Literature DB >> 26989369

Clinical Effect of Switching from a Luteinizing Hormone-Releasing Hormone Agonist to an Antagonist in Patients with Castration-Resistant Prostate Cancer and Serum Testosterone Level ≥ 20 ng/dl.

Norihito Soga1, Takumi Kageyama1, Yuji Ogura1, Tomomi Yamada2, Norio Hayashi1.   

Abstract

INTRODUCTION: The efficacy of conversion from a luteinizing hormone-releasing hormone agonist to an antagonist was evaluated prospectively in patients with castration-resistant prostate cancer.
MATERIALS AND METHODS: From October 2012 to December 2014, 8 cases with a serum testosterone level ≥ 20 ng/dl during following androgen deprivation therapy were enrolled and received degarelix monthly. The primary end-pointgoal was to determine the effective prostate-specific antigen response rate. The secondary end-pointgoal was to assess the proportion of cases with a decrease in serum testosterone level to < 20 ng/ml.
RESULTS: One patient achieved a complete response, with a prostate-specific antigen level of 0.02 ng/ml at the nadirend of the study. The effective response rate was 25.0% (2/8), and the proportion of cases with prostate-specific antigen decline was 62.5% (5/8). In 5/8 cases (5/8, 62.5%), serum testosterone levels declined to < 20 ng/dl.
CONCLUSION: Switching to a luteinizing hormone-releasing hormone antagonist in patients with testosterone levels ≥ 20 ng/dl may be an option in sequential androgen deprivation therapy for some patients.

Entities:  

Keywords:  Castration-resistant; Degarelix; Luteinizing hormone-releasing hormone; Prostatic neoplasms; Testosterone

Year:  2016        PMID: 26989369      PMCID: PMC4789873          DOI: 10.1159/000442848

Source DB:  PubMed          Journal:  Curr Urol        ISSN: 1661-7649


  13 in total

1.  [EAU guidelines on prostate cancer. Part II: treatment of advanced, relapsing, and castration-resistant prostate cancer].

Authors:  N Mottet; J Bellmunt; M Bolla; S Joniau; M Mason; V Matveev; H P Schmid; T van der Kwast; T Wiegel; F Zattoni; A Heidenreich
Journal:  Actas Urol Esp       Date:  2011-07-14       Impact factor: 0.994

Review 2.  Castration-resistant prostate cancer: current and emerging treatment strategies.

Authors:  Giuseppe Di Lorenzo; Carlo Buonerba; Riccardo Autorino; Sabino De Placido; Cora N Sternberg
Journal:  Drugs       Date:  2010-05-28       Impact factor: 9.546

3.  The long-term results with delayed-combined androgen blockade therapy in local or locally advanced prostate cancer.

Authors:  Norihito Soga; Yasuhide Hori; Yuji Ogura; Norio Hayashi; Yoshiki Sugimura
Journal:  Jpn J Clin Oncol       Date:  2012-03-20       Impact factor: 3.019

4.  Efficacy and safety of androgen deprivation therapy after switching from monthly leuprolide to monthly degarelix in patients with prostate cancer.

Authors:  J de la Rosette; R Davis; D Frankel; T Kold Olesen
Journal:  Int J Clin Pract       Date:  2011-02-22       Impact factor: 2.503

5.  Reassessment of the definition of castrate levels of testosterone: implications for clinical decision making.

Authors:  M G Oefelein; A Feng; M J Scolieri; D Ricchiutti; M I Resnick
Journal:  Urology       Date:  2000-12-20       Impact factor: 2.649

6.  Effect of enzalutamide on health-related quality of life, pain, and skeletal-related events in asymptomatic and minimally symptomatic, chemotherapy-naive patients with metastatic castration-resistant prostate cancer (PREVAIL): results from a randomised, phase 3 trial.

Authors:  Yohann Loriot; Kurt Miller; Cora N Sternberg; Karim Fizazi; Johann S De Bono; Simon Chowdhury; Celestia S Higano; Sarah Noonberg; Stefan Holmstrom; Harry Mansbach; Frank G Perabo; De Phung; Cristina Ivanescu; Konstantina Skaltsa; Tomasz M Beer; Bertrand Tombal
Journal:  Lancet Oncol       Date:  2015-04-14       Impact factor: 41.316

7.  A switch from GnRH agonist to GnRH antagonist in castration-resistant prostate cancer patients leads to a low response rate on PSA.

Authors:  Alexandra Masson-Lecomte; Laurent Guy; Philippe Pedron; Franck Bruyere; Morgan Rouprêt; Bonaventure Nsabimbona; Mickael Dahan; Patrice Hoffman; Laurent Salomon; Dimitri Vordos; Andras Hoznek; Philippe Le Corvoisier; Pierrick Morel; Claude Abbou; Alexandre de la Taille
Journal:  World J Urol       Date:  2012-04-15       Impact factor: 4.226

8.  A phase III extension trial with a 1-arm crossover from leuprolide to degarelix: comparison of gonadotropin-releasing hormone agonist and antagonist effect on prostate cancer.

Authors:  E David Crawford; Bertrand Tombal; Kurt Miller; Laurent Boccon-Gibod; Fritz Schröder; Neal Shore; Judd W Moul; Jens-Kristian Jensen; Tine Kold Olesen; Bo-Eric Persson
Journal:  J Urol       Date:  2011-07-23       Impact factor: 7.450

9.  The efficacy and safety of degarelix: a 12-month, comparative, randomized, open-label, parallel-group phase III study in patients with prostate cancer.

Authors:  Laurence Klotz; Laurent Boccon-Gibod; Neal D Shore; Cal Andreou; Bo-Eric Persson; Per Cantor; Jens-Kristian Jensen; Tine Kold Olesen; Fritz H Schröder
Journal:  BJU Int       Date:  2008-12       Impact factor: 5.588

10.  Redefining clinically significant castration levels in patients with prostate cancer receiving continuous androgen deprivation therapy.

Authors:  Juan Morote; Anna Orsola; Jacques Planas; Enrique Trilla; Carles X Raventós; Lluís Cecchini; Roberto Catalán
Journal:  J Urol       Date:  2007-08-14       Impact factor: 7.450

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  3 in total

Review 1.  Maximal testosterone suppression in the management of recurrent and metastatic prostate cancer.

Authors:  Laurence Klotz; Rodney H Breau; Loretta L Collins; Martin E Gleave; Tom Pickles; Frederic Pouliot; Fred Saad
Journal:  Can Urol Assoc J       Date:  2017 Jan-Feb       Impact factor: 1.862

2.  Switching from a gonadotropin-releasing hormone (GnRH) agonist to a GnRH antagonist in prostate cancer patients: A systematic review and meta-analysis.

Authors:  Kaleem S Atchia; Christopher J D Wallis; Neil Fleshner; Paul Toren
Journal:  Can Urol Assoc J       Date:  2019-07-23       Impact factor: 1.862

Review 3.  Androgen-targeted therapy in men with prostate cancer: evolving practice and future considerations.

Authors:  E David Crawford; Axel Heidenreich; Nathan Lawrentschuk; Bertrand Tombal; Antonio C L Pompeo; Arturo Mendoza-Valdes; Kurt Miller; Frans M J Debruyne; Laurence Klotz
Journal:  Prostate Cancer Prostatic Dis       Date:  2018-08-21       Impact factor: 5.554

  3 in total

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