Literature DB >> 25343227

Translating pharmacological findings from hypothyroid rodents to euthyroid humans: is there a functional role of endogenous 3,5-T2?

Maik Pietzner1, Ina Lehmphul, Nele Friedrich, Claudia Schurmann, Till Ittermann, Marcus Dörr, Matthias Nauck, René Laqua, Uwe Völker, Georg Brabant, Henry Völzke, Josef Köhrle, Georg Homuth, Henri Wallaschofski.   

Abstract

BACKGROUND: During the last two decades, it has become obvious that 3,5-diiodothyronine (3,5-T2), a well-known endogenous metabolite of the thyroid hormones thyroxine (T4) or triiodothyronine (T3), not only represents a simple degradation intermediate of the former but also exhibits specific metabolic activities. Administration of 3,5-T2 to hypothyroid rodents rapidly stimulated their basal metabolic rate, prevented high-fat diet-induced obesity as well as steatosis, and increased oxidation of long-chain fatty acids.
OBJECTIVE: The aim of the present study was to analyze associations between circulating 3,5-T2 in human serum and different epidemiological parameters, including age, sex, or smoking, as well as measures of anthropometry, glucose, and lipid metabolism.
METHODS: 3,5-T2 concentrations were measured by a recently developed immunoassay in sera of 761 euthyroid participants of the population-based Study of Health in Pomerania. Subsequently, analysis of variance and multivariate linear regression analysis were performed.
RESULTS: Serum 3,5-T2 concentrations exhibited a right-skewed distribution, resulting in a median serum concentration of 0.24 nM (1st quartile: 0.20 nM; 3rd quartile: 0.37 nM). Significant associations between 3,5-T2 and serum fasting glucose, thyrotropin (TSH), as well as leptin concentrations were detected (p<0.05). Interestingly, the association to leptin concentrations seemed to be mediated by TSH. Age, sex, smoking, and blood lipid profile parameters did not show significant associations with circulating 3,5-T2.
CONCLUSION: Our findings from a healthy euthyroid population may point toward a physiological link between circulating 3,5-T2 and glucose metabolism.

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Year:  2014        PMID: 25343227      PMCID: PMC4322092          DOI: 10.1089/thy.2014.0262

Source DB:  PubMed          Journal:  Thyroid        ISSN: 1050-7256            Impact factor:   6.568


  49 in total

1.  3,5-diiodo-L-thyronine increases resting metabolic rate and reduces body weight without undesirable side effects.

Authors:  A Antonelli; P Fallahi; S M Ferrari; A Di Domenicantonio; M Moreno; A Lanni; F Goglia
Journal:  J Biol Regul Homeost Agents       Date:  2011 Oct-Dec       Impact factor: 1.711

2.  Cohort profile: the study of health in Pomerania.

Authors:  Henry Völzke; Dietrich Alte; Carsten Oliver Schmidt; Dörte Radke; Roberto Lorbeer; Nele Friedrich; Nicole Aumann; Katharina Lau; Michael Piontek; Gabriele Born; Christoph Havemann; Till Ittermann; Sabine Schipf; Robin Haring; Sebastian E Baumeister; Henri Wallaschofski; Matthias Nauck; Stephanie Frick; Andreas Arnold; Michael Jünger; Julia Mayerle; Matthias Kraft; Markus M Lerch; Marcus Dörr; Thorsten Reffelmann; Klaus Empen; Stephan B Felix; Anne Obst; Beate Koch; Sven Gläser; Ralf Ewert; Ingo Fietze; Thomas Penzel; Martina Dören; Wolfgang Rathmann; Johannes Haerting; Mario Hannemann; Jürgen Röpcke; Ulf Schminke; Clemens Jürgens; Frank Tost; Rainer Rettig; Jan A Kors; Saskia Ungerer; Katrin Hegenscheid; Jens-Peter Kühn; Julia Kühn; Norbert Hosten; Ralf Puls; Jörg Henke; Oliver Gloger; Alexander Teumer; Georg Homuth; Uwe Völker; Christian Schwahn; Birte Holtfreter; Ines Polzer; Thomas Kohlmann; Hans J Grabe; Dieter Rosskopf; Heyo K Kroemer; Thomas Kocher; Reiner Biffar; Ulrich John; Wolfgang Hoffmann
Journal:  Int J Epidemiol       Date:  2010-02-18       Impact factor: 7.196

3.  3,5-Diiodo-L-thyronine prevents high-fat-diet-induced insulin resistance in rat skeletal muscle through metabolic and structural adaptations.

