Literature DB >> 26519363

Doublet BRAF/MEK inhibition versus single-agent BRAF inhibition in the management of BRAF-mutant advanced melanoma, biological rationale and meta-analysis of published data.

O Abdel-Rahman1, H ElHalawani2, H Ahmed3.   

Abstract

BACK GROUND: We executed a comparative systematic review and meta-analysis of the efficacy and toxicity of doublet BRAF/MEK inhibition versus single-agent BRAF inhibitor in the management of BRAF-mutant advanced melanoma.
METHODS: Eligible studies included prospective studies evaluating doublet regimens versus BRAF-inhibitor monotherapy for the management of BRAF-mutant advanced melanoma.
RESULTS: Our search strategy yielded 200 potentially relevant citations from searched databases. After preclusion of ineligible studies, four studies were included in the final analysis. Efficacy analyses demonstrate that BRAF/MEK inhibition strategy is associated with a significant improvement in ORR [OR 1.35; 95 % CI (1.16, 1.58); P = 0.0002], PFS [HR 0.56; 95 % CI (0.49, 0.64); P < 0.00001] and OS [HR 0.70; 95 % CI (0.58, 0.84); P = 0.0001]. Moreover, this combination is associated with a higher RR for diarrhea [1.30; 95 % CI (1.30, 1.49); P = 0.0002], decreased ejection fraction [4.63; 95 % CI (2.56, 8.37); P = <0.00001], acneiform dermatitis [1.61; 95 % CI (1.03, 2.53); P = 0.04] and pyrexia [1.98; 95 % CI (1.72, 2.27); P < 0.00001].
CONCLUSIONS: Our meta-analysis has demonstrated that combination of MEK/BRAF inhibitors is associated with higher ORR, PFS and OS. However, this comes at the expense of a higher risk of selected toxicities.

Entities:  

Keywords:  Dabrafenib; Melanoma; Trametinib; Vemurafenib

Mesh:

Substances:

Year:  2015        PMID: 26519363     DOI: 10.1007/s12094-015-1438-0

Source DB:  PubMed          Journal:  Clin Transl Oncol        ISSN: 1699-048X            Impact factor:   3.405


  28 in total

1.  Improved overall survival in melanoma with combined dabrafenib and trametinib.

Authors:  Caroline Robert; Boguslawa Karaszewska; Jacob Schachter; Piotr Rutkowski; Andrzej Mackiewicz; Daniil Stroiakovski; Michael Lichinitser; Reinhard Dummer; Florent Grange; Laurent Mortier; Vanna Chiarion-Sileni; Kamil Drucis; Ivana Krajsova; Axel Hauschild; Paul Lorigan; Pascal Wolter; Georgina V Long; Keith Flaherty; Paul Nathan; Antoni Ribas; Anne-Marie Martin; Peng Sun; Wendy Crist; Jeff Legos; Stephen D Rubin; Shonda M Little; Dirk Schadendorf
Journal:  N Engl J Med       Date:  2014-11-16       Impact factor: 91.245

2.  Combined BRAF and MEK inhibition versus BRAF inhibition alone in melanoma.

Authors:  Georgina V Long; Daniil Stroyakovskiy; Helen Gogas; Evgeny Levchenko; Filippo de Braud; James Larkin; Claus Garbe; Thomas Jouary; Axel Hauschild; Jean Jacques Grob; Vanna Chiarion Sileni; Celeste Lebbe; Mario Mandalà; Michael Millward; Ana Arance; Igor Bondarenko; John B A G Haanen; Johan Hansson; Jochen Utikal; Virginia Ferraresi; Nadezhda Kovalenko; Peter Mohr; Volodymyr Probachai; Dirk Schadendorf; Paul Nathan; Caroline Robert; Antoni Ribas; Douglas J DeMarini; Jhangir G Irani; Michelle Casey; Daniele Ouellet; Anne-Marie Martin; Ngocdiep Le; Kiran Patel; Keith Flaherty
Journal:  N Engl J Med       Date:  2014-09-29       Impact factor: 91.245

Review 3.  RAF protein-serine/threonine kinases: structure and regulation.

Authors:  Robert Roskoski
Journal:  Biochem Biophys Res Commun       Date:  2010-07-30       Impact factor: 3.575

4.  [Cutaneous side effects of anti-tumor therapy with BRAF and MEK inhibitors].

Authors:  R Gutzmer; J C Hassel; K C Kähler; C Loquai; R Mössner; S Ugurel; L Zimmer; Für Komitee Kutane Nebenwirkungen Ado der das Ado
Journal:  Hautarzt       Date:  2014-07       Impact factor: 0.751

5.  Overall survival in patients with metastatic melanoma.

Authors:  Xue Song; Zhongyun Zhao; Beth Barber; Amanda M Farr; Boris Ivanov; Marilyn Novich
Journal:  Curr Med Res Opin       Date:  2015-03-18       Impact factor: 2.580

Review 6.  Gaining momentum: New options and opportunities for the treatment of advanced melanoma.

