Literature DB >> 26550044

Click Reaction: An Applicable Radiolabeling Method for Molecular Imaging.

Ji Young Choi1, Byung Chul Lee2.   

Abstract

In recent years, the click reaction has found rapidly growing applications in the field of radiochemistry, ranging from a practical labeling method to molecular imaging of biomacromolecules. This present review details the development of highly reliable, powerful and selective click chemistry reactions for the rapid synthesis of new radiotracers for molecular imaging.

Keywords:  18F; Click reaction; CuAAC; Molecular imaging; Pretargeting

Year:  2015        PMID： 26550044      PMCID： PMC4630337          DOI： 10.1007/s13139-015-0377-6

Source DB:  PubMed          Journal:  Nucl Med Mol Imaging        ISSN： 1869-3474


  49 in total

1.  Strain-promoted copper-free "click" chemistry for 18F radiolabeling of bombesin.

Authors:  Lachlan S Campbell-Verduyn; Leila Mirfeizi; Anne K Schoonen; Rudi A Dierckx; Philip H Elsinga; Ben L Feringa
Journal:  Angew Chem Int Ed Engl       Date:  2011-09-28       Impact factor: 15.336

2.  In vivo chemistry for pretargeted tumor imaging in live mice.

Authors:  Raffaella Rossin; Pascal Renart Verkerk; Sandra M van den Bosch; Roland C M Vulders; Iris Verel; Johan Lub; Marc S Robillard
Journal:  Angew Chem Int Ed Engl       Date:  2010-04-26       Impact factor: 15.336

3.  F-18 labeling protocol of peptides based on chemically orthogonal strain-promoted cycloaddition under physiologically friendly reaction conditions.

Authors:  Kalme Sachin; Vinod H Jadhav; Eun-Mi Kim; Hye Lan Kim; Sang Bong Lee; Hwan-Jeong Jeong; Seok Tae Lim; Myung-Hee Sohn; Dong Wook Kim
Journal:  Bioconjug Chem       Date:  2012-07-23       Impact factor: 4.774

4.  Labeling of an antisense oligonucleotide with [(18)F]FPy5yne.

Authors:  James A H Inkster; Michael J Adam; Tim Storr; Thomas J Ruth
Journal:  Nucleosides Nucleotides Nucleic Acids       Date:  2009-11       Impact factor: 1.381

5.  General method for labeling siRNA by click chemistry with fluorine-18 for the purpose of PET imaging.

Authors:  Frédéric Mercier; Jérôme Paris; Geoffroy Kaisin; David Thonon; Jessica Flagothier; Nathalie Teller; Christian Lemaire; André Luxen
Journal:  Bioconjug Chem       Date:  2010-12-21       Impact factor: 4.774

6.  Development of a new epidermal growth factor receptor positron emission tomography imaging agent based on the 3-cyanoquinoline core: synthesis and biological evaluation.

Authors:  Federica Pisaneschi; Quang-De Nguyen; Elham Shamsaei; Matthias Glaser; Edward Robins; Maciej Kaliszczak; Graham Smith; Alan C Spivey; Eric O Aboagye
Journal:  Bioorg Med Chem       Date:  2010-08-06       Impact factor: 3.641

7.  (18)F-glyco-RGD peptides for PET imaging of integrin expression: efficient radiosynthesis by click chemistry and modulation of biodistribution by glycosylation.

Authors:  Simone Maschauer; Roland Haubner; Torsten Kuwert; Olaf Prante
Journal:  Mol Pharm       Date:  2013-12-16       Impact factor: 4.939

8.  Fully automated radiosynthesis of [1-(2-[18 F]fluoroethyl),1H[1,2,3]triazole 4-ethylene] triphenylphosphonium bromide as a potential positron emission tomography tracer for imaging apoptosis.

Authors:  Anna Haslop; Antony Gee; Christophe Plisson; Nicholas Long
Journal:  J Labelled Comp Radiopharm       Date:  2013-01-30       Impact factor: 1.921

9.  A fully automated two-step synthesis of an (18)F-labelled tyrosine kinase inhibitor for EGFR kinase activity imaging in tumors.

Authors:  D Kobus; Y Giesen; R Ullrich; H Backes; B Neumaier
Journal:  Appl Radiat Isot       Date:  2009-08-03       Impact factor: 1.513

10.  Methods for 18F-labeling of RGD peptides: comparison of aminooxy [18F]fluorobenzaldehyde condensation with 'click labeling' using 2-[18F]fluoroethylazide, and S-alkylation with [18F]fluoropropanethiol.

Authors:  Matthias Glaser; Magne Solbakken; David R Turton; Roger Pettitt; Jon Barnett; Joseph Arukwe; Hege Karlsen; Alan Cuthbertson; Sajinder K Luthra; Erik Arstad
Journal:  Amino Acids       Date:  2008-11-15       Impact factor: 3.520
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  4 in total

1.  Automated, Resin-Based Method to Enhance the Specific Activity of Fluorine-18 Clicked PET Radiotracers.

Authors:  Federica Pisaneschi; Lindsay E Kelderhouse; Amanda Hardy; Brian J Engel; Uday Mukhopadhyay; Carlos Gonzalez-Lepera; Joshua P Gray; Argentina Ornelas; Terry T Takahashi; Richard W Roberts; Stephen V Fiacco; David Piwnica-Worms; Steven W Millward
Journal:  Bioconjug Chem       Date:  2017-02-02       Impact factor: 4.774

Review 2.  Radio-graphene in Theranostic Perspectives.

Authors:  Do Won Hwang
Journal:  Nucl Med Mol Imaging       Date:  2016-03-18

3.  Mechanistic Insights into the Reaction of Amidines with 1,2,3-Triazines and 1,2,3,5-Tetrazines.

Authors:  Zhi-Chen Wu; K N Houk; Dale L Boger; Dennis Svatunek
Journal:  J Am Chem Soc       Date:  2022-06-06       Impact factor: 16.383

4.  Peptide ligands for targeting the extracellular domain of EGFR: Comparison between linear and cyclic peptides.

Authors:  Tyrslai M Williams; Rushikesh Sable; Sitanshu Singh; Maria Graca H Vicente; Seetharama D Jois
Journal:  Chem Biol Drug Des       Date:  2017-11-16       Impact factor: 2.817
  4 in total

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