Literature DB >> 26839440

Direct C7 Functionalization of Tryptophan. Synthesis of Methyl (S)-2-((tert-Butoxycarbonyl)amino)-3-(7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indol-3-yl)propanoate.

Kazuma Amaike1, Richard P Loach1, Mohammad Movassaghi1.   

Abstract

Entities:  

Year:  2015        PMID： 26839440      PMCID： PMC4733874          DOI： 10.15227/orgsyn.092.0373

Source DB:  PubMed          Journal:  Organic Synth        ISSN： 0078-6209


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  46 in total

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Journal:  Angew Chem Int Ed Engl       Date:  2011-02-17       Impact factor: 15.336

6.  Iridium-catalyzed, silyl-directed borylation of nitrogen-containing heterocycles.

Authors:  Daniel W Robbins; Timothy A Boebel; John F Hartwig
Journal:  J Am Chem Soc       Date:  2010-03-31       Impact factor: 15.419

7.  Identification of pyrrolo[2,3-g]indazoles as new Pim kinase inhibitors.

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8.  Boc groups as protectors and directors for Ir-catalyzed C-H borylation of heterocycles.

Authors:  Venkata A Kallepalli; Feng Shi; Sulagna Paul; Edith N Onyeozili; Robert E Maleczka; Milton R Smith
Journal:  J Org Chem       Date:  2009-12-04       Impact factor: 4.354

9.  Scope of the Suzuki-Miyaura cross-coupling reactions of potassium heteroaryltrifluoroborates.

Authors:  Gary A Molander; Belgin Canturk; Lauren E Kennedy
Journal:  J Org Chem       Date:  2009-02-06       Impact factor: 4.354

10.  C7-derivatization of C3-alkylindoles including tryptophans and tryptamines.

Authors:  Richard P Loach; Owen S Fenton; Kazuma Amaike; Dustin S Siegel; Erhan Ozkal; Mohammad Movassaghi
Journal:  J Org Chem       Date:  2014-11-10       Impact factor: 4.354
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2.  Enantioselective Synthesis of (-)-Vallesine: Late-Stage C17-Oxidation via Complex Indole Boronation.

Authors:  Alyssa H Antropow; Nicholas R Garcia; Kolby L White; Mohammad Movassaghi
Journal:  Org Lett       Date:  2018-06-04       Impact factor: 6.005

3.  Regioselective Diversification of 2,1-Borazaronaphthalenes: Unlocking Isosteric Space via C-H Activation.

Authors:  Geraint H M Davies; Matthieu Jouffroy; Fatemeh Sherafat; Borna Saeednia; Casey Howshall; Gary A Molander
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  3 in total

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