Literature DB >> 26144217

[(18)F]-NHC-BF3 adducts as water stable radio-prosthetic groups for PET imaging.

Kantapat Chansaenpak1, Mengzhe Wang, Zhanhong Wu, Rehmat Zaman, Zibo Li, François P Gabbaï.   

Abstract

The radiofluorination of N-heterocyclic carbene (NHC) boron trifluoride adducts affords novel [(18)F]-positron emission tomography probes which resist hydrolytic fluoride release. The labelling protocol relies on an (18)F-(19)F isotopic exchange reaction promoted by the Lewis acid SnCl4. Modification of the NHC backbone with a maleimide functionality provides access to a model peptide conjugate which shows no evidence of defluorination when imaged in vivo.

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Year:  2015        PMID： 26144217      PMCID： PMC5457534          DOI： 10.1039/c5cc04545b

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  17 in total

1.  Novel matrix metalloproteinase inhibitor [18F]marimastat-aryltrifluoroborate as a probe for in vivo positron emission tomography imaging in cancer.

Authors:  Ulrich auf dem Keller; Caroline L Bellac; Ying Li; Yuanmei Lou; Philipp F Lange; Richard Ting; Curtis Harwig; Reinhild Kappelhoff; Shoukat Dedhar; Michael J Adam; Thomas J Ruth; François Bénard; David M Perrin; Christopher M Overall
Journal:  Cancer Res       Date:  2010-08-20       Impact factor: 12.701

Review 2.  Synthesis of 11C, 18F, 15O, and 13N radiolabels for positron emission tomography.

Authors:  Philip W Miller; Nicholas J Long; Ramon Vilar; Antony D Gee
Journal:  Angew Chem Int Ed Engl       Date:  2008       Impact factor: 15.336

3.  Rapid aqueous [18F]-labeling of a bodipy dye for positron emission tomography/fluorescence dual modality imaging.

Authors:  Zibo Li; Tzu-Pin Lin; Shuanglong Liu; Chiun-Wei Huang; Todd W Hudnall; François P Gabbaï; Peter S Conti
Journal:  Chem Commun (Camb)       Date:  2011-07-21       Impact factor: 6.222

4.  Dual mode fluorescent (18)F-PET tracers: efficient modular synthesis of rhodamine-[cRGD]2-[(18)F]-organotrifluoroborate, rapid, and high yielding one-step (18)F-labeling at high specific activity, and correlated in vivo PET imaging and ex vivo fluorescence.

Authors:  Zhibo Liu; Mark Alex Radtke; May Q Wong; Kuo-Shyan Lin; Donald T Yapp; David M Perrin
Journal:  Bioconjug Chem       Date:  2014-09-29       Impact factor: 4.774

5.  o-Boronato- and o-Trifluoroborato-Phosphonium Salts Supported by L-α-Amino Acid Side Chain.

Authors:  Julie Bernard; Raluca Malacea-Kabbara; Gonçalo S Clemente; Benjamin P Burke; Marie-Joëlle Eymin; Stephen J Archibald; Sylvain Jugé
Journal:  J Org Chem       Date:  2015-04-14       Impact factor: 4.354

6.  From minutes to years: predicting organotrifluoroborate solvolysis rates.

Authors:  Zhibo Liu; Daniel Chao; Ying Li; Richard Ting; Jihyoon Oh; David M Perrin
Journal:  Chemistry       Date:  2015-01-30       Impact factor: 5.236

7.  Stoichiometric leverage: rapid 18F-aryltrifluoroborate radiosynthesis at high specific activity for click conjugation.

Authors:  Zhibo Liu; Ying Li; Jerome Lozada; Paul Schaffer; Michael J Adam; Thomas J Ruth; David M Perrin
Journal:  Angew Chem Int Ed Engl       Date:  2013-01-11       Impact factor: 15.336

8.  Arylfluoroborates and alkylfluorosilicates as potential PET imaging agents: high-yielding aqueous biomolecular 18F-labeling.

Authors:  Richard Ting; Michael J Adam; Thomas J Ruth; David M Perrin
Journal:  J Am Chem Soc       Date:  2005-09-28       Impact factor: 15.419

9.  Organotrifluoroborate hydrolysis: boronic acid release mechanism and an acid-base paradox in cross-coupling.

Authors:  Alastair J J Lennox; Guy C Lloyd-Jones
Journal:  J Am Chem Soc       Date:  2012-04-19       Impact factor: 15.419

10.  Lewis acid-assisted isotopic 18F-19F exchange in BODIPY dyes: facile generation of positron emission tomography/fluorescence dual modality agents for tumor imaging.

Authors:  Shuanglong Liu; Tzu-Pin Lin; Dan Li; Lauren Leamer; Hong Shan; Zibo Li; François P Gabbaï; Peter S Conti
Journal:  Theranostics       Date:  2013-02-21       Impact factor: 11.556
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  4 in total

1.  Radiofluorination of a NHC-PF5 adduct: toward new probes for 18F PET imaging.

Authors:  Boris Vabre; Kantapat Chansaenpak; Mengzhe Wang; Hui Wang; Zibo Li; François P Gabbaï
Journal:  Chem Commun (Camb)       Date:  2017-07-21       Impact factor: 6.222

Review 2.  Chemistry for Positron Emission Tomography: Recent Advances in 11 C-, 18 F-, 13 N-, and 15 O-Labeling Reactions.

Authors:  Xiaoyun Deng; Jian Rong; Lu Wang; Neil Vasdev; Lei Zhang; Lee Josephson; Steven H Liang
Journal:  Angew Chem Int Ed Engl       Date:  2019-01-14       Impact factor: 15.336

3.  A Novel PET Probe for Brown Adipose Tissue Imaging in Rodents.

Authors:  Hui Wang; Mengzhe Wang; Kantapat Chansaenpak; Yang Liu; Hong Yuan; Jin Xie; Hang Yin; Rosa T Branca; Zibo Li; Zhanhong Wu
Journal:  Mol Imaging Biol       Date:  2020-06       Impact factor: 3.488

Review 4.  Radiolabelled Peptides for Positron Emission Tomography and Endoradiotherapy in Oncology.

Authors:  Christine Rangger; Roland Haubner
Journal:  Pharmaceuticals (Basel)       Date:  2020-01-30
  4 in total

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