Literature DB >> 25738371

A twin study of the trough plasma steady-state concentration of metformin.

Tore B Stage1, Per Damkier, Rasmus S Pedersen, Mette M H Christensen, Lene Christiansen, Kaare Christensen, Kim Brosen.   

Abstract

OBJECTIVE: The aim of this study was to determine the intrapair similarity in trough steady-state plasma concentrations of metformin in monozygotic and dizygotic twin pairs.
METHODS: We included 16 twin pairs (eight monozygotic and eight dizygotic twin pairs) for this study after contacting 524 twin pairs. They were dosed with metformin to steady state (1 g twice daily) for 6 days and on day 7, the trough concentration of metformin was determined 12 h after the last dose.
RESULTS: There was no strong intrapair similarity in trough steady-state plasma concentrations of metformin in either dizygotic or monozygotic twin pairs.
CONCLUSION: The trough steady-state plasma concentration of metformin does not appear to be tightly genetically regulated. The interpretation of this finding is limited by the small sample size.

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Year:  2015        PMID: 25738371     DOI: 10.1097/FPC.0000000000000133

Source DB:  PubMed          Journal:  Pharmacogenet Genomics        ISSN: 1744-6872            Impact factor:   2.089


  6 in total

1.  Endogenous glucose production increases in response to metformin treatment in the glycogen-depleted state in humans: a randomised trial.

Authors:  Mette Marie H Christensen; Kurt Højlund; Ole Hother-Nielsen; Tore B Stage; Per Damkier; Henning Beck-Nielsen; Kim Brøsen
Journal:  Diabetologia       Date:  2015-08-14       Impact factor: 10.122

2.  Steady-state pharmacokinetics of metformin is independent of the OCT1 genotype in healthy volunteers.

Authors:  Mette Marie Hougaard Christensen; Kurt Højlund; Ole Hother-Nielsen; Tore Bjerregaard Stage; Per Damkier; Henning Beck-Nielsen; Kim Brøsen
Journal:  Eur J Clin Pharmacol       Date:  2015-05-05       Impact factor: 2.953

Review 3.  Novel genetic and epigenetic factors of importance for inter-individual differences in drug disposition, response and toxicity.

Authors:  Volker M Lauschke; Yitian Zhou; Magnus Ingelman-Sundberg
Journal:  Pharmacol Ther       Date:  2019-01-22       Impact factor: 12.310

Review 4.  A Comprehensive Review of Drug-Drug Interactions with Metformin.

Authors:  Tore Bjerregaard Stage; Kim Brøsen; Mette Marie Hougaard Christensen
Journal:  Clin Pharmacokinet       Date:  2015-08       Impact factor: 6.447

5.  Low metformin dose and its therapeutic serum concentration in prediabetes.

Authors:  Edyta Sutkowska; Paulina Fortuna; Jerzy Wisniewski; Karolina Sutkowska; Pawel Hodurek; Andrzej Gamian; Bernadetta Kaluza
Journal:  Sci Rep       Date:  2021-06-03       Impact factor: 4.379

6.  Solute Carrier Transportome in Chemotherapy-Induced Adverse Drug Reactions.

Authors:  Jason T Anderson; Kevin M Huang; Maryam B Lustberg; Alex Sparreboom; Shuiying Hu
Journal:  Rev Physiol Biochem Pharmacol       Date:  2022       Impact factor: 7.500

  6 in total

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