Literature DB >> 24113254

Relationship between 17-alpha hydroxyprogesterone caproate concentration and spontaneous preterm birth.

Steve N Caritis1, Raman Venkataramanan1, Elizabeth Thom2, Margaret Harper3, Mark A Klebanoff4, Yoram Sorokin5, John M Thorp3, Michael W Varner6, Ronald J Wapner7, Jay D Iams8, Marshall W Carpenter9, William A Grobman10, Brian M Mercer11, Anthony Sciscione12, Dwight J Rouse13, Susan Ramin14.   

Abstract

OBJECTIVE: 17-alpha hydroxyprogesterone caproate 250 mg weekly reduces recurrent spontaneous preterm birth in women with a prior spontaneous preterm birth by 33%. The dose is not based on pharmacologic considerations. A therapeutic concentration has not been determined hampering any attempt to optimize treatment. This study evaluated the relationship between 17-alpha hydroxyprogesterone caproate plasma concentrations and the rate of spontaneous preterm birth in women with singleton gestation. STUDY
DESIGN: A single blood sample was obtained between 25 and 28 weeks' gestation from 315 women with a spontaneous preterm birth who participated in a placebo-controlled, prospective, randomized clinical trial evaluating the benefit of omega-3 supplementation in reducing preterm birth. All women in the parent study received 17-alpha hydroxyprogesterone caproate and 434 received omega-3 supplementation and 418 received a placebo. Plasma from 315 consenting women was analyzed for 17-alpha hydroxyprogesterone caproate concentration.
RESULTS: There were no differences between placebo and omega-3 supplemented groups in demographic variables, outcomes or in mean 17-alpha hydroxyprogesterone caproate concentration. Plasma concentrations of 17-alpha hydroxyprogesterone caproate ranged from 3.7-56 ng/mL. Women with plasma concentrations of 17-alpha hydroxyprogesterone caproate in the lowest quartile had a significantly higher risk of spontaneous preterm birth (P = .03) and delivered at significantly earlier gestational ages (P = .002) than did women in the second to fourth quartiles. The lowest preterm birth rates were seen when median 17-alpha hydroxyprogesterone caproate concentrations exceeded 6.4 ng/mL.
CONCLUSION: Low plasma 17-alpha hydroxyprogesterone caproate concentration is associated with an increased risk of spontaneous preterm birth. This finding validates efficacy of this treatment but suggests that additional studies are needed to determine the optimal dosage.
Copyright © 2014 Mosby, Inc. All rights reserved.

Entities:  

Keywords:  17-hydroxyprogesterone caproate concentration-response; dose response; pharmacodynamics

Mesh:

Substances:

Year:  2013        PMID: 24113254      PMCID: PMC3926421          DOI: 10.1016/j.ajog.2013.10.008

Source DB:  PubMed          Journal:  Am J Obstet Gynecol        ISSN: 0002-9378            Impact factor:   8.661


  18 in total

1.  ACOG Committee Opinion number 419 October 2008 (replaces no. 291, November 2003). Use of progesterone to reduce preterm birth.

Authors: 
Journal:  Obstet Gynecol       Date:  2008-10       Impact factor: 7.661

2.  Progestogen administration in pregnancy may prevent preterm delivery.

Authors:  M J Keirse
Journal:  Br J Obstet Gynaecol       Date:  1990-02

3.  Prevention of preterm delivery by 17 alpha-hydroxyprogesterone caproate in asymptomatic twin pregnancies with a short cervix: a randomized controlled trial.

Authors:  Marie-Victoire Senat; Raphael Porcher; Norbert Winer; Christophe Vayssière; Philippe Deruelle; Marianne Capelle; Florence Bretelle; Frank Perrotin; Yves Laurent; Laure Connan; Bruno Langer; Aymeric Mantel; Shohreh Azimi; Patrick Rozenberg
Journal:  Am J Obstet Gynecol       Date:  2013-03       Impact factor: 8.661

4.  Inefficacy of 17 alpha-hydroxyprogesterone caproate in the prevention of prematurity in twin pregnancy.

Authors:  A L Hartikainen-Sorri; A Kauppila; R Tuimala
Journal:  Obstet Gynecol       Date:  1980-12       Impact factor: 7.661

5.  Relationship between mirtazapine dose, plasma concentration, response, and side effects in clinical practice.

Authors:  K Grasmäder; P L Verwohlt; K-U Kühn; C Frahnert; C Hiemke; A Dragicevic; O von Widdern; A Zobel; W Maier; M L Rao
Journal:  Pharmacopsychiatry       Date:  2005-05       Impact factor: 5.788

Review 6.  Antipsychotic dosing strategies in acute schizophrenia.

