Literature DB >> 24934348

Boronic acid-based enzyme inhibitors: a review of recent progress.

H Fu, H Fang, Jie Sun, H Wang, A Liu, J Sun, Z Wu1.   

Abstract

Since Bortezomib was approved by US FDA as the first drug to treat multiple myeloma, various boronic acid compounds have been developed as enzyme inhibitors. This paper reviewed the progress of boronic acid-based inhibitors against enzymes including proteasome, serine protease, HDACs and other enzymes in the past decade.

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Year:  2014        PMID： 24934348     DOI： 10.2174/0929867321666140601200803

Source DB:  PubMed          Journal:  Curr Med Chem        ISSN： 0929-8673            Impact factor:   4.530


  12 in total

1.  A Comparison of the Structure and Bonding in the Aliphatic Boronic R-B(OH)2 and Borinic R-BH(OH) acids (R=H; NH2, OH, and F): A Computational Investigation.

Authors:  Niny Z Rao; Joseph D Larkin; Charles W Bock
Journal:  Struct Chem       Date:  2015-12-30       Impact factor: 1.887

Review 2.  Amino Acid Based Antimicrobial Agents - Synthesis and Properties.

Authors:  Michał G Nowak; Andrzej S Skwarecki; Maria J Milewska
Journal:  ChemMedChem       Date:  2021-10-01       Impact factor: 3.540

Review 3.  β-Lactamases and β-Lactamase Inhibitors in the 21st Century.

Authors:  Catherine L Tooke; Philip Hinchliffe; Eilis C Bragginton; Charlotte K Colenso; Viivi H A Hirvonen; Yuiko Takebayashi; James Spencer
Journal:  J Mol Biol       Date:  2019-04-05       Impact factor: 5.469

Review 4.  Enzyme Inhibitors: The Best Strategy to Tackle Superbug NDM-1 and Its Variants.

Authors:  Xiaoting Li; Dongmei Zhao; Weina Li; Jichao Sun; Xiuying Zhang
Journal:  Int J Mol Sci       Date:  2021-12-24       Impact factor: 5.923

Review 5.  Merging the Versatile Functionalities of Boronic Acid with Peptides.

Authors:  Yahong Tan; Junjie Wu; Lulu Song; Mengmeng Zhang; Christopher John Hipolito; Changsheng Wu; Siyuan Wang; Youming Zhang; Yizhen Yin
Journal:  Int J Mol Sci       Date:  2021-11-30       Impact factor: 5.923

Review 6.  Recent advances in activity-based probes (ABPs) and affinity-based probes (AfBPs) for profiling of enzymes.

Authors:  Haixiao Fang; Bo Peng; Sing Yee Ong; Qiong Wu; Lin Li; Shao Q Yao
Journal:  Chem Sci       Date:  2021-05-18       Impact factor: 9.825

7.  Discovering simple phenylboronic acid and benzoxaborole derivatives for experimental oncology - phase cycle-specific inducers of apoptosis in A2780 ovarian cancer cells.

Authors:  Mateusz Psurski; Agnieszka Łupicka-Słowik; Agnieszka Adamczyk-Woźniak; Joanna Wietrzyk; Andrzej Sporzyński
Journal:  Invest New Drugs       Date:  2018-05-19       Impact factor: 3.850

8.  The Role of Electron Transfer in the Fragmentation of Phenyl and Cyclohexyl Boronic Acids.

Authors:  Ana Isabel Lozano; Beatriz Pamplona; Tymon Kilich; Marta Łabuda; Mónica Mendes; João Pereira-da-Silva; Gustavo García; Pedro M P Gois; Filipe Ferreira da Silva; Paulo Limão-Vieira
Journal:  Int J Mol Sci       Date:  2019-11-08       Impact factor: 5.923

Review 9.  Emerging Strategies to Combat β-Lactamase Producing ESKAPE Pathogens.

Authors:  Corneliu Ovidiu Vrancianu; Irina Gheorghe; Elena-Georgiana Dobre; Ilda Czobor Barbu; Roxana Elena Cristian; Marcela Popa; Sang Hee Lee; Carmen Limban; Ilinca Margareta Vlad; Mariana Carmen Chifiriuc
Journal:  Int J Mol Sci       Date:  2020-11-12       Impact factor: 6.208

10.  Boronic Acid-Mediated Activity Control of Split 10-23 DNAzymes.

Authors:  Mégane Debiais; Amandine Lelievre; Jean-Jacques Vasseur; Sabine Müller; Michael Smietana
Journal:  Chemistry       Date:  2020-12-15       Impact factor: 5.020
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