Literature DB >> 26166854

Synthesis, structure, and tuberculostatic activity of dimethyl benzoylcarbonohydrazonodithioates.

Katarzyna Gobis1, Henryk Foks1, Zofia Zwolska2, Ewa Augustynowicz-Kopeć2, Marek L Główka3, Andrzej Olczak3, Michał Sabisz4.   

Abstract

ABSTRACT: New dimethyl benzoylcarbonohydrazonodithioates were obtained by CS2 addition to arylcarboxylic acid hydrazides and methylation of the formed adduct. The new derivatives were tested for their activity against Mycobacterium tuberculosis. Some compounds exhibited high activity toward sensitive and resistant strains.

Entities:  

Keywords:  Benzohydrazides; Crystal structure; Hydrogen bonds; Structure–activity relationship; Tuberculostatic activity

Year:  2011        PMID： 26166854      PMCID： PMC4494766          DOI： 10.1007/s00706-011-0572-9

Source DB:  PubMed          Journal:  Monatsh Chem        ISSN： 0026-9247            Impact factor:   1.451


  11 in total

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9.  Tuberculosis research in the European union: past achievements and future challenges.

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10.  Synthesis and structure-antituberculosis activity relationship of 1H-indole-2,3-dione derivatives.

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  1 in total

1.  Synthesis, characterization, and tuberculostatic activity of novel 2-(4-nitrobenzoyl)hydrazinecarbodithioic acid derivatives.

Authors:  Katarzyna Gobis; Henryk Foks; Ewa Augustynowicz-Kopec; Agnieszka Napiorkowska; Malgorzata Szczesio; Andrzej Olczak; Marek L Glowka
Journal:  Monatsh Chem       Date:  2012-01-24       Impact factor: 1.451
  1 in total

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