Literature DB >> 25482145

Carfilzomib, lenalidomide, and dexamethasone for relapsed multiple myeloma.

A Keith Stewart1, S Vincent Rajkumar, Meletios A Dimopoulos, Tamás Masszi, Ivan Špička, Albert Oriol, Roman Hájek, Laura Rosiñol, David S Siegel, Georgi G Mihaylov, Vesselina Goranova-Marinova, Péter Rajnics, Aleksandr Suvorov, Ruben Niesvizky, Andrzej J Jakubowiak, Jesus F San-Miguel, Heinz Ludwig, Michael Wang, Vladimír Maisnar, Jiri Minarik, William I Bensinger, Maria-Victoria Mateos, Dina Ben-Yehuda, Vishal Kukreti, Naseem Zojwalla, Margaret E Tonda, Xinqun Yang, Biao Xing, Philippe Moreau, Antonio Palumbo.   

Abstract

BACKGROUND: Lenalidomide plus dexamethasone is a reference treatment for relapsed multiple myeloma. The combination of the proteasome inhibitor carfilzomib with lenalidomide and dexamethasone has shown efficacy in a phase 1 and 2 study in relapsed multiple myeloma.
METHODS: We randomly assigned 792 patients with relapsed multiple myeloma to carfilzomib with lenalidomide and dexamethasone (carfilzomib group) or lenalidomide and dexamethasone alone (control group). The primary end point was progression-free survival.
RESULTS: Progression-free survival was significantly improved with carfilzomib (median, 26.3 months, vs. 17.6 months in the control group; hazard ratio for progression or death, 0.69; 95% confidence interval [CI], 0.57 to 0.83; P=0.0001). The median overall survival was not reached in either group at the interim analysis. The Kaplan-Meier 24-month overall survival rates were 73.3% and 65.0% in the carfilzomib and control groups, respectively (hazard ratio for death, 0.79; 95% CI, 0.63 to 0.99; P=0.04). The rates of overall response (partial response or better) were 87.1% and 66.7% in the carfilzomib and control groups, respectively (P<0.001; 31.8% and 9.3% of patients in the respective groups had a complete response or better; 14.1% and 4.3% had a stringent complete response). Adverse events of grade 3 or higher were reported in 83.7% and 80.7% of patients in the carfilzomib and control groups, respectively; 15.3% and 17.7% of patients discontinued treatment owing to adverse events. Patients in the carfilzomib group reported superior health-related quality of life.
CONCLUSIONS: In patients with relapsed multiple myeloma, the addition of carfilzomib to lenalidomide and dexamethasone resulted in significantly improved progression-free survival at the interim analysis and had a favorable risk-benefit profile. (Funded by Onyx Pharmaceuticals; ClinicalTrials.gov number, NCT01080391.).

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Year:  2014        PMID: 25482145     DOI: 10.1056/NEJMoa1411321

Source DB:  PubMed          Journal:  N Engl J Med        ISSN: 0028-4793            Impact factor:   91.245


  415 in total

1.  Elotuzumab in combination with lenalidomide and dexamethasone in patients with relapsed multiple myeloma: final phase 2 results from the randomised, open-label, phase 1b-2 dose-escalation study.

Authors:  Paul G Richardson; Sundar Jagannath; Philippe Moreau; Andrzej J Jakubowiak; Marc S Raab; Thierry Facon; Ravi Vij; Darrell White; Donna E Reece; Lotfi Benboubker; Jeffrey Zonder; L Claire Tsao; Kenneth C Anderson; Eric Bleickardt; Anil K Singhal; Sagar Lonial
Journal:  Lancet Haematol       Date:  2015-11-16       Impact factor: 18.959

2.  Carfilzomib significantly improves the progression-free survival of high-risk patients in multiple myeloma.

Authors:  Hervé Avet-Loiseau; Rafael Fonseca; David Siegel; Meletios A Dimopoulos; Ivan Špička; Tamás Masszi; Roman Hájek; Laura Rosiñol; Vesselina Goranova-Marinova; Georgi Mihaylov; Vladimír Maisnar; Maria-Victoria Mateos; Michael Wang; Ruben Niesvizky; Albert Oriol; Andrzej Jakubowiak; Jiri Minarik; Antonio Palumbo; William Bensinger; Vishal Kukreti; Dina Ben-Yehuda; A Keith Stewart; Mihaela Obreja; Philippe Moreau
Journal:  Blood       Date:  2016-07-20       Impact factor: 22.113

3.  p53-related protein kinase confers poor prognosis and represents a novel therapeutic target in multiple myeloma.

