Literature DB >> 26732384

Diagnostic performance and safety of NMK36 (trans-1-amino-3-[18F]fluorocyclobutanecarboxylic acid)-PET/CT in primary prostate cancer: multicenter Phase IIb clinical trial.

Hiroyoshi Suzuki1, Yusuke Inoue2, Hiroyuki Fujimoto3, Junji Yonese4, Kazunari Tanabe5, Satoshi Fukasawa6, Tomio Inoue7, Shiro Saito8, Munehisa Ueno9, Akiharu Otaka10.   

Abstract

OBJECTIVE: We performed a multicenter Phase IIb clinical trial of NMK36, a novel amino acid analog for positron emission tomography containing trans-1-amino-3-[(18)F]fluorocyclobutanecarboxylic acid, to evaluate its safety and diagnostic performance for primary prostate cancer.
METHODS: Sixty-eight subjects with primary prostate cancer scheduled for radical prostatectomy or hormone therapy underwent whole-body positron emission tomography/computed tomography after injection of NMK36. The diagnostic performances of NMK36-positron emission tomography/computed tomography were evaluated for (i) regional lymph node metastasis: comparison with contrast-enhanced computed tomography under setting reference standard (histopathology or 6-month follow-up), (ii) bone metastasis: concordance rate with conventional imaging (combination of bone scintigraphy and contrast-enhanced computed tomography) and (iii) primary lesion: comparison with histopathological findings.
RESULTS: The accuracy of NMK36-positron emission tomography/computed tomography and contrast-enhanced computed tomography for regional lymph node metastasis were 85.5 and 87.3%, respectively. NMK36-positron emission tomography/computed tomography showed positive findings for regional lymph nodes with short-axis diameters of 5-9 mm at 23 regions in 13 patients of hormone therapy cohort, but they were not confirmed with reference standard in this study. The concordance rate of NMK36-positron emission tomography/computed tomography with conventional imaging for bone metastases was 83.3%, and seven patients had positive findings only by NMK36-positron emission tomography/computed tomography. The sensitivity and specificity of NMK36-positron emission tomography/computed tomography for primary lesion in six-segment analysis was 92.5 and 90.1%, respectively. Seven of non-serious adverse events were observed in six patients.
CONCLUSIONS: This study showed the comparable diagnostic performance of NMK36-positron emission tomography/computed tomography compared with conventional imaging. Some lesions of lymph node and bone were positive solely by NMK36-positron emission tomography/computed tomography, which needs to be confirmed with reference standard in future study to evaluate the usefulness of NMK36-positron emission tomography/computed tomography in staging prostate cancer.
© The Author 2016. Published by Oxford University Press. All rights reserved. For Permissions, please email: journals.permissions@oup.com.

Entities:  

Keywords:  NMK36; anti-[18F]FACBC; clinical trial; positron emission tomography; prostate cancer

Mesh:

Substances:

Year:  2016        PMID: 26732384     DOI: 10.1093/jjco/hyv181

Source DB:  PubMed          Journal:  Jpn J Clin Oncol        ISSN: 0368-2811            Impact factor:   3.019


  14 in total

Review 1.  PET Tracers Beyond FDG in Prostate Cancer.

Authors:  David M Schuster; Cristina Nanni; Stefano Fanti
Journal:  Semin Nucl Med       Date:  2016-09-07       Impact factor: 4.446

2.  18F-Fluciclovine PET/MRI for preoperative lymph node staging in high-risk prostate cancer patients.

Authors:  Kirsten M Selnæs; Brage Krüger-Stokke; Mattijs Elschot; Frode Willoch; Øystein Størkersen; Elise Sandsmark; Siver A Moestue; May-Britt Tessem; Dag Halvorsen; Eirik Kjøbli; Anders Angelsen; Sverre Langørgen; Helena Bertilsson; Tone F Bathen
Journal:  Eur Radiol       Date:  2018-01-02       Impact factor: 5.315

3.  18F-Fluciclovine versus PSMA PET Imaging in Primary Tumor Detection during Initial Staging of High-Risk Prostate Cancer: A Systematic Review and Meta-Analysis.

Authors:  Divya Yadav; Hyunsoo Hwang; Wei Qiao; Rituraj Upadhyay; Brian F Chapin; Chad Tang; Ana Aparicio; Maria A Lopez-Olivo; Stella K Kang; Homer A Macapinlac; Tharakeswara K Bathala; Devaki Shilpa Surasi
Journal:  Radiol Imaging Cancer       Date:  2022-03

Review 4.  Role of molecular imaging in the detection of localized prostate cancer.

Authors:  Samuel J Galgano; Janelle T West; Soroush Rais-Bahrami
Journal:  Ther Adv Urol       Date:  2022-06-21

5.  Diagnostic Performance of 18F-Fluciclovine in Detection of Prostate Cancer Bone Metastases.

Authors:  Albert Chau; Peter Gardiner; Patrick M Colletti; Hossein Jadvar
Journal:  Clin Nucl Med       Date:  2018-07       Impact factor: 7.794

6.  PET Tracer 18F-Fluciclovine Can Detect Histologically Proven Bone Metastatic Lesions: A Preclinical Study in Rat Osteolytic and Osteoblastic Bone Metastasis Models.

Authors:  Shuntaro Oka; Masaru Kanagawa; Yoshihiro Doi; David M Schuster; Mark M Goodman; Hirokatsu Yoshimura
Journal:  Theranostics       Date:  2017-05-15       Impact factor: 11.556

Review 7.  Fluorine-18 labeled amino acids for tumor PET/CT imaging.

Authors:  Yiqiang Qi; Xiaohui Liu; Jun Li; Huiqian Yao; Shuanghu Yuan
Journal:  Oncotarget       Date:  2017-08-04

Review 8.  Novel PET imaging methods for prostate cancer.

Authors:  Esther Mena; Peter C Black; Soroush Rais-Bahrami; Michael Gorin; Mohamad Allaf; Peter Choyke
Journal:  World J Urol       Date:  2020-07-15       Impact factor: 4.226

9.  Assessment of Amino Acid/Drug Transporters for Renal Transport of [18F]Fluciclovine (anti-[18F]FACBC) in Vitro.

Authors:  Masahiro Ono; Atsumi Baden; Hiroyuki Okudaira; Masato Kobayashi; Keiichi Kawai; Shuntaro Oka; Hirokatsu Yoshimura
Journal:  Int J Mol Sci       Date:  2016-10-14       Impact factor: 5.923

Review 10.  Surgical management of high-risk, localized prostate cancer.

Authors:  Lamont J Wilkins; Jeffrey J Tosoian; Debasish Sundi; Ashley E Ross; Dominic Grimberg; Eric A Klein; Brian F Chapin; Yaw A Nyame
Journal:  Nat Rev Urol       Date:  2020-11-10       Impact factor: 14.432

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