Literature DB >> 25379166

Late-stage [18F]Fluorination: New Solutions to Old Problems.

Allen F Brooks1, Joseph J Topczewski2, Naoko Ichiishi2, Melanie S Sanford2, Peter J H Scott3.   

Abstract

The last 2-3 years have seen numerous relationships develop between organometallic chemists, fluorine chemists and PET Centers around the world. These collaborations have led to the development of many new strategies for the late-stage introduction of fluorine-18 into complex bioactive molecules. In this perspective we highlight recent developments and key milestones since 2011.

Entities:  

Year:  2014        PMID： 25379166      PMCID： PMC4217215          DOI： 10.1039/C4SC02099E

Source DB:  PubMed          Journal:  Chem Sci        ISSN： 2041-6520            Impact factor:   9.825


  41 in total

Review 1.  PET and the role of in vivo molecular imaging in personalized medicine.

Authors:  Richard Pither
Journal:  Expert Rev Mol Diagn       Date:  2003-11       Impact factor: 5.225

2.  FDG PET reimbursement.

Authors:  Jim Bietendorf
Journal:  J Nucl Med Technol       Date:  2004-03

Review 3.  Positron emission tomography molecular imaging for drug development.

Authors:  Paul M Matthews; Eugenii A Rabiner; Jan Passchier; Roger N Gunn
Journal:  Br J Clin Pharmacol       Date:  2012-02       Impact factor: 4.335

Review 4.  Synthesis of 11C, 18F, 15O, and 13N radiolabels for positron emission tomography.

Authors:  Philip W Miller; Nicholas J Long; Ramon Vilar; Antony D Gee
Journal:  Angew Chem Int Ed Engl       Date:  2008       Impact factor: 15.336

5.  Rapid and Efficient Radiosyntheses of Meta-substituted [F]Fluoroarenes from [F]Fluoride Ion and Diaryliodonium Tosylates within a Microreactor.

Authors:  Joong-Hyun Chun; Shuiyu Lu; Victor W Pike
Journal:  European J Org Chem       Date:  2011-08

6.  Synthesis, 18F-radiolabeling, and in vivo biodistribution studies of N-fluorohydroxybutyl isatin sulfonamides using positron emission tomography.

Authors:  Panupun Limpachayaporn; Stefan Wagner; Klaus Kopka; Sven Hermann; Michael Schäfers; Günter Haufe
Journal:  J Med Chem       Date:  2013-05-29       Impact factor: 7.446

7.  Cu(I)-mediated (18)F-trifluoromethylation of arenes: rapid synthesis of (18)F-labeled trifluoromethyl arenes.

Authors:  T Rühl; W Rafique; V T Lien; P J Riss
Journal:  Chem Commun (Camb)       Date:  2014-04-28       Impact factor: 6.222

8.  Synthesis and imaging validation of [¹⁸F]MDL100907 enabled by Ni-mediated fluorination.

Authors:  Hong Ren; Hsiao-Ying Wey; Martin Strebl; Ramesh Neelamegam; Tobias Ritter; Jacob M Hooker
Journal:  ACS Chem Neurosci       Date:  2014-06-03       Impact factor: 4.418

Review 9.  Regulatory Requirements for PET Drug Production.

Authors:  Sally W Schwarz; David Dick; Henry F VanBrocklin; John M Hoffman
Journal:  J Nucl Med       Date:  2014-06-09       Impact factor: 10.057

10.  A general copper-mediated nucleophilic 18F fluorination of arenes.

Authors:  Matthew Tredwell; Sean M Preshlock; Nicholas J Taylor; Stefan Gruber; Mickael Huiban; Jan Passchier; Joël Mercier; Christophe Génicot; Véronique Gouverneur
Journal:  Angew Chem Int Ed Engl       Date:  2014-06-10       Impact factor: 15.336
View more
  74 in total

Review 1.  Fluorine-18 patents (2009-2015). Part 1: novel radiotracers.

Authors:  Allen F Brooks; Lindsey R Drake; Megan N Stewart; Brian P Cary; Isaac M Jackson; Dale Mallette; Andrew V Mossine; Peter J H Scott
Journal:  Pharm Pat Anal       Date:  2015-12-16

2.  Evaluation of Enzyme Substrate Radiotracers as PET/MRS Hybrid Imaging Agents.

Authors:  Allen F Brooks; Lindsey R Drake; Xia Shao; Austin Zhao; Peter J H Scott; Michael R Kilbourn
Journal:  ACS Med Chem Lett       Date:  2018-10-03       Impact factor: 4.345

3.  Synthesis of (18) F-Difluoromethylarenes from Aryl (Pseudo) Halides.

Authors:  Hang Shi; Augustin Braun; Lu Wang; Steven H Liang; Neil Vasdev; Tobias Ritter
Journal:  Angew Chem Int Ed Engl       Date:  2016-08-05       Impact factor: 15.336

4.  One-pot synthesis of high molar activity 6-[18F]fluoro-l-DOPA by Cu-mediated fluorination of a BPin precursor.

Authors:  Andrew V Mossine; Sean S Tanzey; Allen F Brooks; Katarina J Makaravage; Naoko Ichiishi; Jason M Miller; Bradford D Henderson; Marc B Skaddan; Melanie S Sanford; Peter J H Scott
Journal:  Org Biomol Chem       Date:  2019-09-19       Impact factor: 3.876

5.  (Radio)fluoroclick Reaction Enabled by a Hydrogen-Bonding Cluster.

Authors:  Xiaojun Zeng; Junling Li; Chin K Ng; Gerald B Hammond; Bo Xu
Journal:  Angew Chem Int Ed Engl       Date:  2018-02-13       Impact factor: 15.336

Review 6.  Considerations in the Development of Reversibly Binding PET Radioligands for Brain Imaging.

Authors:  Victor W Pike
Journal:  Curr Med Chem       Date:  2016       Impact factor: 4.530

Review 7.  Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.

Authors:  Andrew V Mossine; Stephen Thompson; Allen F Brooks; Alexandra R Sowa; Jason M Miller; Peter Jh Scott
Journal:  Pharm Pat Anal       Date:  2016-09

8.  Copper-Mediated Aminoquinoline-Directed Radiofluorination of Aromatic C-H Bonds with K18 F.

Authors:  So Jeong Lee; Katarina J Makaravage; Allen F Brooks; Peter J H Scott; Melanie S Sanford
Journal:  Angew Chem Int Ed Engl       Date:  2019-01-18       Impact factor: 15.336

9.  Difluorocarbene-Derived Trifluoromethylthiolation and [(18)F]Trifluoromethylthiolation of Aliphatic Electrophiles.

Authors:  Jian Zheng; Lu Wang; Jin-Hong Lin; Ji-Chang Xiao; Steven H Liang
Journal:  Angew Chem Int Ed Engl       Date:  2015-09-21       Impact factor: 15.336

10.  Facile room temperature synthesis of fluorine-18 labeled fluoronicotinic acid-2,3,5,6-tetrafluorophenyl ester without azeotropic drying of fluorine-18.

Authors:  Falguni Basuli; Xiang Zhang; Elaine M Jagoda; Peter L Choyke; Rolf E Swenson
Journal:  Nucl Med Biol       Date:  2016-08-30       Impact factor: 2.408
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.