Authors:  Olivier Michielin; Christoph Hoeller
Journal:  Cancer Treat Rev       Date:  2015-06-04       Impact factor: 12.111

7.  Cutaneous Toxic Effects of BRAF Inhibitors Alone and in Combination With MEK Inhibitors for Metastatic Melanoma.

Authors:  Giuliana Carlos; Rachael Anforth; Arthur Clements; Alexander M Menzies; Matteo S Carlino; Shaun Chou; Pablo Fernandez-Peñas
Journal:  JAMA Dermatol       Date:  2015-10       Impact factor: 10.282

8.  Survival in BRAF V600-mutant advanced melanoma treated with vemurafenib.

Authors:  Jeffrey A Sosman; Kevin B Kim; Lynn Schuchter; Rene Gonzalez; Anna C Pavlick; Jeffrey S Weber; Grant A McArthur; Thomas E Hutson; Stergios J Moschos; Keith T Flaherty; Peter Hersey; Richard Kefford; Donald Lawrence; Igor Puzanov; Karl D Lewis; Ravi K Amaravadi; Bartosz Chmielowski; H Jeffrey Lawrence; Yu Shyr; Fei Ye; Jiang Li; Keith B Nolop; Richard J Lee; Andrew K Joe; Antoni Ribas
Journal:  N Engl J Med       Date:  2012-02-23       Impact factor: 91.245

Review 9.  Risk of selected dermatological toxicities in cancer patients treated with MEK inhibitors: a comparative systematic review and meta-analysis.

Authors:  Omar Abdel-Rahman; Hesham ElHalawani; Hoda Ahmed
Journal:  Future Oncol       Date:  2015-11-12       Impact factor: 3.404

Review 10.  Risk of Selected Cardiovascular Toxicities in Patients With Cancer Treated With MEK Inhibitors: A Comparative Systematic Review and Meta-Analysis.

Authors:  Omar Abdel-Rahman; Hesham ElHalawani; Hoda Ahmed
Journal:  J Glob Oncol       Date:  2015-11-25
View more
  9 in total

Review 1.  Comprehensive review of cardiovascular toxicity of drugs and related agents.

Authors:  Přemysl Mladěnka; Lenka Applová; Jiří Patočka; Vera Marisa Costa; Fernando Remiao; Jana Pourová; Aleš Mladěnka; Jana Karlíčková; Luděk Jahodář; Marie Vopršalová; Kurt J Varner; Martin Štěrba
Journal:  Med Res Rev       Date:  2018-01-05       Impact factor: 12.944

Review 2.  Cutaneous toxicities of new treatments for melanoma.

Authors:  A Boada; C Carrera; S Segura; H Collgros; P Pasquali; D Bodet; S Puig; J Malvehy
Journal:  Clin Transl Oncol       Date:  2018-05-24       Impact factor: 3.405

3.  Automatic extraction of quantitative data from ClinicalTrials.gov to conduct meta-analyses.

Authors:  Richeek Pradhan; David C Hoaglin; Matthew Cornell; Weisong Liu; Victoria Wang; Hong Yu
Journal:  J Clin Epidemiol       Date:  2018-09-23       Impact factor: 6.437

Review 4.  Updates in Therapy for Advanced Melanoma.

Authors:  Bhavana P Singh; April K S Salama
Journal:  Cancers (Basel)       Date:  2016-01-15       Impact factor: 6.639

Review 5.  Efficacy and safety of BRAF inhibition alone versus combined BRAF and MEK inhibition in melanoma: a meta-analysis of randomized controlled trials.

Authors:  Mengdong Liu; Xuekang Yang; Jiaqi Liu; Bin Zhao; Weixia Cai; Yan Li; Dahai Hu
Journal:  Oncotarget       Date:  2017-05-09

Review 6.  Tolerability of BRAF/MEK inhibitor combinations: adverse event evaluation and management.

Authors:  Lucie Heinzerling; Thomas K Eigentler; Michael Fluck; Jessica C Hassel; Daniela Heller-Schenck; Jan Leipe; Matthias Pauschinger; Arndt Vogel; Lisa Zimmer; Ralf Gutzmer
Journal:  ESMO Open       Date:  2019-05-23

Review 7.  Clinical outcomes of BRAF plus MEK inhibition in melanoma: A meta-analysis and systematic review.

Authors:  Qingliang Yu; Jiayi Xie; Jiangmiao Li; Yunxin Lu; Liang Liao
Journal:  Cancer Med       Date:  2019-08-08       Impact factor: 4.452

8.  Cardiovascular Adverse Events Associated With BRAF and MEK Inhibitors: A Systematic Review and Meta-analysis.

Authors:  Raluca I Mincu; Amir A Mahabadi; Lars Michel; Simone M Mrotzek; Dirk Schadendorf; Tienush Rassaf; Matthias Totzeck
Journal:  JAMA Netw Open       Date:  2019-08-02

9.  Cardiovascular Toxicity of Targeted Therapies for Cancer: An Overview of Systematic Reviews.

Authors:  Marina T Van Leeuwen; Steven Luu; Howard Gurney; Martin R Brown; Sallie-Anne Pearson; Kate Webber; Lee Hunt; Soojung Hong; Geoffrey P Delaney; Claire M Vajdic
Journal:  JNCI Cancer Spectr       Date:  2020-08-24
  9 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.