Literature DB >> 27018419

Next-day residual effects of gabapentin, diphenhydramine, and triazolam on simulated driving performance in healthy volunteers: a phase 3, randomized, double-blind, placebo-controlled, crossover trial.

Gary G Kay1, Howard I Schwartz2, Mark A Wingertzahn3, Shyamalie Jayawardena3, Russell P Rosenberg4.   

Abstract

OBJECTIVE: Next-day residual effects of a nighttime dose of gabapentin 250 mg were evaluated on simulated driving performance in healthy participants in a randomized, placebo-controlled, double-blind, multicenter, four-period crossover study that included diphenhydramine citrate 76 mg and triazolam 0.5 mg.
METHODS: At treatment visits, participants (n = 59) were dosed at ~23:30, went to bed immediately, and awakened 6.5 h postdose for evaluation. The primary endpoint was the standard deviation of lateral position for the 100-km driving scenario. Additional measures of driving, sleepiness, and cognition were included.
RESULTS: Study sensitivity was established with triazolam, which demonstrated significant next-day impairment on all driving endpoints, relative to placebo (p < 0.001). Gabapentin demonstrated noninferiority to placebo on standard deviation of lateral position and speed deviation but not for lane excursions. Diphenhydramine citrate demonstrated significant impairment relative to gabapentin and placebo on speed deviation (p < 0.05). Other comparisons were either nonsignificant or statistically ineligible per planned, sequential comparisons. Secondary endpoints for sleepiness and cognitive performance were supportive of these conclusions.
CONCLUSIONS: Together, these data suggest that low-dose gabapentin had no appreciable next-day effects on simulated driving performance or cognitive functioning.
Copyright © 2016 John Wiley & Sons, Ltd. Copyright © 2016 John Wiley & Sons, Ltd.

Entities:  

Keywords:  diphenhydramine; gabapentin; residual effects; simulated driving performance; sleep

Mesh:

Substances:

Year:  2016        PMID: 27018419     DOI: 10.1002/hup.2530

Source DB:  PubMed          Journal:  Hum Psychopharmacol        ISSN: 0885-6222            Impact factor:   1.672


  7 in total

1.  Action Control Deficits in Patients With Essential Tremor.

Authors:  Shelby Hughes; Daniel O Claassen; Wery P M van den Wildenberg; Fenna T Phibbs; Elise B Bradley; Scott A Wylie; Nelleke C van Wouwe
Journal:  J Int Neuropsychol Soc       Date:  2018-12-03       Impact factor: 2.892

Review 2.  Medications for Sleep Schedule Adjustments in Athletes.

Authors:  Matthew B Baird; Irfan M Asif
Journal:  Sports Health       Date:  2017-11-21       Impact factor: 3.843

3.  Cross-sectional analysis of sleep-promoting and wake-promoting drug use on health, fatigue-related error, and near-crashes in police officers.

Authors:  Rowan P Ogeil; Laura K Barger; Steven W Lockley; Conor S O'Brien; Jason P Sullivan; Salim Qadri; Dan I Lubman; Charles A Czeisler; Shantha M W Rajaratnam
Journal:  BMJ Open       Date:  2018-09-19       Impact factor: 2.692

4.  Effects of lasmiditan on simulated driving performance: Results of two randomized, blinded, crossover studies with placebo and active controls.

Authors:  Eric M Pearlman; Darren Wilbraham; Ellen B Dennehy; Paul H Berg; Max Tsai; Erin G Doty; Gary G Kay
Journal:  Hum Psychopharmacol       Date:  2020-05-25       Impact factor: 1.672

5.  An assessment of the centrally acting muscle relaxant tolperisone on driving ability and cognitive effects compared to placebo and cyclobenzaprine.

Authors:  Judy Caron; Randall Kaye; Thomas Wessel; Amy Halseth; Gary Kay
Journal:  J Clin Pharm Ther       Date:  2020-05-10       Impact factor: 2.512

Review 6.  The Influence of Migraine on Driving: Current Understanding, Future Directions, and Potential Implications of Findings.

Authors:  Stewart J Tepper; Stephen D Silberstein; Noah L Rosen; Richard B Lipton; Ellen B Dennehy; Sherie A Dowsett; Erin Doty
Journal:  Headache       Date:  2019-12-02       Impact factor: 5.887

7.  A randomized, multicenter trial assessing the effects of rapastinel compared to ketamine, alprazolam, and placebo on simulated driving performance.

Authors:  Shengfang Su; Gary Kay; Thomas Hochadel; Jonathan Rojo; J Christopher Stein; Ramesh Boinpally; Antonia Periclou
Journal:  Clin Transl Sci       Date:  2021-11-07       Impact factor: 4.689

  7 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.