Literature DB >> 25526946

Subconjunctival sirolimus in the treatment of autoimmune non-necrotizing anterior scleritis: results of a phase I/II clinical trial.

Nirali Bhatt1, Monica Dalal1, William Tucker1, Dominic Obiyor1, Robert Nussenblatt1, H Nida Sen2.   

Abstract

PURPOSE: To investigate the safety, tolerability and efficacy of subconjunctival sirolimus injections as a treatment for active, autoimmune, non-necrotizing anterior scleritis.
DESIGN: Phase I/II, single-center, open-label, nonrandomized, prospective pilot study.
METHODS: Five participants with active, autoimmune, non-necrotizing anterior scleritis with scleral inflammatory grade of ≥1+ in at least 1 quadrant with a history of flares were enrolled. A baseline injection was given, with the primary outcome measure of at least a 2-step reduction or reduction to grade zero in the study eye by 8 weeks. Secondary outcomes included changes in visual acuity and intraocular pressure, ability to taper concomitant immunosuppressive regimen, and number of participants who experienced a disease flare requiring reinjection. Safety outcomes included the number and severity of systemic and ocular toxicities, and vision loss ≥15 ETDRS letters. The study included 6 visits over 4 months with an extension phase to 1 year for participants who met the primary outcome.
RESULTS: All participants (N = 5, 100%; 95% CI [0.60, 1.00]) met the primary outcome in the study eye by the week 8 visit. There was no significant change in mean visual acuity or intraocular pressure. Three out of 5 patients (60%) experienced flares requiring reinjection. No systemic toxicities were observed. Two participants (40%) experienced a localized sterile inflammatory reaction at the site of the injection, which resolved without complication.
CONCLUSIONS: Subconjunctival sirolimus leads to a short-term reduction in scleral inflammation, though relapses requiring reinjection do occur. There were no serious adverse events, though a local sterile conjunctival inflammatory reaction was observed. Published by Elsevier Inc.

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Year:  2014        PMID: 25526946      PMCID: PMC4329278          DOI: 10.1016/j.ajo.2014.12.009

Source DB:  PubMed          Journal:  Am J Ophthalmol        ISSN: 0002-9394            Impact factor:   5.258


  24 in total

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Journal:  Am J Ophthalmol       Date:  2000-10       Impact factor: 5.258

2.  Subconjunctival corticosteroid injection for the treatment of non-necrotising anterior scleritis.

Authors:  H N Sen; R Ursea; R B Nussenblatt; R R Buggage
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9.  Comparison of conjunctival and corneal surface areas in rabbit and human.

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2.  Ocular Manifestations of Rheumatoid Arthritis: Implications of Recent Clinical Trials.

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Review 4.  Rheumatoid Arthritis Associated Episcleritis and Scleritis: An Update on Treatment Perspectives.

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