat Rev       Date:  2020-01-17       Impact factor: 12.111

2.  Corrigendum: mdw197, mdw434 and mdw695.

Authors: 
Journal:  Ann Oncol       Date:  2018-04-01       Impact factor: 32.976

3.  Comparison of Three Real-Time PCR Assays for the Detection of PIK3CA Somatic Mutations in Formalin-Fixed Paraffin Embedded Tissues of Patients with Breast Carcinomas.

Authors:  A Lambert; J Salleron; M Lion; M Rouyer; N Lozano; A Leroux; J L Merlin; Alexandre Harlé
Journal:  Pathol Oncol Res       Date:  2018-11-13       Impact factor: 3.201

Review 4.  Neoadjuvant Model as a Platform for Research in Breast Cancer and Novel Targets under Development in this Field.

Authors:  Santiago Escrivá-de-Romaní; Miriam Arumí; Esther Zamora; Meritxell Bellet
Journal:  Breast Care (Basel)       Date:  2018-08-14       Impact factor: 2.860

5.  MK-2206 and Standard Neoadjuvant Chemotherapy Improves Response in Patients With Human Epidermal Growth Factor Receptor 2-Positive and/or Hormone Receptor-Negative Breast Cancers in the I-SPY 2 Trial.

Authors:  A Jo Chien; Debasish Tripathy; Kathy S Albain; W Fraser Symmans; Hope S Rugo; Michelle E Melisko; Anne M Wallace; Richard Schwab; Teresa Helsten; Andres Forero-Torres; Erica Stringer-Reasor; Erin D Ellis; Henry G Kaplan; Rita Nanda; Nora Jaskowiak; Rashmi Murthy; Constantine Godellas; Judy C Boughey; Anthony D Elias; Barbara B Haley; Kathleen Kemmer; Claudine Isaacs; Amy S Clark; Julie E Lang; Janice Lu; Larissa Korde; Kirsten K Edmiston; Donald W Northfelt; Rebecca K Viscusi; Douglas Yee; Jane Perlmutter; Nola M Hylton; Laura J Van't Veer; Angela DeMichele; Amy Wilson; Garry Peterson; Meredith B Buxton; Melissa Paoloni; Julia Clennell; Scott Berry; Jeffrey B Matthews; Katherine Steeg; Ruby Singhrao; Gillian L Hirst; Ashish Sanil; Christina Yau; Smita M Asare; Donald A Berry; Laura J Esserman
Journal:  J Clin Oncol       Date:  2019-02-07       Impact factor: 44.544

6.  Concurrent mutations associated with trastuzumab-resistance revealed by single cell sequencing.

Authors:  Yan Gao; Ning Wu; Shuai Wang; Xue Yang; Xin Wang; Bo Xu
Journal:  Breast Cancer Res Treat       Date:  2021-04-27       Impact factor: 4.872

Review 7.  De-escalation of treatment in HER2-positive breast cancer: Determinants of response and mechanisms of resistance.

Authors:  Jamunarani Veeraraghavan; Carmine De Angelis; Jorge S Reis-Filho; Tomás Pascual; Aleix Prat; Mothaffar F Rimawi; C Kent Osborne; Rachel Schiff
Journal:  Breast       Date:  2017-07-04       Impact factor: 4.380

8.  A multivariable prognostic score to guide systemic therapy in early-stage HER2-positive breast cancer: a retrospective study with an external evaluation.

Authors:  Aleix Prat; Valentina Guarneri; Laia Paré; Gaia Griguolo; Tomás Pascual; Maria V Dieci; Núria Chic; Blanca González-Farré; Antonio Frassoldati; Esther Sanfeliu; Juan M Cejalvo; Montserrat Muñoz; Giancarlo Bisagni; Fara Brasó-Maristany; Loredana Urso; Maria Vidal; Alba A Brandes; Barbara Adamo; Antonino Musolino; Federica Miglietta; Benedetta Conte; Mafalda Oliveira; Cristina Saura; Sònia Pernas; Jesús Alarcón; Antonio Llombart-Cussac; Javier Cortés; Luis Manso; Rafael López; Eva Ciruelos; Francesco Schettini; Patricia Villagrasa; Lisa A Carey; Charles M Perou; Federico Piacentini; Roberto D'Amico; Enrico Tagliafico; Joel S Parker; Pierfranco Conte
Journal:  Lancet Oncol       Date:  2020-11       Impact factor: 41.316

9.  What Is the Real Impact of Estrogen Receptor Status on the Prognosis and Treatment of HER2-Positive Early Breast Cancer?

Authors:  Mariana Brandão; Rafael Caparica; Luca Malorni; Aleix Prat; Lisa A Carey; Martine Piccart
Journal:  Clin Cancer Res       Date:  2020-02-11       Impact factor: 12.531

Review 10.  Towards personalized treatment for early stage HER2-positive breast cancer.

Authors:  Kristina Goutsouliak; Jamunarani Veeraraghavan; Vidyalakshmi Sethunath; Carmine De Angelis; C Kent Osborne; Mothaffar F Rimawi; Rachel Schiff
Journal:  Nat Rev Clin Oncol       Date:  2019-12-13       Impact factor: 66.675

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