Literature DB >> 26641128

An Investigation of (Diacetoxyiodo)arenes as Precursors for Preparing No-Carrier-Added [(18)F]Fluoroarenes from Cyclotron-Produced [(18)F]Fluoride Ion.

Mohammad B Haskali1, Sanjay Telu1, Yong-Sok Lee2, Cheryl L Morse1, Shuiyu Lu1, Victor W Pike1.   

Abstract

Treatment of (diacetoxyiodo)arenes (1a-1u) with cyclotron-produced [(18)F]fluoride ion rapidly affords no-carrier-added [(18)F]fluoroarenes (2a-2u) in useful yields and constitutes a new method for converting substituted iodoarenes into substituted [(18)F]fluoroarenes in just two steps.

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Year:  2015        PMID： 26641128      PMCID： PMC5573187          DOI： 10.1021/acs.joc.5b02332

Source DB:  PubMed          Journal:  J Org Chem        ISSN： 0022-3263            Impact factor:   4.354


  12 in total

1.  Regiospecific syntheses of functionalized diaryliodonium tosylates via [hydroxy(tosyloxy)iodo]arenes generated in situ from (diacetoxyiodo)arenes.

Authors:  Joong-Hyun Chun; Victor W Pike
Journal:  J Org Chem       Date:  2012-02-09       Impact factor: 4.354

2.  Fully automated preparation of n.c.a. 4-[18F]fluorobenzoic acid and N-succinimidyl 4-[18F]fluorobenzoate using a Siemens/CTI chemistry process control unit (CPCU).

Authors:  Jan Marik; Julie L Sutcliffe
Journal:  Appl Radiat Isot       Date:  2006-08-28       Impact factor: 1.513

3.  Rapid and Efficient Radiosyntheses of Meta-substituted [F]Fluoroarenes from [F]Fluoride Ion and Diaryliodonium Tosylates within a Microreactor.

Authors:  Joong-Hyun Chun; Shuiyu Lu; Victor W Pike
Journal:  European J Org Chem       Date:  2011-08

Review 4.  18F labeling of arenes.

Authors:  Matthew Tredwell; Véronique Gouverneur
Journal:  Angew Chem Int Ed Engl       Date:  2012-10-19       Impact factor: 15.336

5.  Fast and high-yield microreactor syntheses of ortho-substituted [(18)F]fluoroarenes from reactions of [(18)F]fluoride ion with diaryliodonium salts.

Authors:  Joong-Hyun Chun; Shuiyu Lu; Yong-Sok Lee; Victor W Pike
Journal:  J Org Chem       Date:  2010-05-21       Impact factor: 4.354

6.  Labeling proteins with fluorine-18 using N-succinimidyl 4-[18F]fluorobenzoate.

Authors:  G Vaidyanathan; M R Zalutsky
Journal:  Int J Rad Appl Instrum B       Date:  1992-04

7.  A method for detecting water in organic solvents.

Authors:  Haoran Sun; Bijia Wang; Stephen G DiMagno
Journal:  Org Lett       Date:  2008-09-12       Impact factor: 6.005

8.  Diaryliodonium salts: a journey from obscurity to fame.

Authors:  Eleanor A Merritt; Berit Olofsson
Journal:  Angew Chem Int Ed Engl       Date:  2009       Impact factor: 15.336

9.  Nucleophilic 18F-fluorination of heteroaromatic iodonium salts with no-carrier-added [18F]fluoride.

Authors:  Tobias L Ross; Johannes Ermert; Carsten Hocke; Heinz H Coenen
Journal:  J Am Chem Soc       Date:  2007-05-31       Impact factor: 15.419

10.  Single-step syntheses of no-carrier-added functionalized [18F]fluoroarenes as labeling synthons from diaryliodonium salts.

Authors:  Joong-Hyun Chun; Victor W Pike
Journal:  Org Biomol Chem       Date:  2013-10-07       Impact factor: 3.876
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  2 in total

Review 1.  Chemistry for Positron Emission Tomography: Recent Advances in 11 C-, 18 F-, 13 N-, and 15 O-Labeling Reactions.

Authors:  Xiaoyun Deng; Jian Rong; Lu Wang; Neil Vasdev; Lei Zhang; Lee Josephson; Steven H Liang
Journal:  Angew Chem Int Ed Engl       Date:  2019-01-14       Impact factor: 15.336

2.  Cu-Mediated C-H 18F-Fluorination of Electron-Rich (Hetero)arenes.

Authors:  Matthew S McCammant; Stephen Thompson; Allen F Brooks; Shane W Krska; Peter J H Scott; Melanie S Sanford
Journal:  Org Lett       Date:  2017-06-30       Impact factor: 6.005
  2 in total

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