Literature DB >> 24332623

Synthesis of a novel series of artemisinin dimers with potent anticancer activity involving Sonogashira cross-coupling reaction.

Pori Buragohain1, Bishwajit Saikia1, Naresh Surineni1, Nabin C Barua1, Ajit K Saxena2, Nitasha Suri2.   

Abstract

A series of C-10 acetal artemisinin dimers were synthesized using Sonogashira cross-coupling reaction. All these novel semisynthetic artemisinin dimers exhibited excellent growth inhibitory activity against Lung A-549 human cancer cell line.
Copyright © 2013 Elsevier Ltd. All rights reserved.

Entities:  

Keywords:  Anticancer; Artemisinin; Artemisinin dimer; Dihydroartemisinin; Sonogashira cross-coupling

Mesh：

Substances：

Year:  2013        PMID： 24332623     DOI： 10.1016/j.bmcl.2013.11.032

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  7 in total

1.  Stereoselective chlorothiolation of artemisinin-derived C-10 oxa terminal alkynes.

Authors:  Naresh Surineni; Pori Buragohain; Nabin C Barua
Journal:  Mol Divers       Date:  2015-06-19       Impact factor: 2.943

2.  Worldwide Research Trends on Artemisinin: A Bibliometric Analysis From 2000 to 2021.

Authors:  Yankai Dong; Lina Liu; Jie Han; Lianqing Zhang; Yi Wang; Juan Li; Yuexiang Li; He Liu; Kun Zhou; Luyao Li; Xin Wang; Xue Shen; Meiling Zhang; Bo Zhang; Xiaofei Hu
Journal:  Front Med (Lausanne)       Date:  2022-05-06

Review 3.  Anti-malarial drug, artemisinin and its derivatives for the treatment of respiratory diseases.

Authors:  Dorothy H J Cheong; Daniel W S Tan; Fred W S Wong; Thai Tran
Journal:  Pharmacol Res       Date:  2020-05-13       Impact factor: 7.658

Review 4.  Primaquine derivatives: Modifications of the terminal amino group.

Authors:  Branka Zorc; Ivana Perković; Kristina Pavić; Zrinka Rajić; Maja Beus
Journal:  Eur J Med Chem       Date:  2019-08-23       Impact factor: 6.514

5.  Optical Properties of Artemisinin and Its Derivatives.

Authors:  Jialin Ma; Wenhua Qiao; Xijiao Mu; Jun Dong; Jun Quan; Chunhua Tian
Journal:  ACS Omega       Date:  2020-11-23

Review 6.  Antitumor Research on Artemisinin and Its Bioactive Derivatives.

Authors:  Yunqin Zhang; Guowei Xu; Shuqun Zhang; Dong Wang; P Saravana Prabha; Zhili Zuo
Journal:  Nat Prod Bioprospect       Date:  2018-04-09

7.  Inhibition of prostate cancer cell line (PC-3) by anhydrodihydroartemisinin (ADHA) through caspase-dependent pathway.

Authors:  Faiz Ahmad; Amit Sarder; Rajesh Gour; Shibendra Kumar Lal Karna; Priya Arora; K P Ravindranathan Kartha; Yuba Raj Pokharel
Journal:  EXCLI J       Date:  2020-05-11       Impact factor: 4.068
  7 in total

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