Authors:  Maria Moreno; Elena Silvestri; Rita De Matteis; Pieter de Lange; Assunta Lombardi; Daniela Glinni; Rosalba Senese; Federica Cioffi; Anna Maria Salzano; Andrea Scaloni; Antonia Lanni; Fernando Goglia
Journal:  FASEB J       Date:  2011-06-13       Impact factor: 5.191

4.  3,5-diiodo-L-thyronine regulates glucose-6-phosphate dehydrogenase activity in the rat.

Authors:  A Lombardi; L Beneduce; M Moreno; S Diano; V Colantuoni; M V Ursini; A Lanni; F Goglia
Journal:  Endocrinology       Date:  2000-05       Impact factor: 4.736

5.  3,5-diiodo-L-thyronine powerfully reduces adiposity in rats by increasing the burning of fats.

Authors:  Antonia Lanni; Maria Moreno; Assunta Lombardi; Pieter de Lange; Elena Silvestri; Maurizio Ragni; Paola Farina; Gabriella Chieffi Baccari; Pupah Fallahi; Alessandro Antonelli; Fernando Goglia
Journal:  FASEB J       Date:  2005-07-12       Impact factor: 5.191

6.  3,5-Diiodo-l-thyronine ameliorates diabetic nephropathy in streptozotocin-induced diabetic rats.

Authors:  Guoguo Shang; Pan Gao; Zhonghua Zhao; Qi Chen; Tao Jiang; Nong Zhang; Hui Li
Journal:  Biochim Biophys Acta       Date:  2013-02-08

7.  Serum concentrations of 3, 3'-diiodothyronine, 3', 5'-diiodothyronine, and 3, 5-diiodothyronine in altered thyroid states.

Authors:  M Nishikawa; M Inada; K Naito; H Ishii; K Tanaka; Y Mashio; H Imura
Journal:  Endocrinol Jpn       Date:  1983-04

8.  3,5-T2 is an alternative ligand for the thyroid hormone receptor β1.

Authors:  A Mendoza; P Navarrete-Ramírez; G Hernández-Puga; P Villalobos; G Holzer; J P Renaud; V Laudet; A Orozco
Journal:  Endocrinology       Date:  2013-06-04       Impact factor: 4.736

Review 9.  Thyroid hormone regulation of metabolism.

Authors:  Rashmi Mullur; Yan-Yun Liu; Gregory A Brent
Journal:  Physiol Rev       Date:  2014-04       Impact factor: 37.312

10.  A radioimmunoassay of serum 3,5-diiodothyronine.

Authors:  C Kirkegaard; J Faber; K Siersbaek-Nielsen; T Friis
Journal:  Acta Endocrinol (Copenh)       Date:  1981-06
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  14 in total

1.  Nonthyroidal Illness Syndrome in Cardiac Illness Involves Elevated Concentrations of 3,5-Diiodothyronine and Correlates with Atrial Remodeling.