Authors:  P G Janicak; J M Davis
Journal:  Int Clin Psychopharmacol       Date:  1996-05       Impact factor: 1.659

7.  Prevention of premature labor by 17 alpha-hydroxyprogesterone caproate.

Authors:  M Yemini; R Borenstein; E Dreazen; Z Apelman; B M Mogilner; I Kessler; M Lancet
Journal:  Am J Obstet Gynecol       Date:  1985-03-01       Impact factor: 8.661

8.  Cervical length changes during preterm cervical ripening: effects of 17-alpha-hydroxyprogesterone caproate.

Authors:  Fabio Facchinetti; Simone Paganelli; Giuseppina Comitini; Giulia Dante; Annibale Volpe
Journal:  Am J Obstet Gynecol       Date:  2007-05       Impact factor: 8.661

9.  Cimetidine plasma concentration-response relationships.

Authors:  R Gugler; G Fuchs; M Dieckmann; A A Somogyi
Journal:  Clin Pharmacol Ther       Date:  1981-06       Impact factor: 6.875

10.  Prevention of recurrent preterm delivery by 17 alpha-hydroxyprogesterone caproate.

Authors:  Paul J Meis; Mark Klebanoff; Elizabeth Thom; Mitchell P Dombrowski; Baha Sibai; Atef H Moawad; Catherine Y Spong; John C Hauth; Menachem Miodovnik; Michael W Varner; Kenneth J Leveno; Steve N Caritis; Jay D Iams; Ronald J Wapner; Deborah Conway; Mary J O'Sullivan; Marshall Carpenter; Brian Mercer; Susan M Ramin; John M Thorp; Alan M Peaceman; Steven Gabbe
Journal:  N Engl J Med       Date:  2003-06-12       Impact factor: 91.245

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  18 in total

1.  Does 17-alpha hydroxyprogesterone caproate prevent recurrent preterm birth in obese women?

Authors:  Kent D Heyborne; Amanda A Allshouse; J Christopher Carey
Journal:  Am J Obstet Gynecol       Date:  2015-08-12       Impact factor: 8.661

2.  Route of administration and formulation dependent pharmacokinetics of 17-hydroxyprogesterone caproate in rats.

Authors:  Imam H Shaik; Jaime R Bastian; Yang Zhao; Steve N Caritis; Raman Venkataramanan
Journal:  Xenobiotica       Date:  2015-07-07       Impact factor: 1.908

Review 3.  What we have learned about the role of 17-alpha-hydroxyprogesterone caproate in the prevention of preterm birth.

Authors:  Steve N Caritis; Maisa N Feghali; William A Grobman; Dwight J Rouse
Journal:  Semin Perinatol       Date:  2016-04-19       Impact factor: 3.300

Review 4.  Prevention of preterm delivery with 17-hydroxyprogesterone caproate: pharmacologic considerations.

Authors:  Maisa Feghali; Raman Venkataramanan; Steve Caritis
Journal:  Semin Perinatol       Date:  2014-09-23       Impact factor: 3.300

5.  Impact of Pregnancy History and 17-Hydroxyprogesterone Caproate on Cervical Cytokines and Matrix Metalloproteinases.

Authors:  Steve N Caritis; Gary Hankins; Mary Hebert; David M Haas; Mahmoud Ahmed; Hyagriv Simhan; Laura A Haneline; John Harris; Justine Chang; Alyssa Stephenson Famy; Patrick Yorio; Zhaoxia Ren; Mary E D'Alton; Raman Venkataramanan
Journal:  Am J Perinatol       Date:  2017-11-15       Impact factor: 1.862

6.  The association among cytochrome P450 3A, progesterone receptor polymorphisms, plasma 17-alpha hydroxyprogesterone caproate concentrations, and spontaneous preterm birth.

Authors:  Martha L Bustos; Steve N Caritis; Kathleen A Jablonski; Uma M Reddy; Yoram Sorokin; Tracy Manuck; Michael W Varner; Ronald J Wapner; Jay D Iams; Marshall W Carpenter; Alan M Peaceman; Brian M Mercer; Anthony Sciscione; Dwight J Rouse; Susan M Ramin
Journal:  Am J Obstet Gynecol       Date:  2017-05-15       Impact factor: 8.661

7.  17-alpha Hydroxyprogesterone caproate did not reduce the rate of recurrent preterm birth in a prospective cohort study.

Authors:  David B Nelson; Donald D McIntire; Jeffrey McDonald; John Gard; Paula Turrichi; Kenneth J Leveno
Journal:  Am J Obstet Gynecol       Date:  2017-02-20       Impact factor: 8.661

8.  Smoking, 17 Alpha-Hydroxyprogesterone Caproate, and Preterm Birth.

Authors:  Kent D Heyborne; Amanda A Allshouse
Journal:  Am J Perinatol       Date:  2016-07-27       Impact factor: 1.862

9.  Population pharmacokinetics of 17α-hydroxyprogesterone caproate in singleton gestation.

Authors:  Shringi Sharma; Steve Caritis; Gary Hankins; Menachem Miodovnik; Mary F Hebert; Don Mattison; Raman Venkataramanan
Journal:  Br J Clin Pharmacol       Date:  2016-07-13       Impact factor: 4.335

10.  Epigenetic Regulation of the Nitric Oxide Pathway, 17-α Hydroxyprogesterone Caproate, and Recurrent Preterm Birth.

Authors:  Tracy A Manuck; Lisa Smeester; Elizabeth M Martin; Martha S Tomlinson; Christina Smith; Michael W Varner; Rebecca C Fry
Journal:  Am J Perinatol       Date:  2017-12-14       Impact factor: 1.862

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