Literature DB >> 24005767

Monosubstituted alkenyl amino acids for peptide "stapling".

David J Yeo1, Stuart L Warriner, Andrew J Wilson.   

Abstract

Alkenylglycine amino acids were assessed as potential candidates for hydrocarbon stapling and shown to be effective in stapling of the BID BH3 peptide.

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Year:  2013        PMID： 24005767     DOI： 10.1039/c3cc45231j

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  14 in total

1.  A new strategy for the in vitro selection of stapled peptide inhibitors by mRNA display.

Authors:  Emil S Iqbal; Stacie L Richardson; Nicolas A Abrigo; Kara K Dods; H Estheban Osorio Franco; Heather S Gerrish; Hari Kiran Kotapati; Iain M Morgan; Douglas S Masterson; Matthew C T Hartman
Journal:  Chem Commun (Camb)       Date:  2019-07-10       Impact factor: 6.222

2.  Convergent diversity-oriented side-chain macrocyclization scan for unprotected polypeptides.

Authors:  Yekui Zou; Alexander M Spokoyny; Chi Zhang; Mark D Simon; Hongtao Yu; Yu-Shan Lin; Bradley L Pentelute
Journal:  Org Biomol Chem       Date:  2014-01-28       Impact factor: 3.876

3.  The role of olefin geometry in the activity of hydrocarbon stapled peptides targeting eukaryotic translation initiation factor 4E (eIF4E).

Authors:  James M Song; Erin E Gallagher; Arya Menon; Lauren D Mishra; Amanda L Garner
Journal:  Org Biomol Chem       Date:  2019-06-19       Impact factor: 3.876

4.  Discovery of an Orally Bioavailable Small-Molecule Inhibitor for the β-Catenin/B-Cell Lymphoma 9 Protein-Protein Interaction.

Authors:  Zhen Wang; Min Zhang; Victor Quereda; Sylvia M Frydman; Qianqian Ming; Vincent C Luca; Derek R Duckett; Haitao Ji
Journal:  J Med Chem       Date:  2021-08-12       Impact factor: 8.039

Review 5.  Structure-Based Design of Inhibitors of Protein-Protein Interactions: Mimicking Peptide Binding Epitopes.

Authors:  Marta Pelay-Gimeno; Adrian Glas; Oliver Koch; Tom N Grossmann
Journal:  Angew Chem Int Ed Engl       Date:  2015-06-26       Impact factor: 15.336

6.  Orthogonal functionalisation of α-helix mimetics.

Authors:  Anna Barnard; Kérya Long; David J Yeo; Jennifer A Miles; Valeria Azzarito; George M Burslem; Panchami Prabhakaran; Thomas A Edwards; Andrew J Wilson
Journal:  Org Biomol Chem       Date:  2014-09-21       Impact factor: 3.876

7.  Stereocontrolled protein surface recognition using chiral oligoamide proteomimetic foldamers.

Authors:  Valeria Azzarito; Jennifer A Miles; Julie Fisher; Thomas A Edwards; Stuart L Warriner; Andrew J Wilson
Journal:  Chem Sci       Date:  2015-01-30       Impact factor: 9.825

8.  Double quick, double click reversible peptide "stapling".

Authors:  Claire M Grison; George M Burslem; Jennifer A Miles; Ludwig K A Pilsl; David J Yeo; Zeynab Imani; Stuart L Warriner; Michael E Webb; Andrew J Wilson
Journal:  Chem Sci       Date:  2017-05-31       Impact factor: 9.825

9.  Synthesis of 2-aminosuberic acid derivatives as components of some histone deacetylase inhibiting cyclic tetrapeptides.

Authors:  Shital Kumar Chattopadhyay; Suman Sil; Jyoti Prasad Mukherjee
Journal:  Beilstein J Org Chem       Date:  2017-10-17       Impact factor: 2.883

10.  Hydrocarbon constrained peptides - understanding preorganisation and binding affinity.

Authors:  Jennifer A Miles; David J Yeo; Philip Rowell; Silvia Rodriguez-Marin; Christopher M Pask; Stuart L Warriner; Thomas A Edwards; Andrew J Wilson
Journal:  Chem Sci       Date:  2016-02-29       Impact factor: 9.825
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