Literature DB >> 26513009

Effects of metformin on clinical outcome in diabetic patients with advanced HCC receiving sorafenib.

Andrea Casadei Gardini1, Giorgia Marisi2, Emanuela Scarpi3, Mario Scartozzi4, Luca Faloppi5, Nicola Silvestris6, Gianluca Masi7, Caterina Vivaldi7, Oronzo Brunetti6, Stefano Tamberi8, Francesco Giuseppe Foschi9, Emiliano Tamburini10, Elena Tenti11, Salvatore Ricca Rosellini12, Paola Ulivi2, Stefano Cascinu5, Oriana Nanni3, Giovanni Luca Frassineti1.   

Abstract

BACKGROUND AND
OBJECTIVE: Several studies have reported an association between type 2 diabetes mellitus and hepatocellular carcinoma (HCC). Data from several retrospective studies and meta-analyses have highlighted a reduction of about 50% in the risk of developing HCC in cirrhotic patients treated with metformin for diabetes. The aim of this study was to evaluate the different outcomes of patients who received or did not receive metformin during treatment with sorafenib.
METHODS: We analyzed 93 patients consecutively treated with sorafenib. Forty-two (45.2%) patients were diabetic, of whom 31 were on metformin. Progression-free survival (PFS) and overall survival (OS) were estimated with the Kaplan-Meier method and compared with the log-rank test.
RESULTS: The concomitant use of sorafenib and metformin was associated with a median PFS of 2.6 months (95% CI 1.9-3.3) compared to 5.0 months (95% CI 2.5-8.2) for patients receiving sorafenib alone (p = 0.029). The median OS of patients treated with the combination was 10.4 months (95% CI 3.9-14.4) compared to 15.1 months (95% CI 11.7-17.8) for those who were not given metformin (p = 0.014).
CONCLUSIONS: Our findings could be the result of increased tumor aggressiveness and resistance to sorafenib in metformin-treated patients.

Entities:  

Keywords:  diabetes; hepatocellular carcinoma; insulin; metformin; sorafenib

Mesh:

Substances:

Year:  2015        PMID: 26513009     DOI: 10.1517/14656566.2015.1102887

Source DB:  PubMed          Journal:  Expert Opin Pharmacother        ISSN: 1465-6566            Impact factor:   3.889


  36 in total

1.  Association of liver cirrhosis severity with type 2 diabetes mellitus in hepatocellular carcinoma.

Authors:  Ankita Makol; Shruthi Kanthaje; Radha K Dhiman; Naveen Kalra; Yogesh K Chawla; Anuradha Chakraborti
Journal:  Exp Biol Med (Maywood)       Date:  2017-11-29

Review 2.  Roles of mitochondria in liver cancer stem cells.

Authors:  Ching-Wen Chang; Jeng-Fan Lo; Xin Wei Wang
Journal:  Differentiation       Date:  2019-05-30       Impact factor: 3.880

3.  Sorafenib and metformin: to be, or not to be, that is the question.

Authors:  Giulia Orsi; Andrea Casadei-Gardini
Journal:  Hepatobiliary Surg Nutr       Date:  2019-08       Impact factor: 7.293

Review 4.  Diabetes mellitus and metformin in hepatocellular carcinoma.

Authors:  Koji Fujita; Hisakazu Iwama; Hisaaki Miyoshi; Joji Tani; Kyoko Oura; Tomoko Tadokoro; Teppei Sakamoto; Takako Nomura; Asahiro Morishita; Hirohito Yoneyama; Tsutomu Masaki
Journal:  World J Gastroenterol       Date:  2016-07-21       Impact factor: 5.742

5.  Metformin prevents liver tumourigenesis by attenuating fibrosis in a transgenic mouse model of hepatocellular carcinoma.

Authors:  Ram C Shankaraiah; Elisa Callegari; Paola Guerriero; Alessandro Rimessi; Paolo Pinton; Laura Gramantieri; Enrico M Silini; Silvia Sabbioni; Massimo Negrini
Journal:  Oncogene       Date:  2019-08-13       Impact factor: 9.867

6.  Impact of Baseline Characteristics on the Overall Survival of HCC Patients Treated with Sorafenib: Ten Years of Experience.

Authors:  Giulia Rovesti; Giulia Orsi; Andrikou Kalliopi; Caterina Vivaldi; Giorgia Marisi; Luca Faloppi; Francesco Giuseppe Foschi; Nicola Silvestris; Irene Pecora; Giuseppe Aprile; Eleonora Molinaro; Laura Riggi; Paola Ulivi; Matteo Canale; Alessandro Cucchetti; Emiliano Tamburini; Giorgio Ercolani; Lorenzo Fornaro; Pietro Andreone; Patrizia Zavattari; Mario Scartozzi; Stefano Cascinu; Andrea Casadei-Gardini
Journal:  Gastrointest Tumors       Date:  2019-09-12

Review 7.  Hepatocellular carcinoma in non-alcoholic fatty liver disease-a review of an emerging challenge facing clinicians.

Authors:  Daniel Geh; Derek M Manas; Helen L Reeves
Journal:  Hepatobiliary Surg Nutr       Date:  2021-01       Impact factor: 8.265

8.  Early onset of hypertension and serum electrolyte changes as potential predictive factors of activity in advanced HCC patients treated with sorafenib: results from a retrospective analysis of the HCC-AVR group.

Authors:  Andrea Casadei Gardini; Emanuela Scarpi; Giorgia Marisi; Francesco Giuseppe Foschi; Gabriele Donati; Emanuela Giampalma; Luca Faloppi; Mario Scartozzi; Nicola Silvestris; Marcello Bisulli; Jody Corbelli; Andrea Gardini; Giuliano La Barba; Luigi Veneroni; Stefano Tamberi; Stefano Cascinu; Giovanni Luca Frassineti
Journal:  Oncotarget       Date:  2016-03-22

9.  Impact of Diabetes on Outcomes of Sorafenib Therapy for Hepatocellular Carcinoma.

Authors:  Giovan Giuseppe Di Costanzo; Raffaella Tortora; Filomena Morisco; Luigi Addario; Maria Guarino; Gabriella Cordone; Luigia Falco; Nicola Caporaso
Journal:  Target Oncol       Date:  2017-02       Impact factor: 4.864

Review 10.  Hepatocellular Carcinoma in Pakistan: National Trends and Global Perspective.

Authors:  Abu Bakar Hafeez Bhatti; Faisal Saud Dar; Anum Waheed; Kashif Shafique; Faisal Sultan; Najmul Hassan Shah
Journal:  Gastroenterol Res Pract       Date:  2016-02-03       Impact factor: 2.260

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