Literature DB >> 25558307

New and emerging drugs and targets for type 2 diabetes: reviewing the evidence.

Brien Rex Miller1, Hanh Nguyen1, Charles Jia-Haur Hu1, Chihyi Lin1, Quang T Nguyen2.   

Abstract

BACKGROUND: Diabetes is a deadly and costly disease. The number of adults in the United States with newly diagnosed diabetes has nearly tripled from 1980 to 2011. At the current pace, 1 in 3 US adults will have diabetes in their lifetime. Currently, 14 classes of drugs are available to treat type 2 diabetes mellitus, but only 36% of patients with type 2 diabetes achieve glycemic control with the currently available therapies. Therefore, new treatment options are desperately needed. DISCUSSION: Despite the availability of many pharmacotherapies, in 2011 an estimated 3.1 million (14.9%) patients with type 2 diabetes still reported not taking medications to treat their diabetes. Patient compliance is a major obstacle facing practicing clinicians on a daily basis. New treatment options are desperately needed, but efficacy and tolerability are no longer the only criteria contributing to the success of a drug. Ease of administration, convenient dosing frequency, being weight control friendly, and having a low risk for hypoglycemia are important factors for the survival of a new drug in the US healthcare system. The present review is focused on important new drugs and drug classes in the pipeline, as well as on recently approved drugs, including sodium glucose cotransporter-2 inhibitors, glucagon-like peptide-1 agents, and new insulin therapies, as well as on the technologic improvements in the delivery and dosing frequency of some of the currently available drugs.
CONCLUSIONS: In the United States, diabetes can be expected to continue to wreak significant human and financial tolls. The associated complications will continue to climb if they are not controlled and stopped. New therapies for diabetes are clearly needed that will better address these unmet needs. The common threads among the emerging therapies are their convenience of administration and dosing frequency, which are important to the improvement of patient adherence.

Entities:  

Year:  2014        PMID: 25558307      PMCID: PMC4280522     

Source DB:  PubMed          Journal:  Am Health Drug Benefits        ISSN: 1942-2962


  43 in total

1.  Empagliflozin monotherapy in Japanese patients with type 2 diabetes mellitus: a randomized, 12-week, double-blind, placebo-controlled, phase II trial.

Authors:  Takashi Kadowaki; Masakazu Haneda; Nobuya Inagaki; Yasuo Terauchi; Atsushi Taniguchi; Kazuki Koiwai; Henning Rattunde; Hans J Woerle; Uli C Broedl
Journal:  Adv Ther       Date:  2014-06-24       Impact factor: 3.845

2.  The incidence and costs of hypoglycemia in type 2 diabetes.

Authors:  Brian J Quilliam; Jason C Simeone; A Burak Ozbay; Stephen J Kogut
Journal:  Am J Manag Care       Date:  2011-10       Impact factor: 2.229

3.  Ranolazine increases β-cell survival and improves glucose homeostasis in low-dose streptozotocin-induced diabetes in mice.

Authors:  Yun Ning; Wei Zhen; Zhuo Fu; Jenny Jiang; Dongmin Liu; Luiz Belardinelli; Arvinder K Dhalla
Journal:  J Pharmacol Exp Ther       Date:  2011-01-12       Impact factor: 4.030

4.  Efficacy and safety of empagliflozin, a sodium glucose cotransporter 2 (SGLT2) inhibitor, as add-on to metformin in type 2 diabetes with mild hyperglycaemia.

Authors:  J Rosenstock; L J Seman; A Jelaska; S Hantel; S Pinnetti; T Hach; H J Woerle
Journal:  Diabetes Obes Metab       Date:  2013-08-22       Impact factor: 6.577

5.  Dapagliflozin monotherapy in type 2 diabetic patients with inadequate glycemic control by diet and exercise: a randomized, double-blind, placebo-controlled, phase 3 trial.

Authors:  Ele Ferrannini; Silvia Jimenez Ramos; Afshin Salsali; Weihua Tang; James F List
Journal:  Diabetes Care       Date:  2010-06-21       Impact factor: 19.112

6.  The diabetes mellitus medication choice decision aid: a randomized trial.

Authors:  Rebecca J Mullan; Victor M Montori; Nilay D Shah; Teresa J H Christianson; Sandra C Bryant; Gordon H Guyatt; Lilisbeth I Perestelo-Perez; Robert J Stroebel; Barbara P Yawn; Victor Yapuncich; Maggie A Breslin; Laurie Pencille; Steven A Smith
Journal:  Arch Intern Med       Date:  2009-09-28

7.  Rationale, design, and baseline characteristics of the Canagliflozin Cardiovascular Assessment Study (CANVAS)--a randomized placebo-controlled trial.

Authors:  Bruce Neal; Vlado Perkovic; Dick de Zeeuw; Kenneth W Mahaffey; Greg Fulcher; Peter Stein; Mehul Desai; Wayne Shaw; Joel Jiang; Frank Vercruysse; Gary Meininger; David Matthews
Journal:  Am Heart J       Date:  2013-06-24       Impact factor: 4.749

Review 8.  Treatment of type 2 diabetes mellitus with agonists of the GLP-1 receptor or DPP-IV inhibitors.