Authors:  Johannes W Dietrich; Patrick Müller; Fabian Schiedat; Markus Schlömicher; Justus Strauch; Apostolos Chatzitomaris; Harald H Klein; Andreas Mügge; Josef Köhrle; Eddy Rijntjes; Ina Lehmphul
Journal:  Eur Thyroid J       Date:  2015-05-23

2.  Structural insights into thyroid hormone transport mechanisms of the L-type amino acid transporter 2.

Authors:  Katrin M Hinz; Katja Meyer; Anita Kinne; Ralf Schülein; Josef Köhrle; Gerd Krause
Journal:  Mol Endocrinol       Date:  2015-05-06

3.  High levels of thyroid-stimulating hormone are associated with aortic wall thickness in the general population.

Authors:  Till Ittermann; Roberto Lorbeer; Marcus Dörr; Tobias Schneider; Alexander Quadrat; Lydia Heßelbarth; Michael Wenzel; Ina Lehmphul; Josef Köhrle; Birger Mensel; Henry Völzke
Journal:  Eur Radiol       Date:  2016-03-14       Impact factor: 5.315

4.  Involvement of the L-Type Amino Acid Transporter Lat2 in the Transport of 3,3'-Diiodothyronine across the Plasma Membrane.

Authors:  Anita Kinne; Melanie Wittner; Eva K Wirth; Katrin M Hinz; Ralf Schülein; Josef Köhrle; Gerd Krause
Journal:  Eur Thyroid J       Date:  2015-05-28

5.  Urine Metabolomics by (1)H-NMR Spectroscopy Indicates Associations between Serum 3,5-T2 Concentrations and Intermediary Metabolism in Euthyroid Humans.

Authors:  Maik Pietzner; Georg Homuth; Kathrin Budde; Ina Lehmphul; Uwe Völker; Henry Völzke; Matthias Nauck; Josef Köhrle; Nele Friedrich
Journal:  Eur Thyroid J       Date:  2015-05-28

6.  Serum Thyrotropin Concentrations Are Not Associated with the Ankle-Brachial Index: Results from Three Population-Based Studies.

Authors:  Till Ittermann; Roberto Lorbeer; Daniel Tiller; Ina Lehmphul; Alexander Kluttig; Stephan B Felix; Karl Werdan; Karin Halina Greiser; Josef Köhrle; Henry Völzke; Marcus Dörr
Journal:  Eur Thyroid J       Date:  2015-05-27

Review 7.  3,5-Diiodothyronine: A Novel Thyroid Hormone Metabolite and Potent Modulator of Energy Metabolism.

Authors:  Rosalba Senese; Pieter de Lange; Giuseppe Petito; Maria Moreno; Fernando Goglia; Antonia Lanni
Journal:  Front Endocrinol (Lausanne)       Date:  2018-07-25       Impact factor: 5.555

8.  3,5-Diiodo-L-Thyronine Exerts Metabolically Favorable Effects on Visceral Adipose Tissue of Rats Receiving a High-Fat Diet.

Authors:  Elena Silvestri; Rosalba Senese; Federica Cioffi; Rita De Matteis; Davide Lattanzi; Assunta Lombardi; Antonia Giacco; Anna Maria Salzano; Andrea Scaloni; Michele Ceccarelli; Maria Moreno; Fernando Goglia; Antonia Lanni; Pieter de Lange
Journal:  Nutrients       Date:  2019-01-27       Impact factor: 5.717

9.  Assay of Endogenous 3,5-diiodo-L-thyronine (3,5-T2) and 3,3'-diiodo-L-thyronine (3,3'-T2) in Human Serum: A Feasibility Study.

Authors:  Leonardo Lorenzini; Nhat Minh Nguyen; Ginevra Sacripanti; Enrico Serni; Marco Borsò; Federica Saponaro; Elena Cecchi; Tommaso Simoncini; Sandra Ghelardoni; Riccardo Zucchi; Alessandro Saba
Journal:  Front Endocrinol (Lausanne)       Date:  2019-02-19       Impact factor: 5.555

Review 10.  Genomic and Non-Genomic Mechanisms of Action of Thyroid Hormones and Their Catabolite 3,5-Diiodo-L-Thyronine in Mammals.

Authors:  Marco Giammanco; Carlo Maria Di Liegro; Gabriella Schiera; Italia Di Liegro
Journal:  Int J Mol Sci       Date:  2020-06-10       Impact factor: 5.923

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