Literature DB >> 23535705

Development of a (11)C-labeled tetrazine for rapid tetrazine-trans-cyclooctene ligation.

Matthias M Herth1, Valdemar L Andersen, Szabolcs Lehel, Jacob Madsen, Gitte M Knudsen, Jesper L Kristensen.   

Abstract

Tetrazine-trans-cyclooctene ligations are remarkably fast and selective reactions even at low micro-molar concentrations. In bioorthogonal radiochemistry, tools that enable conjugation of radioactive probes to pre-targeted vectors are of great interest. Herein, we describe the successful development of the first (11)C-labelled tetrazine and its reaction with trans-cyclooctenol.

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Year:  2013        PMID： 23535705     DOI： 10.1039/c3cc41027g

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  28 in total

Review 1.  Click Reaction: An Applicable Radiolabeling Method for Molecular Imaging.

Authors:  Ji Young Choi; Byung Chul Lee
Journal:  Nucl Med Mol Imaging       Date:  2015-10-19

Review 2.  Expanding room for tetrazine ligations in the in vivo chemistry toolbox.

Authors:  Jolita Sečkutė; Neal K Devaraj
Journal:  Curr Opin Chem Biol       Date:  2013-09-07       Impact factor: 8.822

3.  Preparation and Evaluation of 99mTc-labeled Tridentate Chelates for Pre-targeting Using Bioorthogonal Chemistry.

Authors:  Holly A Bilton; Zainab Ahmad; Nancy Janzen; Shannon Czorny; John F Valliant
Journal:  J Vis Exp       Date:  2017-02-04       Impact factor: 1.355

4.  AlCl₃-Catalyzed Ring Expansion Cascades of Bicyclic Cyclobutenamides Involving Highly Strained Cis,Trans-Cycloheptadienone Intermediates.

Authors:  Xiao-Na Wang; Elizabeth H Krenske; Ryne C Johnston; K N Houk; Richard P Hsung
Journal:  J Am Chem Soc       Date:  2015-04-20       Impact factor: 15.419

5.  An efficient and mild oxidant for the synthesis of s-tetrazines.

Authors:  Ramajeyam Selvaraj; Joseph M Fox
Journal:  Tetrahedron Lett       Date:  2014       Impact factor: 2.415

Review 6.  Click Chemistry and Radiochemistry: The First 10 Years.

Authors:  Jan-Philip Meyer; Pierre Adumeau; Jason S Lewis; Brian M Zeglis
Journal:  Bioconjug Chem       Date:  2016-11-22       Impact factor: 4.774

7.  Improved metabolic stability for 18F PET probes rapidly constructed via tetrazine trans-cyclooctene ligation.

Authors:  Ramajeyam Selvaraj; Benjamin Giglio; Shuanglong Liu; Hui Wang; Mengzhe Wang; Hong Yuan; Srinivasa R Chintala; Li-Peng Yap; Peter S Conti; Joseph M Fox; Zibo Li
Journal:  Bioconjug Chem       Date:  2015-03-04       Impact factor: 4.774

Review 8.  The inverse electron demand Diels-Alder click reaction in radiochemistry.

Authors:  Thomas Reiner; Brian M Zeglis
Journal:  J Labelled Comp Radiopharm       Date:  2013-12-18       Impact factor: 1.921

9.  A New Highly Reactive and Low Lipophilicity Fluorine-18 Labeled Tetrazine Derivative for Pretargeted PET Imaging.

Authors:  Outi Keinänen; Xiang-Guo Li; Naveen K Chenna; Dave Lumen; Jennifer Ott; Carla F M Molthoff; Mirkka Sarparanta; Kerttuli Helariutta; Tapani Vuorinen; Albert D Windhorst; Anu J Airaksinen
Journal:  ACS Med Chem Lett       Date:  2015-12-10       Impact factor: 4.345

10.  Dendrimer Scaffold for the Amplification of In Vivo Pretargeting Ligations.

Authors:  Brendon E Cook; Rosemery Membreno; Brian M Zeglis
Journal:  Bioconjug Chem       Date:  2018-07-18       Impact factor: 4.774
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