Authors:  Jens Juul Holst
Journal:  Expert Opin Emerg Drugs       Date:  2004-05       Impact factor: 4.191

9.  Dapagliflozin versus glipizide as add-on therapy in patients with type 2 diabetes who have inadequate glycemic control with metformin: a randomized, 52-week, double-blind, active-controlled noninferiority trial.

Authors:  Michael A Nauck; Stefano Del Prato; Juris J Meier; Santiago Durán-García; Katja Rohwedder; Martina Elze; Shamik J Parikh
Journal:  Diabetes Care       Date:  2011-08-04       Impact factor: 19.112

Review 10.  Management of hyperglycemia in type 2 diabetes: a patient-centered approach: position statement of the American Diabetes Association (ADA) and the European Association for the Study of Diabetes (EASD).

Authors:  Silvio E Inzucchi; Richard M Bergenstal; John B Buse; Michaela Diamant; Ele Ferrannini; Michael Nauck; Anne L Peters; Apostolos Tsapas; Richard Wender; David R Matthews
Journal:  Diabetes Care       Date:  2012-04-19       Impact factor: 19.112

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  16 in total

1.  An Extended Minimal Physiologically Based Pharmacokinetic Model: Evaluation of Type II Diabetes Mellitus and Diabetic Nephropathy on Human IgG Pharmacokinetics in Rats.

Authors:  Gurkishan S Chadha; Marilyn E Morris
Journal:  AAPS J       Date:  2015-08-15       Impact factor: 4.009

Review 2.  New and emerging drugs and targets for type 2 diabetes: reviewing the evidence.

Authors:  Brien Rex Miller; Hanh Nguyen; Charles Jia-Haur Hu; Chihyi Lin; Quang T Nguyen
Journal:  Am Health Drug Benefits       Date:  2014-11

3.  Syntheses, in vitro, and in silico studies of rhodanine-based schiff bases as potential α-amylase inhibitors and radicals (DPPH and ABTS) scavengers.

Authors:  Samuel Attah Egu; Irfan Ali; Khalid Mohammed Khan; Sridevi Chigurupati; Urooj Qureshi; Uzma Salar; Muhammad Taha; Shatha Ghazi Felemban; Vijayan Venugopal; Zaheer Ul-Haq
Journal:  Mol Divers       Date:  2022-05-23       Impact factor: 2.943

Review 4.  Tracking the carbons supplying gluconeogenesis.

Authors:  Ankit M Shah; Fredric E Wondisford
Journal:  J Biol Chem       Date:  2020-08-13       Impact factor: 5.157

5.  Non-Persistence and Non-Adherence of Patients with Type 2 Diabetes Mellitus in Therapy with GLP-1 Receptor Agonists: A Retrospective Analysis.

Authors:  Thomas Wilke; Sabrina Mueller; Antje Groth; Bjoern Berg; Andreas Fuchs; Mirko Sikirica; John Logie; Alan Martin; Ulf Maywald
Journal:  Diabetes Ther       Date:  2015-12-22       Impact factor: 2.945

Review 6.  Cost-Effectiveness of Saxagliptin versus Acarbose as Second-Line Therapy in Type 2 Diabetes in China.

Authors:  Shuyan Gu; Yuhang Zeng; Demin Yu; Xiaoqian Hu; Hengjin Dong
Journal:  PLoS One       Date:  2016-11-22       Impact factor: 3.240

7.  Cost-Effectiveness of Dapagliflozin versus Acarbose as a Monotherapy in Type 2 Diabetes in China.

Authors:  Shuyan Gu; Yiming Mu; Suodi Zhai; Yuhang Zeng; Xuemei Zhen; Hengjin Dong
Journal:  PLoS One       Date:  2016-11-02       Impact factor: 3.240

8.  E4orf1: A protein for enhancing glucose uptake despite impaired proximal insulin signaling.

Authors:  Anuradha A Shastri; Vijay Hegde; Swetha Peddibhotla; Zahra Feizy; Nikhil V Dhurandhar
Journal:  PLoS One       Date:  2018-12-06       Impact factor: 3.240

Review 9.  Exenatide once-weekly injection for the treatment of type 2 diabetes in Chinese patients: current perspectives.

Authors:  Wuquan Deng; Sheng Qiu; Gangyi Yang; Bing Chen
Journal:  Ther Clin Risk Manag       Date:  2015-08-10       Impact factor: 2.423

10.  Treatment patterns in patients with type 2 diabetes mellitus treated with glucagon-like peptide-1 receptor agonists: Higher adherence and persistence with dulaglutide compared with once-weekly exenatide and liraglutide.

Authors:  Carlos Alatorre; Laura Fernández Landó; Maria Yu; Katelyn Brown; Leslie Montejano; Paul Juneau; Reema Mody; Ralph Swindle
Journal:  Diabetes Obes Metab       Date:  2017-03-16       Impact factor: 6.577

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