Authors:  Teru Hideshima; Francesca Cottini; Yoshihisa Nozawa; Hyuk-Soo Seo; Hiroto Ohguchi; Mehmet K Samur; Diana Cirstea; Naoya Mimura; Yoshikazu Iwasawa; Paul G Richardson; Nikhil C Munshi; Dharminder Chauhan; Walter Massefski; Teruhiro Utsugi; Sirano Dhe-Paganon; Kenneth C Anderson
Journal:  Blood       Date:  2017-01-12       Impact factor: 22.113

4.  Polymer micelle formulations of proteasome inhibitor carfilzomib for improved metabolic stability and anticancer efficacy in human multiple myeloma and lung cancer cell lines.

Authors:  Lin Ao; Derek Reichel; Di Hu; Hyunyoung Jeong; Kyung Bo Kim; Younsoo Bae; Wooin Lee
Journal:  J Pharmacol Exp Ther       Date:  2015-08-26       Impact factor: 4.030

5.  Critical Appraisal of Published Indirect Comparisons and Network Meta-Analyses of Competing Interventions for Multiple Myeloma.

Authors:  Shannon Cope; Kabirraaj Toor; Evan Popoff; Rafael Fonseca; Ola Landgren; María-Victoria Mateos; Katja Weisel; Jeroen Paul Jansen
Journal:  Value Health       Date:  2020-04-06       Impact factor: 5.725

6.  EphA3 targeting reduces in vitro adhesion and invasion and in vivo growth and angiogenesis of multiple myeloma cells.

Authors:  Francesco La Rocca; Irma Airoldi; Emma Di Carlo; Pina Marotta; Geppino Falco; Vittorio Simeon; Ilaria Laurenzana; Stefania Trino; Luciana De Luca; Katia Todoerti; Oreste Villani; Martin Lackmann; Fiorella D'Auria; Francesco Frassoni; Antonino Neri; Luigi Del Vecchio; Pellegrino Musto; Daniela Cilloni; Antonella Caivano
Journal:  Cell Oncol (Dordr)       Date:  2017-07-18       Impact factor: 6.730

7.  Pomalidomide-dexamethasone in refractory multiple myeloma: long-term follow-up of a multi-cohort phase II clinical trial.

Authors:  S Ailawadhi; J R Mikhael; B R LaPlant; K M Laumann; S Kumar; V Roy; D Dingli; P L Bergsagel; F K Buadi; S V Rajkumar; R Fonseca; M A Gertz; P Kapoor; T Sher; S R Hayman; A K Stewart; A Dispenzieri; R A Kyle; W I Gonsalves; C B Reeder; Y Lin; R S Go; N Leung; T Kourelis; J A Lust; S J Russell; A A Chanan-Khan; M Q Lacy
Journal:  Leukemia       Date:  2017-09-01       Impact factor: 11.528

8.  Carfilzomib, pomalidomide, and dexamethasone for relapsed or refractory myeloma.

Authors:  Jatin J Shah; Edward A Stadtmauer; Rafat Abonour; Adam D Cohen; William I Bensinger; Cristina Gasparetto; Jonathan L Kaufman; Suzanne Lentzsch; Dan T Vogl; Christina L Gomes; Natalia Pascucci; David D Smith; Robert Z Orlowski; Brian G M Durie
Journal:  Blood       Date:  2015-09-17       Impact factor: 22.113

9.  Kyprolis (Carfilzomib) Received New Indications as Combination Therapy for Use in Relapsed and/or Refractory Multiple Myeloma.

Authors:  Lisa A Raedler
Journal:  Am Health Drug Benefits       Date:  2016-03

Review 10.  Novel Treatments for Multiple Myeloma: What Role Do They Have in Older Adults?

Authors:  Hira S Mian; Tanya M Wildes
Journal:  Drugs Aging       Date:  2018-04       Impact factor: 3.923

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